JP2023116489A5 - - Google Patents
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- JP2023116489A5 JP2023116489A5 JP2023084119A JP2023084119A JP2023116489A5 JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5 JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- composition according
- dose
- pharmaceutically acceptable
- acceptable salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762545393P | 2017-08-14 | 2017-08-14 | |
| US62/545,393 | 2017-08-14 | ||
| PCT/US2018/046707 WO2019036472A1 (en) | 2017-08-14 | 2018-08-14 | CORTICOTROPIN RELEASE FACTOR RECEPTOR ANTAGONISTS |
| JP2019572820A JP7285222B2 (ja) | 2017-08-14 | 2018-08-14 | 副腎皮質刺激ホルモン放出因子受容体拮抗薬 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019572820A Division JP7285222B2 (ja) | 2017-08-14 | 2018-08-14 | 副腎皮質刺激ホルモン放出因子受容体拮抗薬 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023116489A JP2023116489A (ja) | 2023-08-22 |
| JP2023116489A5 true JP2023116489A5 (enExample) | 2023-10-26 |
| JP7720354B2 JP7720354B2 (ja) | 2025-08-07 |
Family
ID=65362465
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019572820A Active JP7285222B2 (ja) | 2017-08-14 | 2018-08-14 | 副腎皮質刺激ホルモン放出因子受容体拮抗薬 |
| JP2023084119A Active JP7720354B2 (ja) | 2017-08-14 | 2023-05-22 | 副腎皮質刺激ホルモン放出因子受容体拮抗薬 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019572820A Active JP7285222B2 (ja) | 2017-08-14 | 2018-08-14 | 副腎皮質刺激ホルモン放出因子受容体拮抗薬 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20210137935A1 (enExample) |
| EP (1) | EP3630763A4 (enExample) |
| JP (2) | JP7285222B2 (enExample) |
| KR (1) | KR102644781B1 (enExample) |
| CN (1) | CN110997667A (enExample) |
| AR (1) | AR112471A1 (enExample) |
| AU (3) | AU2018318990B2 (enExample) |
| BR (1) | BR112020002966A2 (enExample) |
| CA (1) | CA3064445A1 (enExample) |
| EA (1) | EA202090321A1 (enExample) |
| MX (2) | MX2019015318A (enExample) |
| TW (2) | TW202400179A (enExample) |
| WO (1) | WO2019036472A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2718918C2 (ru) | 2014-01-21 | 2020-04-15 | Ньюрокрайн Байосайенсиз, Инк. | Антагонисты рецептора cfr1 для лечения врожденной гиперплазии коры надпочечников |
| CN118845788A (zh) | 2017-08-14 | 2024-10-29 | 云杉生物科学公司 | 促肾上腺皮质激素释放因子受体拮抗剂 |
| TW202400179A (zh) * | 2017-08-14 | 2024-01-01 | 美商雲杉生物科技股份有限公司 | 促皮質素釋放因子受體拮抗劑 |
| MX2020011344A (es) * | 2018-04-27 | 2021-02-09 | Spruce Biosciences Inc | Métodos para tratar tumores en reposo suprarrenales testiculares y de ovarios. |
| BR112021010847A2 (pt) | 2018-12-07 | 2021-09-08 | Neurocrine Biosciences Inc. | Antagonista de receptor de crf1, formulações farmacêuticas e formas sólidas das mesmas para o tratamento de hiperplasia adrenal congênita |
| JP2022541550A (ja) * | 2019-07-19 | 2022-09-26 | スプルース バイオサイエンシーズ,インク. | 先天性副腎過形成を処置する方法 |
| US12383536B2 (en) | 2019-09-27 | 2025-08-12 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods of use |
| CN118948857A (zh) * | 2020-08-12 | 2024-11-15 | 云杉生物科学公司 | 用于治疗多囊卵巢综合征的方法和组合物 |
