JP2022515272A5 - - Google Patents
Info
- Publication number
- JP2022515272A5 JP2022515272A5 JP2021537128A JP2021537128A JP2022515272A5 JP 2022515272 A5 JP2022515272 A5 JP 2022515272A5 JP 2021537128 A JP2021537128 A JP 2021537128A JP 2021537128 A JP2021537128 A JP 2021537128A JP 2022515272 A5 JP2022515272 A5 JP 2022515272A5
- Authority
- JP
- Japan
- Prior art keywords
- weight
- sodium
- group
- mixture
- pharmaceutical composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024199593A JP2025032127A (ja) | 2018-12-24 | 2024-11-15 | ピロロピリミジン化合物の治療的使用およびその固形医薬組成物 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201811581815.8 | 2018-12-24 | ||
| CN201811581815 | 2018-12-24 | ||
| CN201910679429 | 2019-07-26 | ||
| CN201910679429.0 | 2019-07-26 | ||
| PCT/CN2019/127837 WO2020135401A1 (zh) | 2018-12-24 | 2019-12-24 | 吡咯并嘧啶化合物的治疗用途及其固体药物组合物 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024199593A Division JP2025032127A (ja) | 2018-12-24 | 2024-11-15 | ピロロピリミジン化合物の治療的使用およびその固形医薬組成物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022515272A JP2022515272A (ja) | 2022-02-17 |
| JP2022515272A5 true JP2022515272A5 (enExample) | 2023-01-06 |
Family
ID=71126879
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021537128A Pending JP2022515272A (ja) | 2018-12-24 | 2019-12-24 | ピロロピリミジン化合物の治療的使用およびその固形医薬組成物 |
| JP2024199593A Pending JP2025032127A (ja) | 2018-12-24 | 2024-11-15 | ピロロピリミジン化合物の治療的使用およびその固形医薬組成物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024199593A Pending JP2025032127A (ja) | 2018-12-24 | 2024-11-15 | ピロロピリミジン化合物の治療的使用およびその固形医薬組成物 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20220072002A1 (enExample) |
| EP (1) | EP3904356A4 (enExample) |
| JP (2) | JP2022515272A (enExample) |
| KR (1) | KR20210132007A (enExample) |
| CN (2) | CN113242859B (enExample) |
| AU (1) | AU2019413421B9 (enExample) |
| CA (1) | CA3123985A1 (enExample) |
| WO (1) | WO2020135401A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2023548855A (ja) * | 2020-11-05 | 2023-11-21 | エグゼリクシス, インコーポレイテッド | キナーゼ阻害剤の医薬組成物 |
| CN118973582A (zh) * | 2022-03-21 | 2024-11-15 | 正大天晴药业集团股份有限公司 | 吡咯并嘧啶化合物治疗中高危骨髓纤维化的用途 |
| WO2024153148A1 (zh) * | 2023-01-18 | 2024-07-25 | 北京普祺医药科技股份有限公司 | 一种杂环化合物、药物组合物及其用途 |
| WO2024230727A1 (zh) * | 2023-05-09 | 2024-11-14 | 正大天晴药业集团股份有限公司 | 一种吡咯并[2,3-c]吡啶酮化合物的联用药物组合物及其用途 |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0775204A1 (en) * | 1994-08-09 | 1997-05-28 | Novartis AG | Antitumor antisense oligonucleotides |
| PL351069A1 (en) * | 1999-12-08 | 2003-03-10 | Pharmacia Corp | Valdecoxib compositions |
| US20070054848A1 (en) * | 2003-03-28 | 2007-03-08 | Masaya Tohyama | Composition and method for nerve regeneration |
| US20050130302A1 (en) * | 2003-09-29 | 2005-06-16 | Reprocell Inc. | Method and composition for regulating expansion of stem cells |
| WO2007089926A2 (en) * | 2006-01-31 | 2007-08-09 | Teva Pharmaceutical Industries Ltd. | Oxcarbazepine pharmaceutical formulation and its method of preparation, wherein oxcarbazepine has a broad and multi-modal particle size distribution |
| KR101566840B1 (ko) * | 2007-03-12 | 2015-11-06 | 와이엠 바이오사이언시즈 오스트레일리아 피티와이 엘티디 | 페닐 아미노 피리미딘 화합물 및 이의 용도 |
