JP4053589B2 - 経口投与のための医薬的および／または栄養学的マイクロカプセル - Google Patents

経口投与のための医薬的および／または栄養学的マイクロカプセル Download PDF

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Publication number
JP4053589B2
JP4053589B2 JP51300696A JP51300696A JP4053589B2 JP 4053589 B2 JP4053589 B2 JP 4053589B2 JP 51300696 A JP51300696 A JP 51300696A JP 51300696 A JP51300696 A JP 51300696A JP 4053589 B2 JP4053589 B2 JP 4053589B2
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Prior art keywords
microcapsule
agent
microcapsules
weight
coating composition
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Expired - Fee Related
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JP51300696A
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English (en)
Japanese (ja)
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JPH10509427A (ja
Inventor
ピエール オータン、
ジャン − フィリップ セル、
ジェラール スーラ、
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Flamel Technologies SA
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Flamel Technologies SA
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Application filed by Flamel Technologies SA filed Critical Flamel Technologies SA
Publication of JPH10509427A publication Critical patent/JPH10509427A/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5015—Organic compounds, e.g. fats, sugars
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

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  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP51300696A 1994-10-18 1995-10-18 経口投与のための医薬的および／または栄養学的マイクロカプセル Expired - Fee Related JP4053589B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9412759A FR2725623A1 (fr) 1994-10-18 1994-10-18 Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os
FR94/12759 1994-10-18
PCT/FR1995/001369 WO1996011675A2 (fr) 1994-10-18 1995-10-18 Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os

Publications (2)

Publication Number Publication Date
JPH10509427A JPH10509427A (ja) 1998-09-14
JP4053589B2 true JP4053589B2 (ja) 2008-02-27

Family

ID=9468196

Family Applications (1)

Application Number Title Priority Date Filing Date
JP51300696A Expired - Fee Related JP4053589B2 (ja) 1994-10-18 1995-10-18 経口投与のための医薬的および／または栄養学的マイクロカプセル

Country Status (14)

Country Link
US (1) US6022562A (https=)
EP (1) EP0709087B1 (https=)
JP (1) JP4053589B2 (https=)
AR (1) AR022930A2 (https=)
AT (1) ATE188117T1 (https=)
AU (1) AU3807795A (https=)
BR (2) BR9509286A (https=)
CA (1) CA2160762C (https=)
DE (1) DE69514192T2 (https=)
ES (1) ES2140641T3 (https=)
FR (1) FR2725623A1 (https=)
IL (1) IL115646A (https=)
WO (1) WO1996011675A2 (https=)
ZA (1) ZA958762B (https=)

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AR022930A2 (es) 2002-09-04
ATE188117T1 (de) 2000-01-15
DE69514192T2 (de) 2000-07-13
WO1996011675A2 (fr) 1996-04-25
WO1996011675A3 (fr) 1996-06-20
US6022562A (en) 2000-02-08
FR2725623B1 (https=) 1997-02-21
BR9509286A (pt) 1997-10-14
ZA958762B (en) 1996-05-09
AU3807795A (en) 1996-05-06
FR2725623A1 (fr) 1996-04-19
CA2160762C (fr) 2004-12-21
JPH10509427A (ja) 1998-09-14
EP0709087A1 (fr) 1996-05-01
ES2140641T3 (es) 2000-03-01
IL115646A (en) 2000-07-16
IL115646A0 (en) 1996-01-19
EP0709087B1 (fr) 1999-12-29
BRPI9509286B8 (pt) 2019-12-17
DE69514192D1 (de) 2000-02-03
CA2160762A1 (fr) 1996-04-19

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