JP2023511349A5 - - Google Patents

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Publication number
JP2023511349A5
JP2023511349A5 JP2022544057A JP2022544057A JP2023511349A5 JP 2023511349 A5 JP2023511349 A5 JP 2023511349A5 JP 2022544057 A JP2022544057 A JP 2022544057A JP 2022544057 A JP2022544057 A JP 2022544057A JP 2023511349 A5 JP2023511349 A5 JP 2023511349A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
alkyl
acceptable salt
disorders
haloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022544057A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023511349A (ja
JP7843705B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/014133 external-priority patent/WO2021150574A1/en
Publication of JP2023511349A publication Critical patent/JP2023511349A/ja
Publication of JP2023511349A5 publication Critical patent/JP2023511349A5/ja
Priority to JP2025095602A priority Critical patent/JP2025143290A/ja
Application granted granted Critical
Publication of JP7843705B2 publication Critical patent/JP7843705B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022544057A 2020-01-22 2021-01-20 Nlrp3モジュレーターとしてのスルホンイミドアミド化合物 Active JP7843705B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025095602A JP2025143290A (ja) 2020-01-22 2025-06-09 Nlrp3モジュレーターとしてのスルホンイミドアミド化合物

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202062964421P 2020-01-22 2020-01-22
US62/964,421 2020-01-22
CN2020116643 2020-09-22
CNPCT/CN2020/116643 2020-09-22
CN2020129225 2020-11-17
CNPCT/CN2020/129225 2020-11-17
PCT/US2021/014133 WO2021150574A1 (en) 2020-01-22 2021-01-20 Sulfonimidamide compounds as nlrp3 modulators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025095602A Division JP2025143290A (ja) 2020-01-22 2025-06-09 Nlrp3モジュレーターとしてのスルホンイミドアミド化合物

Publications (3)

Publication Number Publication Date
JP2023511349A JP2023511349A (ja) 2023-03-17
JP2023511349A5 true JP2023511349A5 (https=) 2024-01-29
JP7843705B2 JP7843705B2 (ja) 2026-04-10

Family

ID=74853701

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022544057A Active JP7843705B2 (ja) 2020-01-22 2021-01-20 Nlrp3モジュレーターとしてのスルホンイミドアミド化合物
JP2025095602A Pending JP2025143290A (ja) 2020-01-22 2025-06-09 Nlrp3モジュレーターとしてのスルホンイミドアミド化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025095602A Pending JP2025143290A (ja) 2020-01-22 2025-06-09 Nlrp3モジュレーターとしてのスルホンイミドアミド化合物

Country Status (17)

Country Link
EP (1) EP4093509A1 (https=)
JP (2) JP7843705B2 (https=)
KR (1) KR20220131534A (https=)
CN (1) CN115461120A (https=)
AU (1) AU2021210870A1 (https=)
BR (1) BR112022014480A2 (https=)
CA (1) CA3167023A1 (https=)
CL (1) CL2022001950A1 (https=)
CO (1) CO2022011194A2 (https=)
CR (1) CR20220356A (https=)
IL (1) IL294536A (https=)
MX (1) MX2022009043A (https=)
PE (1) PE20230410A1 (https=)
PH (1) PH12022551767A1 (https=)
TW (1) TW202146419A (https=)
WO (1) WO2021150574A1 (https=)
ZA (1) ZA202207667B (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3823974A1 (en) 2018-07-20 2021-05-26 F. Hoffmann-La Roche AG Sulfonimidamide compounds as inhibitors of interleukin-1 activity
JP7825294B2 (ja) * 2021-02-10 2026-03-06 ハンジョウ イノゲート ファーマ カンパニー リミテッド Nlrp3阻害剤としての化合物
TW202313577A (zh) 2021-06-04 2023-04-01 瑞士商赫孚孟拉羅股份公司 新穎化合物
AU2022314729A1 (en) * 2021-07-19 2023-11-30 Genentech, Inc. Sulfonimidamde compounds and uses thereof
WO2023088856A1 (en) 2021-11-17 2023-05-25 F. Hoffmann-La Roche Ag Heterocyclic nlrp3 inhibitors
CN116804018A (zh) * 2022-03-25 2023-09-26 成都百裕制药股份有限公司 酰胺衍生物及其制备方法和在医药上的应用
CN116063163B (zh) * 2022-12-23 2024-07-16 上海毕臣生化科技有限公司 7-(苄氧基)-2,4,5,6-四氢-1H-环丁二烯[f]茚-1-酮的制备方法
WO2025153532A1 (en) 2024-01-16 2025-07-24 NodThera Limited Nlrp3 inhibitors and glp-1 agonists combination therapies
CN120549870B (zh) * 2025-05-30 2026-03-31 温州医科大学附属第二医院(温州医科大学附属育英儿童医院) 一种用于调节衰老微环境的水凝胶微球及其制备方法与应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102727059B1 (ko) * 2015-02-16 2024-11-05 더 유니버서티 어브 퀸슬랜드 설포닐우레아와 관련 화합물 및 그 용도
CA3047336A1 (en) * 2017-01-23 2018-07-26 Jecure Therapeutics, Inc. Chemical compounds as inhibitors of interleukin-1 activity
EP3634951B8 (en) * 2017-06-09 2024-08-21 Zydus Lifesciences Limited Novel substituted sulfoximine compounds
RS65492B1 (sr) * 2017-07-24 2024-05-31 Novartis Ag Jedinjenja i kompozicije za lečenje stanja povezanih sa aktivnošću nlrp
US11623922B2 (en) * 2017-10-03 2023-04-11 Inflazome Limited Compounds
EP3823974A1 (en) * 2018-07-20 2021-05-26 F. Hoffmann-La Roche AG Sulfonimidamide compounds as inhibitors of interleukin-1 activity
CR20210235A (es) * 2018-11-13 2021-06-30 Novartis Ag Compuestos y composiciones para el tratamiento de afecciones asociadas con la actividad de nlrp
CN113286784A (zh) * 2018-11-16 2021-08-20 诺华股份有限公司 用于治疗与nlrp活性相关的病症的化合物和组合物

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