JP4149803B2 - 組成物の調製方法 - Google Patents

組成物の調製方法 Download PDF

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Publication number
JP4149803B2
JP4149803B2 JP2002504983A JP2002504983A JP4149803B2 JP 4149803 B2 JP4149803 B2 JP 4149803B2 JP 2002504983 A JP2002504983 A JP 2002504983A JP 2002504983 A JP2002504983 A JP 2002504983A JP 4149803 B2 JP4149803 B2 JP 4149803B2
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JP
Japan
Prior art keywords
weight
dispersion
solution
composition
fatty acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP2002504983A
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English (en)
Japanese (ja)
Other versions
JP2004501184A5 (https=
JP2004501184A (ja
Inventor
ブソーン，パトリック
シュローダー，マルコ
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F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
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Publication date
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Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of JP2004501184A publication Critical patent/JP2004501184A/ja
Publication of JP2004501184A5 publication Critical patent/JP2004501184A5/ja
Application granted granted Critical
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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/12—Aerosols; Foams
    • A61K9/122—Foams; Dry foams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biochemistry (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2002504983A 2000-06-27 2001-06-18 組成物の調製方法 Expired - Lifetime JP4149803B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00113535 2000-06-27
PCT/EP2001/006834 WO2002000201A2 (en) 2000-06-27 2001-06-18 Method for preparing a composition

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2007180722A Division JP2007302683A (ja) 2000-06-27 2007-07-10 組成物の調製方法

Publications (3)

Publication Number Publication Date
JP2004501184A JP2004501184A (ja) 2004-01-15
JP2004501184A5 JP2004501184A5 (https=) 2005-02-03
JP4149803B2 true JP4149803B2 (ja) 2008-09-17

Family

ID=8169074

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2002504983A Expired - Lifetime JP4149803B2 (ja) 2000-06-27 2001-06-18 組成物の調製方法
JP2007180722A Pending JP2007302683A (ja) 2000-06-27 2007-07-10 組成物の調製方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2007180722A Pending JP2007302683A (ja) 2000-06-27 2007-07-10 組成物の調製方法

Country Status (37)

Country Link
US (3) US6534087B2 (https=)
EP (1) EP1296656B1 (https=)
JP (2) JP4149803B2 (https=)
KR (1) KR100557845B1 (https=)
CN (1) CN1236764C (https=)
AR (1) AR029278A1 (https=)
AT (1) ATE334662T1 (https=)
AU (2) AU8184601A (https=)
BR (1) BRPI0112014B1 (https=)
CA (1) CA2411153C (https=)
CY (1) CY1105714T1 (https=)
CZ (1) CZ301813B6 (https=)
DE (1) DE60121953T2 (https=)
DK (1) DK1296656T3 (https=)
EC (1) ECSP024401A (https=)
EG (1) EG24141A (https=)
ES (1) ES2269441T3 (https=)
HR (1) HRP20021009B1 (https=)
HU (1) HU229550B1 (https=)
IL (2) IL153282A0 (https=)
JO (1) JO2247B1 (https=)
MA (1) MA26922A1 (https=)
ME (1) ME00672B (https=)
MX (1) MXPA02012583A (https=)
MY (1) MY129798A (https=)
NO (1) NO332181B1 (https=)
NZ (1) NZ523024A (https=)
PE (1) PE20020101A1 (https=)
PL (1) PL203804B1 (https=)
PT (1) PT1296656E (https=)
RU (1) RU2244542C2 (https=)
SI (1) SI1296656T1 (https=)
TW (1) TWI278325B (https=)
UY (1) UY26799A1 (https=)
WO (1) WO2002000201A2 (https=)
YU (1) YU96602A (https=)
ZA (1) ZA200209649B (https=)

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PL203804B1 (pl) * 2000-06-27 2009-11-30 Hoffmann La Roche Sposób wytwarzania kompozycji farmaceutycznej w postaci spoistej, płytkowej, piankowej, gąbczastej lub ciastowatej struktury i kompozycja farmaceutyczna otrzymana tym sposobem

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AU2001281846B2 (en) 2006-04-27
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