JP2023528014A5 - - Google Patents

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Publication number
JP2023528014A5
JP2023528014A5 JP2022572798A JP2022572798A JP2023528014A5 JP 2023528014 A5 JP2023528014 A5 JP 2023528014A5 JP 2022572798 A JP2022572798 A JP 2022572798A JP 2022572798 A JP2022572798 A JP 2022572798A JP 2023528014 A5 JP2023528014 A5 JP 2023528014A5
Authority
JP
Japan
Prior art keywords
approximately
solid oral
oral formulation
starch
blend
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022572798A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023528014A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/064280 external-priority patent/WO2021239917A1/en
Publication of JP2023528014A publication Critical patent/JP2023528014A/ja
Publication of JP2023528014A5 publication Critical patent/JP2023528014A5/ja
Pending legal-status Critical Current

Links

JP2022572798A 2020-05-29 2021-05-27 ゴナドトロピン放出ホルモンアンタゴニストの組合せ固体経口製剤 Pending JP2023528014A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063032469P 2020-05-29 2020-05-29
US63/032,469 2020-05-29
PCT/EP2021/064280 WO2021239917A1 (en) 2020-05-29 2021-05-27 Combination solid oral dosage forms of gonadotropin-releasing hormone antagonists

Publications (2)

Publication Number Publication Date
JP2023528014A JP2023528014A (ja) 2023-07-03
JP2023528014A5 true JP2023528014A5 (https=) 2024-06-03

Family

ID=76305879

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022572798A Pending JP2023528014A (ja) 2020-05-29 2021-05-27 ゴナドトロピン放出ホルモンアンタゴニストの組合せ固体経口製剤

Country Status (18)

Country Link
US (1) US12551447B2 (https=)
EP (1) EP4157227A1 (https=)
JP (1) JP2023528014A (https=)
KR (1) KR20230028732A (https=)
CN (1) CN115666531B (https=)
AR (1) AR122175A1 (https=)
AU (1) AU2021278303A1 (https=)
BR (1) BR112022023937A2 (https=)
CA (1) CA3185151A1 (https=)
CL (1) CL2022003338A1 (https=)
CO (1) CO2022019160A2 (https=)
EC (1) ECSP22098275A (https=)
IL (1) IL298587A (https=)
MX (1) MX2022015003A (https=)
PE (1) PE20230859A1 (https=)
PY (1) PY2142442A (https=)
UY (1) UY39229A (https=)
WO (1) WO2021239917A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
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EP3518933B2 (en) 2016-09-30 2025-02-26 Sumitomo Pharma Switzerland GmbH Methods of treating uterine fibroids and endometriosis
JP2022551316A (ja) 2019-10-10 2022-12-08 ミオバント サイエンシズ ゲーエムベーハー N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素の結晶形
BR112022023937A2 (pt) 2020-05-29 2022-12-27 Myovant Sciences Gmbh Formas de dosagem oral sólidas de combinação de antagonistas do hormônio liberador de gonadotropina
CN115227648B (zh) * 2022-08-03 2023-09-29 南昌大学 一种瑞卢戈利固体自微乳及其制备方法和应用
CN115068421B (zh) * 2022-08-03 2023-08-04 南昌大学 一种瑞卢戈利纳米混悬液及其制备方法和应用

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BR112022023937A2 (pt) 2020-05-29 2022-12-27 Myovant Sciences Gmbh Formas de dosagem oral sólidas de combinação de antagonistas do hormônio liberador de gonadotropina
EP4243829A1 (en) 2020-11-11 2023-09-20 Myovant Sciences GmbH Methods of administering relugolix
WO2023066941A1 (en) 2021-10-18 2023-04-27 Myovant Sciences Gmbh Crystalline form of an ethanol solvate of n-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxy-3-pyridazinyl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-n'-methoxyurea

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