JP4053589B2 - 経口投与のための医薬的および/または栄養学的マイクロカプセル - Google Patents
経口投与のための医薬的および/または栄養学的マイクロカプセル Download PDFInfo
- Publication number
- JP4053589B2 JP4053589B2 JP51300696A JP51300696A JP4053589B2 JP 4053589 B2 JP4053589 B2 JP 4053589B2 JP 51300696 A JP51300696 A JP 51300696A JP 51300696 A JP51300696 A JP 51300696A JP 4053589 B2 JP4053589 B2 JP 4053589B2
- Authority
- JP
- Japan
- Prior art keywords
- microcapsule
- agent
- microcapsules
- weight
- coating composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
- A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR94/12759 | 1994-10-18 | ||
| FR9412759A FR2725623A1 (fr) | 1994-10-18 | 1994-10-18 | Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os |
| PCT/FR1995/001369 WO1996011675A2 (fr) | 1994-10-18 | 1995-10-18 | Microcapsules medicamenteuses et/ou nutritionnelles pour administration per os |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPH10509427A JPH10509427A (ja) | 1998-09-14 |
| JP4053589B2 true JP4053589B2 (ja) | 2008-02-27 |
Family
ID=9468196
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP51300696A Expired - Fee Related JP4053589B2 (ja) | 1994-10-18 | 1995-10-18 | 経口投与のための医薬的および/または栄養学的マイクロカプセル |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US6022562A (enExample) |
| EP (1) | EP0709087B1 (enExample) |
| JP (1) | JP4053589B2 (enExample) |
| AR (1) | AR022930A2 (enExample) |
| AT (1) | ATE188117T1 (enExample) |
| AU (1) | AU3807795A (enExample) |
| BR (2) | BRPI9509286B8 (enExample) |
| CA (1) | CA2160762C (enExample) |
| DE (1) | DE69514192T2 (enExample) |
| ES (1) | ES2140641T3 (enExample) |
| FR (1) | FR2725623A1 (enExample) |
| IL (1) | IL115646A (enExample) |
| WO (1) | WO1996011675A2 (enExample) |
| ZA (1) | ZA958762B (enExample) |
Families Citing this family (150)
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| BR0108730A (pt) * | 2000-02-28 | 2002-11-05 | Vectura Ltd | Sistema, dispositivo e método para administração de uma droga, bocal de um dispositivo de administração de droga, dispositivo para administração de doses unitárias múltiplas de uma droga, métodos para preparação de um sistema de administração de droga e de uma formulação de droga e para tratamento de um paciente que necessita de doses múltiplas de uma droga, formulação de droga e multiparticulados |
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| WO2019126218A1 (en) | 2017-12-18 | 2019-06-27 | Tris Pharma, Inc. | Modified release drug powder composition comprising gastro-retentive raft forming systems having trigger pulse drug release |
| BR112021006027A2 (pt) | 2018-11-19 | 2021-06-29 | Jazz Pharmaceuticals Ireland Limited | formulações de fármaco resistente a álcool |
| US11400065B2 (en) | 2019-03-01 | 2022-08-02 | Flamel Ireland Limited | Gamma-hydroxybutyrate compositions having improved pharmacokinetics in the fed state |
| US11633405B2 (en) | 2020-02-07 | 2023-04-25 | Therapeuticsmd, Inc. | Steroid hormone pharmaceutical formulations |
| TW202139986A (zh) | 2020-02-21 | 2021-11-01 | 愛爾蘭商爵士製藥愛爾蘭有限責任公司 | 治療原發性嗜睡症之方法 |
| WO2022076824A1 (en) | 2020-10-08 | 2022-04-14 | Jazz Pharmaceuticals Ireland Limited | Sodium oxybate to treat idiopathic hypersomnia |
