JP5389013B2 - 抗菌剤としての三環式含窒素化合物 - Google Patents

抗菌剤としての三環式含窒素化合物 Download PDF

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Publication number
JP5389013B2
JP5389013B2 JP2010503491A JP2010503491A JP5389013B2 JP 5389013 B2 JP5389013 B2 JP 5389013B2 JP 2010503491 A JP2010503491 A JP 2010503491A JP 2010503491 A JP2010503491 A JP 2010503491A JP 5389013 B2 JP5389013 B2 JP 5389013B2
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Japan
Prior art keywords
dihydro
methyl
amino
piperidinyl
dione
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Active
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JP2010503491A
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English (en)
Japanese (ja)
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JP2010524884A5 (cg-RX-API-DMAC7.html
JP2010524884A (ja
Inventor
デイビッド・エバン・デイビーズ
デイビッド・トーマス・デイビーズ
イラリア・ジョルダーノ
アラン・ジョゼフ・ヘネシー
ニール・デイビッド・ピアソン
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Glaxo Group Ltd
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Glaxo Group Ltd
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Priority claimed from GB0707705A external-priority patent/GB0707705D0/en
Priority claimed from GB0720569A external-priority patent/GB0720569D0/en
Priority claimed from GB0805311A external-priority patent/GB0805311D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of JP2010524884A publication Critical patent/JP2010524884A/ja
Publication of JP2010524884A5 publication Critical patent/JP2010524884A5/ja
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
JP2010503491A 2007-04-20 2008-04-16 抗菌剤としての三環式含窒素化合物 Active JP5389013B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GB0707705A GB0707705D0 (en) 2007-04-20 2007-04-20 Compounds
GB0707705.0 2007-04-20
GB0720569A GB0720569D0 (en) 2007-10-19 2007-10-19 Compounds
GB0720569.3 2007-10-19
GB0805311.8 2008-03-20
GB0805311A GB0805311D0 (en) 2008-03-20 2008-03-20 Compounds
PCT/EP2008/054621 WO2008128942A1 (en) 2007-04-20 2008-04-16 Tricyclic nitrogen containing compounds as antibacterial agents

Publications (3)

Publication Number Publication Date
JP2010524884A JP2010524884A (ja) 2010-07-22
JP2010524884A5 JP2010524884A5 (cg-RX-API-DMAC7.html) 2011-06-02
JP5389013B2 true JP5389013B2 (ja) 2014-01-15

Family

ID=39580226

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010503491A Active JP5389013B2 (ja) 2007-04-20 2008-04-16 抗菌剤としての三環式含窒素化合物

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US (1) US8389524B2 (cg-RX-API-DMAC7.html)
EP (1) EP2137196B1 (cg-RX-API-DMAC7.html)
JP (1) JP5389013B2 (cg-RX-API-DMAC7.html)
KR (1) KR101567096B1 (cg-RX-API-DMAC7.html)
CN (1) CN101687887B (cg-RX-API-DMAC7.html)
AR (1) AR066111A1 (cg-RX-API-DMAC7.html)
AT (1) ATE483717T1 (cg-RX-API-DMAC7.html)
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BR (1) BRPI0810064B8 (cg-RX-API-DMAC7.html)
CA (1) CA2684659C (cg-RX-API-DMAC7.html)
CL (1) CL2008001122A1 (cg-RX-API-DMAC7.html)
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DO (1) DOP2009000240A (cg-RX-API-DMAC7.html)
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PE (1) PE20090274A1 (cg-RX-API-DMAC7.html)
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TW (1) TWI431006B (cg-RX-API-DMAC7.html)
UY (1) UY31038A1 (cg-RX-API-DMAC7.html)
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CN111494241B (zh) * 2020-06-01 2023-03-24 湖北洁世达环保科技有限公司 一种纸巾柔润保湿液
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Publication number Publication date
TW200848420A (en) 2008-12-16
KR101567096B1 (ko) 2015-11-06
AU2008240764B2 (en) 2011-04-07
HRP20100574T1 (hr) 2010-12-31
DOP2009000240A (es) 2009-12-31
AR066111A1 (es) 2009-07-22
ATE483717T1 (de) 2010-10-15
UY31038A1 (es) 2008-11-28
PL2137196T3 (pl) 2011-03-31
US20100137282A1 (en) 2010-06-03
NZ579877A (en) 2011-09-30
EA015821B1 (ru) 2011-12-30
CN101687887A (zh) 2010-03-31
DK2137196T3 (da) 2011-01-10
CN101687887B (zh) 2012-08-29
MX2009011317A (es) 2009-11-05
CA2684659A1 (en) 2008-10-30
US8389524B2 (en) 2013-03-05
WO2008128942A1 (en) 2008-10-30
JP2010524884A (ja) 2010-07-22
BRPI0810064A2 (pt) 2019-08-27
EP2137196B1 (en) 2010-10-06
CR11123A (es) 2010-03-08
BRPI0810064B1 (pt) 2021-03-30
CY1111248T1 (el) 2015-06-11
CL2008001122A1 (es) 2008-10-24
SI2137196T1 (sl) 2011-01-31
TWI431006B (zh) 2014-03-21
CO6251368A2 (es) 2011-02-21
HK1138000A1 (en) 2010-08-13
MY149347A (en) 2013-08-30
MA31324B1 (fr) 2010-04-01
IL201204A0 (en) 2010-05-17
PT2137196E (pt) 2010-12-16
CA2684659C (en) 2015-11-24
BRPI0810064B8 (pt) 2021-05-25
EP2137196A1 (en) 2009-12-30
CR20150586A (es) 2016-04-04
KR20100017133A (ko) 2010-02-16
EA200970987A1 (ru) 2010-04-30
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