| AR076794A1 (es) * | 2009-05-22 | 2011-07-06 | Incyte Corp | Derivados de n-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo [2,3-d]pirimidinas y pirrol-3-il-pirrolo [2,3-d ]pirimidinas como inhibidores de la quinasa janus y composiciones farmaceuticas que los contienen |
| EP3354652B1 (en) * | 2010-03-10 | 2020-05-06 | Incyte Holdings Corporation | Piperidin-4-yl azetidine derivatives as jak1 inhibitors |
| PH12013502523A1 (en) * | 2011-06-14 | 2019-10-11 | Novartis Ag | Combination of panobinostat and ruxolitinib in the treatment of cancer such as a myeloproliferative neoplasm |
| NZ714502A (en) * | 2011-07-05 | 2017-04-28 | Vertex Pharma | Processes and intermediates for producing azaindoles |
| CN104418858B (zh) * | 2013-08-30 | 2018-12-11 | 浙江医药股份有限公司新昌制药厂 | 2,6-二含氮取代的嘌呤衍生物及其制备方法和其药物组合物与应用 |
| CN103585126A (zh) * | 2013-11-18 | 2014-02-19 | 南京艾德凯腾生物医药有限责任公司 | 一种托法替尼组合物及制备方法 |
| NZ723859A (en) * | 2014-03-14 | 2023-01-27 | Servier Lab | Pharmaceutical compositions of therapeutically active compounds and their uses |
| AU2015276857B2 (en) * | 2014-06-20 | 2017-10-19 | Vaxart, Inc. | Anhydrous crystalline free base form of-{2-[1-(6-methyl-3-pyridazinyl)-4-piperidinyl]ethoxy}-3-ethoxy-1,2-benzisoxazole |
| CN105777754B (zh) * | 2014-12-16 | 2019-07-26 | 北京赛林泰医药技术有限公司 | 吡咯并嘧啶化合物 |
| KR101964546B1 (ko) * | 2015-07-27 | 2019-04-01 | 유니켐 레버러토리스 리미티드 | 토파시티닙 경구 붕해 정제 |
| CN108368115B (zh) * | 2015-12-15 | 2020-01-03 | 正大天晴药业集团股份有限公司 | 吡咯并嘧啶化合物的盐 |
| CN107334738B (zh) * | 2016-04-28 | 2021-02-09 | 天津科伦药物研究有限公司 | 一种含巴瑞克替尼的药物组合物及其制备方法和用途 |
| CN107759600A (zh) | 2016-06-16 | 2018-03-06 | 正大天晴药业集团股份有限公司 | 作为jak抑制剂的吡咯并嘧啶化合物的结晶 |
| CN107513069A (zh) * | 2016-06-16 | 2017-12-26 | 正大天晴药业集团股份有限公司 | 手性吡咯并嘧啶化合物的制备方法 |
| CN107513067A (zh) * | 2016-06-16 | 2017-12-26 | 北京赛林泰医药技术有限公司 | 含有取代环戊基的吡咯并嘧啶化合物 |
| HRP20240112T1 (hr) * | 2017-03-14 | 2024-04-12 | Galapagos Nv | Farmaceutske tvari koje uključuju inhibitor janus kinaze (jak) |
| WO2018204787A1 (en) * | 2017-05-05 | 2018-11-08 | Memorial Sloan Kettering Cancer Center | Methods of treatment of myeloproliferative neoplasm |
| US12447154B2 (en) * | 2020-03-09 | 2025-10-21 | Chia Tai Tianqing Pharmaceutical Group Co., Ltd. | Use of pyrrolopyrimidine compound for treating hemophagocytic syndrome |
| CA3222218A1 (en) * | 2021-06-21 | 2022-12-29 | Lifan TU | Use of pyrrolopyrimidine compound and pharmaceutical composition thereof for treating chronic graft versus host disease |
-
2019
- 2019-12-24 CA CA3123985A patent/CA3123985A1/en active Pending
- 2019-12-24 WO PCT/CN2019/127837 patent/WO2020135401A1/zh not_active Ceased
- 2019-12-24 EP EP19905962.7A patent/EP3904356A4/en active Pending
- 2019-12-24 KR KR1020217023608A patent/KR20210132007A/ko not_active Ceased
- 2019-12-24 US US17/417,712 patent/US20220072002A1/en active Pending
- 2019-12-24 AU AU2019413421A patent/AU2019413421B9/en active Active
- 2019-12-24 CN CN201980081492.2A patent/CN113242859B/zh active Active
- 2019-12-24 JP JP2021537128A patent/JP2022515272A/ja active Pending
- 2019-12-24 CN CN202310447777.1A patent/CN116473973A/zh active Pending
-
2024
- 2024-11-15 JP JP2024199593A patent/JP2025032127A/ja active Pending
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