JP2023513793A5 - - Google Patents

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Publication number
JP2023513793A5
JP2023513793A5 JP2022549144A JP2022549144A JP2023513793A5 JP 2023513793 A5 JP2023513793 A5 JP 2023513793A5 JP 2022549144 A JP2022549144 A JP 2022549144A JP 2022549144 A JP2022549144 A JP 2022549144A JP 2023513793 A5 JP2023513793 A5 JP 2023513793A5
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JP
Japan
Prior art keywords
alkyl
independently
heterocycloalkyl
cycloalkyl
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022549144A
Other languages
English (en)
Japanese (ja)
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JP2023513793A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/018038 external-priority patent/WO2021163627A1/en
Publication of JP2023513793A publication Critical patent/JP2023513793A/ja
Publication of JP2023513793A5 publication Critical patent/JP2023513793A5/ja
Pending legal-status Critical Current

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JP2022549144A 2020-02-14 2021-02-12 大環状ulk1/2阻害剤 Pending JP2023513793A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062977039P 2020-02-14 2020-02-14
US62/977,039 2020-02-14
PCT/US2021/018038 WO2021163627A1 (en) 2020-02-14 2021-02-12 Macrocyclic ulk1/2 inhibitors

Publications (2)

Publication Number Publication Date
JP2023513793A JP2023513793A (ja) 2023-04-03
JP2023513793A5 true JP2023513793A5 (https=) 2024-02-20

Family

ID=77292762

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022549144A Pending JP2023513793A (ja) 2020-02-14 2021-02-12 大環状ulk1/2阻害剤

Country Status (8)

Country Link
US (1) US12594277B2 (https=)
EP (1) EP4103183A4 (https=)
JP (1) JP2023513793A (https=)
KR (1) KR20220153582A (https=)
CN (1) CN115515588A (https=)
AU (1) AU2021221162A1 (https=)
CA (1) CA3171185A1 (https=)
WO (1) WO2021163627A1 (https=)

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WO2022072668A1 (en) * 2020-09-30 2022-04-07 Salk Institute For Biological Studies Patient selection biomarkers for treatment with ulk inhibitors
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WO2024017258A1 (zh) * 2022-07-19 2024-01-25 百极弘烨(南通)医药科技有限公司 Egfr小分子抑制剂、含其的药物组合物及其用途
WO2024233766A1 (en) * 2023-05-10 2024-11-14 Erasca, Inc. Macrocyclic ulk1/2 inhibitors and their use thereof

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WO2022072668A1 (en) 2020-09-30 2022-04-07 Salk Institute For Biological Studies Patient selection biomarkers for treatment with ulk inhibitors

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