| JP2023540223A (ja) * | 2020-08-26 | 2023-09-22 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | Crf受容体アンタゴニストおよび使用方法 |
| US11708372B2 (en) | 2021-11-19 | 2023-07-25 | Spruce Biosciences, Inc. | Crystalline composition of tildacerfont and methods of use and preparation thereof |
| WO2025188842A1 (en) * | 2024-03-08 | 2025-09-12 | Spruce Biosciences, Inc. | Amorphous solid dispersion of tildacerfont formulations |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE880523T1 (de) * | 1996-02-07 | 2002-07-04 | Janssen Pharmaceutica N.V., Beerse | Pyrazolopyrimidine als crf rezeptor-antagonisten |
| EP1049699B1 (en) * | 1998-01-28 | 2004-04-21 | Bristol-Myers Squibb Pharma Company | Pyrazolotriazines as crf antagonists |
| IL137019A (en) * | 1998-01-28 | 2010-11-30 | Du Pont Pharm Co | 2,7 - dimethyl - 4 - (substituted amino) - 8 - arylpyrazolo [1,5-a] triazine derivatives and pharmaceutical compositions containing them |
| WO2001041761A2 (en) * | 1999-12-08 | 2001-06-14 | Pharmacia Corporation | Valdecoxib compositions |
| JP2008503444A (ja) * | 2004-02-13 | 2008-02-07 | エスビー・ファルムコ・プエルト・リコ・インコーポレイテッド | Crf受容体アンタゴニスト、その調製法、その医薬組成物およびその使用 |
| PL1869049T3 (pl) * | 2005-03-21 | 2009-07-31 | Lilly Co Eli | Związki imidazopirydazyny |
| MX2009003098A (es) | 2006-09-20 | 2009-04-01 | Lilly Co Eli | Compuestos de tiofen pirazolopirimidina. |
| CA2663511C (en) * | 2006-09-20 | 2012-12-04 | Eli Lilly And Company | Thiazole pyrazolopyrimidines as crf1 receptor antagonists |
| BRPI0920838A2 (pt) * | 2008-10-02 | 2018-10-16 | Lilly Co Eli | composto de tiazolil-pirazolopirimidina como intermediários sintéticos e processos sintéticos relacionados |
| TW202400179A (zh) | 2017-08-14 | 2024-01-01 | 美商雲杉生物科技股份有限公司 | 促皮質素釋放因子受體拮抗劑 |
-
2018
- 2018-08-14 TW TW112117030A patent/TW202400179A/zh unknown
- 2018-08-14 EA EA202090321A patent/EA202090321A1/ru unknown
- 2018-08-14 WO PCT/US2018/046707 patent/WO2019036472A1/en not_active Ceased
- 2018-08-14 CA CA3064445A patent/CA3064445A1/en active Pending
- 2018-08-14 EP EP18846043.0A patent/EP3630763A4/en active Pending
- 2018-08-14 CN CN201880038596.0A patent/CN110997667A/zh active Pending
- 2018-08-14 AR ARP180102314 patent/AR112471A1/es unknown
- 2018-08-14 US US16/639,540 patent/US20210137935A1/en not_active Abandoned
- 2018-08-14 TW TW107128345A patent/TWI803504B/zh active
- 2018-08-14 JP JP2019572820A patent/JP7285222B2/ja active Active
- 2018-08-14 MX MX2019015318A patent/MX2019015318A/es unknown
- 2018-08-14 BR BR112020002966-1A patent/BR112020002966A2/pt not_active Application Discontinuation
- 2018-08-14 KR KR1020207005534A patent/KR102644781B1/ko active Active
- 2018-08-14 AU AU2018318990A patent/AU2018318990B2/en not_active Ceased
-
2019
- 2019-12-16 MX MX2022015858A patent/MX2022015858A/es unknown
-
2023
- 2023-03-20 AU AU2023201703A patent/AU2023201703B2/en not_active Ceased
- 2023-05-22 JP JP2023084119A patent/JP7720354B2/ja active Active
-
2024
- 2024-12-16 AU AU2024278470A patent/AU2024278470A1/en not_active Abandoned
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