JP4011109B2 - アニリン誘導体 - Google Patents

アニリン誘導体 Download PDF

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Publication number
JP4011109B2
JP4011109B2 JP51581696A JP51581696A JP4011109B2 JP 4011109 B2 JP4011109 B2 JP 4011109B2 JP 51581696 A JP51581696 A JP 51581696A JP 51581696 A JP51581696 A JP 51581696A JP 4011109 B2 JP4011109 B2 JP 4011109B2
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JP
Japan
Prior art keywords
alkylamino
amino
alkoxy
alkyl
mixture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
JP51581696A
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English (en)
Japanese (ja)
Other versions
JPH10508616A (ja
Inventor
サザーランド ブラウン ディアーグ
ジェームズ モリス ジェフリー
ピーター トーマス アンドルー
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca UK Ltd
Original Assignee
AstraZeneca UK Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB9422866A external-priority patent/GB9422866D0/en
Priority claimed from GBGB9507308.6A external-priority patent/GB9507308D0/en
Application filed by AstraZeneca UK Ltd filed Critical AstraZeneca UK Ltd
Publication of JPH10508616A publication Critical patent/JPH10508616A/ja
Application granted granted Critical
Publication of JP4011109B2 publication Critical patent/JP4011109B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
JP51581696A 1994-11-12 1995-11-08 アニリン誘導体 Expired - Fee Related JP4011109B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB9422866A GB9422866D0 (en) 1994-11-12 1994-11-12 Aniline derivatives
GBGB9507308.6A GB9507308D0 (en) 1995-04-07 1995-04-07 Aniline derivatives
GB9507308.6 1995-04-07
GB9422866.5 1995-04-07
PCT/GB1995/002606 WO1996015118A1 (en) 1994-11-12 1995-11-08 Aniline derivatives

Publications (2)

Publication Number Publication Date
JPH10508616A JPH10508616A (ja) 1998-08-25
JP4011109B2 true JP4011109B2 (ja) 2007-11-21

Family

ID=26305974

Family Applications (1)

Application Number Title Priority Date Filing Date
JP51581696A Expired - Fee Related JP4011109B2 (ja) 1994-11-12 1995-11-08 アニリン誘導体

Country Status (16)

Country Link
US (1) US5821246A (US08088782-20120103-C00002.png)
EP (1) EP0790986B1 (US08088782-20120103-C00002.png)
JP (1) JP4011109B2 (US08088782-20120103-C00002.png)
AT (1) ATE175962T1 (US08088782-20120103-C00002.png)
AU (1) AU703328B2 (US08088782-20120103-C00002.png)
CA (1) CA2200871C (US08088782-20120103-C00002.png)
DE (1) DE69507505T2 (US08088782-20120103-C00002.png)
DK (1) DK0790986T3 (US08088782-20120103-C00002.png)
ES (1) ES2128092T3 (US08088782-20120103-C00002.png)
FI (1) FI119933B (US08088782-20120103-C00002.png)
IL (1) IL115959A (US08088782-20120103-C00002.png)
MX (1) MX9702956A (US08088782-20120103-C00002.png)
NO (1) NO307178B1 (US08088782-20120103-C00002.png)
NZ (1) NZ294917A (US08088782-20120103-C00002.png)
TW (1) TW321649B (US08088782-20120103-C00002.png)
WO (1) WO1996015118A1 (US08088782-20120103-C00002.png)

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CA2200871A1 (en) 1996-05-23
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EP0790986B1 (en) 1999-01-20
IL115959A0 (en) 1996-01-31
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US5821246A (en) 1998-10-13
NO972152D0 (no) 1997-05-09
FI971970A0 (fi) 1997-05-07
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IL115959A (en) 2004-06-20
NO972152L (no) 1997-05-12
WO1996015118A1 (en) 1996-05-23
EP0790986A1 (en) 1997-08-27
NO307178B1 (no) 2000-02-21
NZ294917A (en) 1999-02-25
FI119933B (fi) 2009-05-15
JPH10508616A (ja) 1998-08-25
AU703328B2 (en) 1999-03-25
DE69507505T2 (de) 1999-06-02
ATE175962T1 (de) 1999-02-15

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