JP4465048B2 - Ｎ−置換３−ヒドロキシピラゾールの製造方法 - Google Patents

Ｎ−置換３−ヒドロキシピラゾールの製造方法 Download PDF

Info

Publication number
JP4465048B2
JP4465048B2 JP52724998A JP52724998A JP4465048B2 JP 4465048 B2 JP4465048 B2 JP 4465048B2 JP 52724998 A JP52724998 A JP 52724998A JP 52724998 A JP52724998 A JP 52724998A JP 4465048 B2 JP4465048 B2 JP 4465048B2
Authority
JP
Japan
Prior art keywords
formula
process according
hydroxypyrazole
compound
oxygen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
JP52724998A
Other languages
English (en)
Japanese (ja)
Other versions
JP2001506244A (ja
Inventor
フォーゲルバッハー，ウヴェ
カイル，ミヒャエル
クリンツ，ラルフ
ヴァール，ヨーゼフ
ヴィンゲルト，ホルスト
ケーニヒ，ハルトマン
ラック，ミヒャエル
ゲツ，ローラント
テレス，ヨーアキム，ヘンリク
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Publication of JP2001506244A publication Critical patent/JP2001506244A/ja
Application granted granted Critical
Publication of JP4465048B2 publication Critical patent/JP4465048B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP52724998A 1996-12-17 1997-12-04 Ｎ−置換３−ヒドロキシピラゾールの製造方法 Expired - Fee Related JP4465048B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19652516.0 1996-12-17
DE19652516A DE19652516A1 (de) 1996-12-17 1996-12-17 Verfahren zur Herstellung von N-substituierten 3-hydroxypyrazolen
PCT/EP1997/006780 WO1998027062A1 (de) 1996-12-17 1997-12-04 Verfahren zur herstellung von n-substituierten 3-hydroxypyrazolen

Publications (2)

Publication Number Publication Date
JP2001506244A JP2001506244A (ja) 2001-05-15
JP4465048B2 true JP4465048B2 (ja) 2010-05-19

Family

ID=7815027

Family Applications (1)

Application Number Title Priority Date Filing Date
JP52724998A Expired - Fee Related JP4465048B2 (ja) 1996-12-17 1997-12-04 Ｎ−置換３−ヒドロキシピラゾールの製造方法

Country Status (25)

Country Link
US (1) US6040458A (index.php)
EP (1) EP0946514B1 (index.php)
JP (1) JP4465048B2 (index.php)
KR (1) KR100508594B1 (index.php)
CN (1) CN1098253C (index.php)
AR (1) AR008944A1 (index.php)
AT (1) ATE238994T1 (index.php)
AU (1) AU746496B2 (index.php)
BR (1) BR9713951A (index.php)
CA (1) CA2275253C (index.php)
CO (1) CO5011024A1 (index.php)
CZ (1) CZ292280B6 (index.php)
DE (2) DE19652516A1 (index.php)
DK (1) DK0946514T3 (index.php)
EA (1) EA001630B1 (index.php)
ES (1) ES2199382T3 (index.php)
HU (1) HU228235B1 (index.php)
IL (1) IL130125A (index.php)
IN (1) IN185466B (index.php)
NZ (1) NZ335953A (index.php)
PL (1) PL191331B1 (index.php)
SK (1) SK282689B6 (index.php)
UA (1) UA53678C2 (index.php)
WO (1) WO1998027062A1 (index.php)
ZA (1) ZA9711238B (index.php)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2151433A1 (en) 2008-08-05 2010-02-10 Institut Pasteur Alkoxypyrazoles and the process for their preparation
WO2011113884A1 (en) 2010-03-18 2011-09-22 Basf Se N-carbomethoxy-n-methoxy-(2-chloromethyl)-anilines, their preparation and their use as precursors for preparing 2-(pyrazol-3'-yloxymethylene)-anilides
US9744066B2 (en) 2011-06-10 2017-08-29 The Regents Of The University Of California Trunk supporting exoskeleton and method of use
US9022956B2 (en) 2011-06-10 2015-05-05 U.S. Bionics, Inc. Trunk supporting exoskeleton and method of use
EP2815647A1 (en) 2013-06-18 2014-12-24 Basf Se Novel strobilurin-type compounds for combating phytopathogenic fungi
EP3112350B1 (en) * 2014-02-28 2018-04-04 Sumitomo Chemical Company, Limited Method for producing pyrazole compound
UA124524C2 (uk) 2015-05-18 2021-10-05 Шеньян Сайнокем Аґрокемікалз Р&Д Ко., Лтд. Сполукa заміщеного піразолу, якa містить піримідиніл, її одержання і застосування
CN105061322B (zh) * 2015-07-27 2018-07-24 北京颖泰嘉和生物科技股份有限公司 N-取代的3-羟基吡唑化合物的制备方法
CN106008350A (zh) * 2016-07-21 2016-10-12 山东益丰生化环保股份有限公司 一种1-(4-氯苯基)-3-吡唑醇的制备方法
EP3541788B1 (en) * 2016-11-17 2020-09-02 Basf Se Process for the purification of 1-(4-chlorophenyl)pyrazol-3-ol
CN107778246A (zh) * 2017-12-05 2018-03-09 利民化工股份有限公司 一种杀菌剂吡唑醚菌酯中间体吡唑醇的精制方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3415385A1 (de) * 1984-04-25 1985-11-07 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von pyrazolen
UA48189C2 (uk) * 1995-07-14 2002-08-15 Басф Акцієнгезельшафт Спосіб одержання n-заміщених 3-гідроксипіразолів

