AU2002219175A1 - Crystalline forms of cerivastatin sodium - Google Patents
Crystalline forms of cerivastatin sodiumInfo
- Publication number
- AU2002219175A1 AU2002219175A1 AU2002219175A AU1917502A AU2002219175A1 AU 2002219175 A1 AU2002219175 A1 AU 2002219175A1 AU 2002219175 A AU2002219175 A AU 2002219175A AU 1917502 A AU1917502 A AU 1917502A AU 2002219175 A1 AU2002219175 A1 AU 2002219175A1
- Authority
- AU
- Australia
- Prior art keywords
- crystalline forms
- cerivastatin sodium
- cerivastatin
- sodium
- crystalline
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- GPUADMRJQVPIAS-QCVDVZFFSA-M cerivastatin sodium Chemical compound [Na+].COCC1=C(C(C)C)N=C(C(C)C)C(\C=C\[C@@H](O)C[C@@H](O)CC([O-])=O)=C1C1=CC=C(F)C=C1 GPUADMRJQVPIAS-QCVDVZFFSA-M 0.000 title 1
- 229940052311 cerivastatin sodium Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/55—Acids; Esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pyridine Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP00811225 | 2000-12-21 | ||
EP00811225 | 2000-12-21 | ||
PCT/EP2001/014602 WO2002050036A1 (en) | 2000-12-21 | 2001-12-12 | Crystalline forms of cerivastatin sodium |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2002219175A1 true AU2002219175A1 (en) | 2002-07-01 |
Family
ID=8175095
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002219175A Abandoned AU2002219175A1 (en) | 2000-12-21 | 2001-12-12 | Crystalline forms of cerivastatin sodium |
Country Status (4)
Country | Link |
---|---|
US (1) | US20040063961A1 (en) |
EP (1) | EP1345903A1 (en) |
AU (1) | AU2002219175A1 (en) |
WO (1) | WO2002050036A1 (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2006500337A (en) * | 2002-07-26 | 2006-01-05 | チバ スペシャルティ ケミカルズ ホールディング インコーポレーテッド | Polymorphic and amorphous forms of benazepril hydrochloride |
JP5192147B2 (en) * | 2003-02-12 | 2013-05-08 | 日産化学工業株式会社 | Crystalline form of pitavastatin calcium |
EP2001887B1 (en) | 2006-04-06 | 2010-09-15 | Glaxo Group Limited | Pyrrolo-quinoxalinone derivatives as antibacterials |
EP2007377A4 (en) | 2006-04-06 | 2011-08-17 | Glaxo Group Ltd | Antibacterial agents |
EP1992628A1 (en) | 2007-05-18 | 2008-11-19 | Glaxo Group Limited | Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones |
AR065670A1 (en) | 2007-03-09 | 2009-06-24 | Indigene Pharmaceuticals Inc | COMBINATION OF METFORMIN R - (+) LIPOATE AND ANTIHIPERLIPIDEMIC AGENTS FOR THE TREATMENT OF DIABETIC HYPERGLUCEMIA AND DIABETIC COMPLICATIONS |
SI2137196T1 (en) * | 2007-04-20 | 2011-01-31 | Glaxo Group Ltd Glaxo Welcome House | Tricyclic nitrogen containing compounds as antibacterial agents |
EP2080761A1 (en) | 2008-01-18 | 2009-07-22 | Glaxo Group Limited | Compounds |
EP2352734A1 (en) | 2008-10-17 | 2011-08-10 | Glaxo Group Limited | Tricyclic nitrogen compounds used as antibacterials |
JP5653935B2 (en) | 2009-01-15 | 2015-01-14 | グラクソ グループ リミテッドGlaxo Group Limited | Naphthyridin-2 (1H) -one compounds useful as antibacterial agents |
AR101674A1 (en) | 2014-08-22 | 2017-01-04 | Glaxosmithkline Ip Dev Ltd | USE OF A TRICYCLIC COMPOUND CONTAINING NITROGEN |
TW201722965A (en) | 2015-08-16 | 2017-07-01 | 葛蘭素史密斯克藍智慧財產發展有限公司 | Compounds for use in antibacterial applications |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5177080A (en) * | 1990-12-14 | 1993-01-05 | Bayer Aktiengesellschaft | Substituted pyridyl-dihydroxy-heptenoic acid and its salts |
DE4309553A1 (en) * | 1993-03-24 | 1994-09-29 | Bayer Ag | Process for the preparation of 3R, 5S - (+) - sodium erythro- (E) -7- (4- (4-flurophenyl) -2,6-diisopropyl-5-methoxymethyl-pyrid-3-yl) -3, 5-dihydroxy-hept-6-enoate |
US6531507B1 (en) * | 2000-06-09 | 2003-03-11 | Lek Pharmaceuticals D.D. | Stabilized pharmaceutically effective composition and pharmaceutical formulation comprising the same |
-
2001
- 2001-12-12 AU AU2002219175A patent/AU2002219175A1/en not_active Abandoned
- 2001-12-12 EP EP01271357A patent/EP1345903A1/en not_active Withdrawn
- 2001-12-12 WO PCT/EP2001/014602 patent/WO2002050036A1/en not_active Application Discontinuation
- 2001-12-12 US US10/451,133 patent/US20040063961A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US20040063961A1 (en) | 2004-04-01 |
EP1345903A1 (en) | 2003-09-24 |
WO2002050036A1 (en) | 2002-06-27 |
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