JP5608746B2 - 薬物誤用に対する新規の医薬製剤 - Google Patents

薬物誤用に対する新規の医薬製剤 Download PDF

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Publication number
JP5608746B2
JP5608746B2 JP2012524263A JP2012524263A JP5608746B2 JP 5608746 B2 JP5608746 B2 JP 5608746B2 JP 2012524263 A JP2012524263 A JP 2012524263A JP 2012524263 A JP2012524263 A JP 2012524263A JP 5608746 B2 JP5608746 B2 JP 5608746B2
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granule
granules
active ingredient
core
granule according
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Japanese (ja)
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JP2013501763A (ja
JP2013501763A5 (enExample
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スュプリ、パスカル
ルボン、クリストフ
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Debregeas Et Associes Pharma SAS
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Debregeas Et Associes Pharma SAS
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2012524263A 2009-08-12 2010-08-11 薬物誤用に対する新規の医薬製剤 Expired - Fee Related JP5608746B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0955642A FR2949062B1 (fr) 2009-08-12 2009-08-12 Nouvelles formulations pharmaceutiques contre le mesusage des medicaments
FR0955642 2009-08-12
PCT/FR2010/051697 WO2011018583A2 (fr) 2009-08-12 2010-08-11 Nouvelles formulations pharmaceutiques contre le mésusage des médicaments

Publications (3)

Publication Number Publication Date
JP2013501763A JP2013501763A (ja) 2013-01-17
JP2013501763A5 JP2013501763A5 (enExample) 2014-06-05
JP5608746B2 true JP5608746B2 (ja) 2014-10-15

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JP2012524263A Expired - Fee Related JP5608746B2 (ja) 2009-08-12 2010-08-11 薬物誤用に対する新規の医薬製剤

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Country Link
US (1) US8999392B2 (enExample)
EP (1) EP2464342B1 (enExample)
JP (1) JP5608746B2 (enExample)
KR (1) KR101450974B1 (enExample)
CN (1) CN102573801B (enExample)
AR (1) AR077865A1 (enExample)
AU (1) AU2010283609B2 (enExample)
BR (1) BR112012003286B1 (enExample)
CA (1) CA2771054C (enExample)
CL (1) CL2012000377A1 (enExample)
CY (1) CY1115195T1 (enExample)
DK (1) DK2464342T3 (enExample)
EA (1) EA021856B1 (enExample)
ES (1) ES2465523T3 (enExample)
FR (1) FR2949062B1 (enExample)
HR (1) HRP20140452T1 (enExample)
IL (1) IL218071A (enExample)
IN (1) IN2012DN01859A (enExample)
MA (1) MA33522B1 (enExample)
MX (1) MX2012001879A (enExample)
NZ (1) NZ598471A (enExample)
PE (1) PE20120916A1 (enExample)
PL (1) PL2464342T3 (enExample)
PT (1) PT2464342E (enExample)
SG (1) SG180306A1 (enExample)
SI (1) SI2464342T1 (enExample)
SM (1) SMT201400076B (enExample)
TN (1) TN2012000069A1 (enExample)
TW (1) TWI465261B (enExample)
UA (1) UA104902C2 (enExample)
WO (1) WO2011018583A2 (enExample)
ZA (1) ZA201201712B (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2938431B1 (fr) 2008-11-14 2013-12-20 Debregeas Et Associes Pharma Nouvelle composition a base d'acide gamma-hydroxybutyrique
EP2405754A4 (en) * 2009-03-09 2015-10-14 Relmada Therapeutics Inc PHARMACEUTICAL BUPRENORPHINE COMPOSITIONS WITH MODIFIED RELEASE
FR2949061B1 (fr) 2009-08-12 2013-04-19 Debregeas Et Associes Pharma Microgranules flottants
US9125867B2 (en) * 2010-02-24 2015-09-08 Invincible Biotechnology Diversion- and/or abuse-resistant compositions and methods for making the same
FR2968992B1 (fr) * 2010-12-16 2013-02-08 Sanofi Aventis Comprime pharmaceutique orodispersible a base de zolpidem
FR2971422B1 (fr) * 2011-02-11 2016-05-20 Debregeas Et Associes Pharma Granules d'acide gamma-hydroxybutyrique
US9173941B1 (en) 2012-08-02 2015-11-03 Jeff Shear Sustained release bittering composition
WO2015065547A1 (en) 2013-10-31 2015-05-07 Cima Labs Inc. Immediate release abuse-deterrent granulated dosage forms
US11504347B1 (en) 2016-07-22 2022-11-22 Flamel Ireland Limited Modified release gamma-hydroxybutyrate formulations having improved pharmacokinetics
US11602512B1 (en) 2016-07-22 2023-03-14 Flamel Ireland Limited Modified release gamma-hydroxybutyrate formulations having improved pharmacokinetics
US11000498B2 (en) 2016-07-22 2021-05-11 Flamel Ireland Limited Modified release gamma-hydroxybutyrate formulations having improved pharmacokinetics
UY37341A (es) 2016-07-22 2017-11-30 Flamel Ireland Ltd Formulaciones de gamma-hidroxibutirato de liberación modificada con farmacocinética mejorada
US12186296B1 (en) 2016-07-22 2025-01-07 Flamel Ireland Limited Modified release gamma-hydroxybutyrate formulations having improved pharmacokinetics
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WO2011018583A3 (fr) 2011-04-07
PE20120916A1 (es) 2012-08-08
ES2465523T3 (es) 2014-06-06
FR2949062A1 (fr) 2011-02-18
CY1115195T1 (el) 2017-01-04
CL2012000377A1 (es) 2012-12-07
IL218071A (en) 2015-10-29
AR077865A1 (es) 2011-09-28
SMT201400076B (it) 2014-09-08
SI2464342T1 (sl) 2014-07-31
HK1172845A1 (en) 2013-05-03
EP2464342A2 (fr) 2012-06-20
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IL218071A0 (en) 2012-04-30
BR112012003286A2 (pt) 2016-03-01
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US8999392B2 (en) 2015-04-07
US20120164228A1 (en) 2012-06-28
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EP2464342B1 (fr) 2014-02-26
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CN102573801A (zh) 2012-07-11
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BR112012003286B1 (pt) 2021-12-07
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