| US12029719B2 (en) | 2021-04-16 | 2024-07-09 | Allen Morgan | Compounds comprising cannabinoids and other natural ingredients for alieving premenstrual, menstrual and menopausal symptoms |
| US11583510B1 (en) | 2022-02-07 | 2023-02-21 | Flamel Ireland Limited | Methods of administering gamma hydroxybutyrate formulations after a high-fat meal |
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| JP2026513019A (ja) | 2023-02-03 | 2026-04-22 | トリス・フアルマ・インコーポレーテツド | 1晩1回の低ナトリウムオキシベート組成物 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4461759A (en) * | 1983-01-03 | 1984-07-24 | Verex Laboratories, Inc. | Constant release rate solid oral dosage formulations of veropamil |
| LU85943A1 (fr) * | 1985-06-12 | 1987-01-13 | Galephar | Comprimes pharmaceutiques permettant l'administration aisee de pellets, leur preparation et leur utilisation |
| US5028434A (en) * | 1988-07-21 | 1991-07-02 | Alza Corporation | Method for administering nilvadipine for treating cardiovascular symptoms |
| IT1227899B (it) * | 1988-12-23 | 1991-05-14 | Poli Ind Chimica Spa | Rivestimento totale o parziale di principi attivi farmaceutici e relative composizioni |
| US5286497A (en) * | 1991-05-20 | 1994-02-15 | Carderm Capital L.P. | Diltiazem formulation |
-
1994
- 1994-10-18 FR FR9412759A patent/FR2725623A1/fr active Granted
-
1995
- 1995-10-17 CA CA002160762A patent/CA2160762C/fr not_active Expired - Fee Related
- 1995-10-17 IL IL11564695A patent/IL115646A/xx not_active IP Right Cessation
- 1995-10-17 ZA ZA958762A patent/ZA958762B/xx unknown
- 1995-10-17 US US08/544,208 patent/US6022562A/en not_active Expired - Lifetime
- 1995-10-18 AT AT95420286T patent/ATE188117T1/de not_active IP Right Cessation
- 1995-10-18 JP JP51300696A patent/JP4053589B2/ja not_active Expired - Fee Related
- 1995-10-18 WO PCT/FR1995/001369 patent/WO1996011675A2/fr not_active Ceased
- 1995-10-18 BR BRPI9509286A patent/BRPI9509286B8/pt unknown
- 1995-10-18 ES ES95420286T patent/ES2140641T3/es not_active Expired - Lifetime
- 1995-10-18 DE DE69514192T patent/DE69514192T2/de not_active Expired - Lifetime
- 1995-10-18 EP EP95420286A patent/EP0709087B1/fr not_active Expired - Lifetime
- 1995-10-18 BR BR9509286A patent/BR9509286A/pt active IP Right Grant
- 1995-10-18 AU AU38077/95A patent/AU3807795A/en not_active Abandoned
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2000
- 2000-03-15 AR ARP000101126A patent/AR022930A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2160762C (fr) | 2004-12-21 |
| IL115646A (en) | 2000-07-16 |
| JPH10509427A (ja) | 1998-09-14 |
| DE69514192T2 (de) | 2000-07-13 |
| AR022930A2 (es) | 2002-09-04 |
| BRPI9509286B8 (pt) | 2019-12-17 |
| ES2140641T3 (es) | 2000-03-01 |
| DE69514192D1 (de) | 2000-02-03 |
| IL115646A0 (en) | 1996-01-19 |
| FR2725623B1 (enExample) | 1997-02-21 |
| ATE188117T1 (de) | 2000-01-15 |
| WO1996011675A2 (fr) | 1996-04-25 |
| ZA958762B (en) | 1996-05-09 |
| AU3807795A (en) | 1996-05-06 |
| US6022562A (en) | 2000-02-08 |
| WO1996011675A3 (fr) | 1996-06-20 |
| EP0709087B1 (fr) | 1999-12-29 |
| CA2160762A1 (fr) | 1996-04-19 |
| FR2725623A1 (fr) | 1996-04-19 |
| BR9509286A (pt) | 1997-10-14 |
| EP0709087A1 (fr) | 1996-05-01 |
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