Also Published As

Publication number Publication date
HUP0000554A2 (hu) 2000-06-28
WO1998027062A1 (de) 1998-06-25
EP0946514B1 (de) 2003-05-02
HU228235B1 (hu) 2013-02-28
CA2275253C (en) 2007-03-27
UA53678C2 (uk) 2003-02-17
AU746496B2 (en) 2002-05-02
NZ335953A (en) 2000-09-29
SK77699A3 (en) 2000-04-10
CZ292280B6 (cs) 2003-08-13
AR008944A1 (es) 2000-02-23
CZ214799A3 (cs) 1999-09-15
US6040458A (en) 2000-03-21
CA2275253A1 (en) 1998-06-25
CN1098253C (zh) 2003-01-08
KR100508594B1 (ko) 2005-08-17
DE19652516A1 (de) 1998-06-18
ZA9711238B (en) 1999-06-15
EA001630B1 (ru) 2001-06-25
SK282689B6 (sk) 2002-11-06
CN1240433A (zh) 2000-01-05
CO5011024A1 (es) 2001-02-28
ATE238994T1 (de) 2003-05-15
IN185466B (index.php) 2001-01-27
IL130125A (en) 2003-05-29
IL130125A0 (en) 2000-06-01
KR20000057599A (ko) 2000-09-25
HUP0000554A3 (en) 2002-01-28
EP0946514A1 (de) 1999-10-06
PL191331B1 (pl) 2006-04-28
DE59709989D1 (de) 2003-06-05
DK0946514T3 (da) 2003-08-25
JP2001506244A (ja) 2001-05-15
AU5753698A (en) 1998-07-15
BR9713951A (pt) 2000-03-21
EA199900536A1 (ru) 1999-12-29
PL333984A1 (en) 2000-01-31
ES2199382T3 (es) 2004-02-16

Similar Documents

Publication Publication Date Title
HRP20020438A2 (en) Process for preparing 4-trifluoromethylsulphinylpyrazole derivative
JP3981153B2 (ja) Ｎ−置換３−ヒドロキシピラゾールの製造方法
CN101796021A (zh) 制备吡唑的方法
JP4465048B2 (ja) Ｎ−置換３−ヒドロキシピラゾールの製造方法
JP5167283B2 (ja) フェニルトリアゾリノン類の製造法
EP0596684B1 (en) Preparation of substituted aryl compounds
US9024030B2 (en) Process for the synthesis of etoricoxib
CA2048456C (en) The preparation of 3-methylpyrazole
JPS624247A (ja) ４，４’−ジニトロジベンジル類の製造方法
JPH0680049B2 (ja) １，２，４−トリアゾ−ル−３−カルボン酸誘導体の製造方法
EP2349980B1 (en) Process for preparing 2-amino-6-nitro-benzoic acid
JPH04360879A (ja) 芳香族トリアゾール類の精製方法
JP4273271B2 (ja) ピラゾール化合物及びその製造法
US20070027211A1 (en) Process for production of bicalutamide
JPH01168674A (ja) １．３−ジアルキルピラゾール−４−カルボン酸誘導体の製造方法
JPH10175958A (ja) ２−ホルミルイミダゾール誘導体の製造法
JPH06256316A (ja) ２−ｎ−ブチル−４−イミダゾールジチオカルボン酸

Legal Events

Date Code Title Description
A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20040714

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20080507

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20080731

A72 Notification of change in name of applicant

Free format text: JAPANESE INTERMEDIATE CODE: A721

Effective date: 20080731

A602 Written permission of extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A602

Effective date: 20080908

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20080902

A602 Written permission of extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A602

Effective date: 20081010

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20081001

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20090811

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20091110

TRDD Decision of grant or rejection written
A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

Effective date: 20100126

A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

A61 First payment of annual fees (during grant procedure)

Free format text: JAPANESE INTERMEDIATE CODE: A61

Effective date: 20100222

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20130226

Year of fee payment: 3

R150 Certificate of patent or registration of utility model

Free format text: JAPANESE INTERMEDIATE CODE: R150

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20140226

Year of fee payment: 4

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

LAPS Cancellation because of no payment of annual fees