JP4053589B2 - 経口投与のための医薬的および/または栄養学的マイクロカプセル - Google Patents
経口投与のための医薬的および/または栄養学的マイクロカプセル Download PDFInfo
- Publication number
- JP4053589B2 JP4053589B2 JP51300696A JP51300696A JP4053589B2 JP 4053589 B2 JP4053589 B2 JP 4053589B2 JP 51300696 A JP51300696 A JP 51300696A JP 51300696 A JP51300696 A JP 51300696A JP 4053589 B2 JP4053589 B2 JP 4053589B2
- Authority
- JP
- Japan
- Prior art keywords
- microcapsule
- agent
- microcapsules
- weight
- coating composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
- A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR94/12759 | 1994-10-18 | ||
| FR9412759A FR2725623A1 (fr) | 1994-10-18 | 1994-10-18 | Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os |
| PCT/FR1995/001369 WO1996011675A2 (fr) | 1994-10-18 | 1995-10-18 | Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPH10509427A JPH10509427A (ja) | 1998-09-14 |
| JP4053589B2 true JP4053589B2 (ja) | 2008-02-27 |
Family
ID=9468196
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP51300696A Expired - Fee Related JP4053589B2 (ja) | 1994-10-18 | 1995-10-18 | 経口投与のための医薬的および/または栄養学的マイクロカプセル |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US6022562A (https=) |
| EP (1) | EP0709087B1 (https=) |
| JP (1) | JP4053589B2 (https=) |
| AR (1) | AR022930A2 (https=) |
| AT (1) | ATE188117T1 (https=) |
| AU (1) | AU3807795A (https=) |
| BR (2) | BRPI9509286B8 (https=) |
| CA (1) | CA2160762C (https=) |
| DE (1) | DE69514192T2 (https=) |
| ES (1) | ES2140641T3 (https=) |
| FR (1) | FR2725623A1 (https=) |
| IL (1) | IL115646A (https=) |
| WO (1) | WO1996011675A2 (https=) |
| ZA (1) | ZA958762B (https=) |
Families Citing this family (150)
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4461759A (en) * | 1983-01-03 | 1984-07-24 | Verex Laboratories, Inc. | Constant release rate solid oral dosage formulations of veropamil |
| LU85943A1 (fr) * | 1985-06-12 | 1987-01-13 | Galephar | Comprimes pharmaceutiques permettant l'administration aisee de pellets, leur preparation et leur utilisation |
| US5028434A (en) * | 1988-07-21 | 1991-07-02 | Alza Corporation | Method for administering nilvadipine for treating cardiovascular symptoms |
| IT1227899B (it) * | 1988-12-23 | 1991-05-14 | Poli Ind Chimica Spa | Rivestimento totale o parziale di principi attivi farmaceutici e relative composizioni |
| US5286497A (en) * | 1991-05-20 | 1994-02-15 | Carderm Capital L.P. | Diltiazem formulation |
-
1994
- 1994-10-18 FR FR9412759A patent/FR2725623A1/fr active Granted
-
1995
- 1995-10-17 US US08/544,208 patent/US6022562A/en not_active Expired - Lifetime
- 1995-10-17 ZA ZA958762A patent/ZA958762B/xx unknown
- 1995-10-17 IL IL11564695A patent/IL115646A/xx not_active IP Right Cessation
- 1995-10-17 CA CA002160762A patent/CA2160762C/fr not_active Expired - Fee Related
- 1995-10-18 ES ES95420286T patent/ES2140641T3/es not_active Expired - Lifetime
- 1995-10-18 AT AT95420286T patent/ATE188117T1/de not_active IP Right Cessation
- 1995-10-18 DE DE69514192T patent/DE69514192T2/de not_active Expired - Lifetime
- 1995-10-18 WO PCT/FR1995/001369 patent/WO1996011675A2/fr not_active Ceased
- 1995-10-18 BR BRPI9509286A patent/BRPI9509286B8/pt unknown
- 1995-10-18 JP JP51300696A patent/JP4053589B2/ja not_active Expired - Fee Related
- 1995-10-18 BR BR9509286A patent/BR9509286A/pt active IP Right Grant
- 1995-10-18 EP EP95420286A patent/EP0709087B1/fr not_active Expired - Lifetime
- 1995-10-18 AU AU38077/95A patent/AU3807795A/en not_active Abandoned
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2000
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Also Published As
| Publication number | Publication date |
|---|---|
| CA2160762C (fr) | 2004-12-21 |
| EP0709087B1 (fr) | 1999-12-29 |
| JPH10509427A (ja) | 1998-09-14 |
| WO1996011675A2 (fr) | 1996-04-25 |
| BR9509286A (pt) | 1997-10-14 |
| US6022562A (en) | 2000-02-08 |
| WO1996011675A3 (fr) | 1996-06-20 |
| IL115646A (en) | 2000-07-16 |
| DE69514192T2 (de) | 2000-07-13 |
| ZA958762B (en) | 1996-05-09 |
| AR022930A2 (es) | 2002-09-04 |
| FR2725623A1 (fr) | 1996-04-19 |
| EP0709087A1 (fr) | 1996-05-01 |
| IL115646A0 (en) | 1996-01-19 |
| ES2140641T3 (es) | 2000-03-01 |
| CA2160762A1 (fr) | 1996-04-19 |
| AU3807795A (en) | 1996-05-06 |
| BRPI9509286B8 (pt) | 2019-12-17 |
| ATE188117T1 (de) | 2000-01-15 |
| DE69514192D1 (de) | 2000-02-03 |
| FR2725623B1 (https=) | 1997-02-21 |
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