JP2023116489A5 - - Google Patents

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Publication number
JP2023116489A5
JP2023116489A5 JP2023084119A JP2023084119A JP2023116489A5 JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5 JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
dose
pharmaceutically acceptable
acceptable salt
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Application number
JP2023084119A
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English (en)
Japanese (ja)
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JP7720354B2 (ja
JP2023116489A (ja
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Priority claimed from PCT/US2018/046707 external-priority patent/WO2019036472A1/en
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Publication of JP2023116489A publication Critical patent/JP2023116489A/ja
Publication of JP2023116489A5 publication Critical patent/JP2023116489A5/ja
Application granted granted Critical
Publication of JP7720354B2 publication Critical patent/JP7720354B2/ja
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JP2023084119A 2017-08-14 2023-05-22 副腎皮質刺激ホルモン放出因子受容体拮抗薬 Active JP7720354B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201762545393P 2017-08-14 2017-08-14
US62/545,393 2017-08-14
PCT/US2018/046707 WO2019036472A1 (en) 2017-08-14 2018-08-14 CORTICOTROPIN RELEASE FACTOR RECEPTOR ANTAGONISTS
JP2019572820A JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2019572820A Division JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Publications (3)

Publication Number Publication Date
JP2023116489A JP2023116489A (ja) 2023-08-22
JP2023116489A5 true JP2023116489A5 (enExample) 2023-10-26
JP7720354B2 JP7720354B2 (ja) 2025-08-07

Family

ID=65362465

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2019572820A Active JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬
JP2023084119A Active JP7720354B2 (ja) 2017-08-14 2023-05-22 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2019572820A Active JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Country Status (13)

Country Link
US (1) US20210137935A1 (enExample)
EP (1) EP3630763A4 (enExample)
JP (2) JP7285222B2 (enExample)
KR (1) KR102644781B1 (enExample)
CN (1) CN110997667A (enExample)
AR (1) AR112471A1 (enExample)
AU (3) AU2018318990B2 (enExample)
BR (1) BR112020002966A2 (enExample)
CA (1) CA3064445A1 (enExample)
EA (1) EA202090321A1 (enExample)
MX (2) MX2019015318A (enExample)
TW (2) TW202400179A (enExample)
WO (1) WO2019036472A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2718918C2 (ru) 2014-01-21 2020-04-15 Ньюрокрайн Байосайенсиз, Инк. Антагонисты рецептора cfr1 для лечения врожденной гиперплазии коры надпочечников
CN118845788A (zh) 2017-08-14 2024-10-29 云杉生物科学公司 促肾上腺皮质激素释放因子受体拮抗剂
TW202400179A (zh) * 2017-08-14 2024-01-01 美商雲杉生物科技股份有限公司 促皮質素釋放因子受體拮抗劑
MX2020011344A (es) * 2018-04-27 2021-02-09 Spruce Biosciences Inc Métodos para tratar tumores en reposo suprarrenales testiculares y de ovarios.
BR112021010847A2 (pt) 2018-12-07 2021-09-08 Neurocrine Biosciences Inc. Antagonista de receptor de crf1, formulações farmacêuticas e formas sólidas das mesmas para o tratamento de hiperplasia adrenal congênita
JP2022541550A (ja) * 2019-07-19 2022-09-26 スプルース バイオサイエンシーズ,インク. 先天性副腎過形成を処置する方法
US12383536B2 (en) 2019-09-27 2025-08-12 Neurocrine Biosciences, Inc. CRF receptor antagonists and methods of use
CN118948857A (zh) * 2020-08-12 2024-11-15 云杉生物科学公司 用于治疗多囊卵巢综合征的方法和组合物
JP2023540223A (ja) * 2020-08-26 2023-09-22 ニューロクライン バイオサイエンシーズ,インコーポレイテッド Crf受容体アンタゴニストおよび使用方法
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof
WO2025188842A1 (en) * 2024-03-08 2025-09-12 Spruce Biosciences, Inc. Amorphous solid dispersion of tildacerfont formulations

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE880523T1 (de) * 1996-02-07 2002-07-04 Janssen Pharmaceutica N.V., Beerse Pyrazolopyrimidine als crf rezeptor-antagonisten
EP1049699B1 (en) * 1998-01-28 2004-04-21 Bristol-Myers Squibb Pharma Company Pyrazolotriazines as crf antagonists
IL137019A (en) * 1998-01-28 2010-11-30 Du Pont Pharm Co 2,7 - dimethyl - 4 - (substituted amino) - 8 - arylpyrazolo [1,5-a] triazine derivatives and pharmaceutical compositions containing them
WO2001041761A2 (en) * 1999-12-08 2001-06-14 Pharmacia Corporation Valdecoxib compositions
JP2008503444A (ja) * 2004-02-13 2008-02-07 エスビー・ファルムコ・プエルト・リコ・インコーポレイテッド Crf受容体アンタゴニスト、その調製法、その医薬組成物およびその使用
PL1869049T3 (pl) * 2005-03-21 2009-07-31 Lilly Co Eli Związki imidazopirydazyny
MX2009003098A (es) 2006-09-20 2009-04-01 Lilly Co Eli Compuestos de tiofen pirazolopirimidina.
CA2663511C (en) * 2006-09-20 2012-12-04 Eli Lilly And Company Thiazole pyrazolopyrimidines as crf1 receptor antagonists
BRPI0920838A2 (pt) * 2008-10-02 2018-10-16 Lilly Co Eli composto de tiazolil-pirazolopirimidina como intermediários sintéticos e processos sintéticos relacionados
TW202400179A (zh) 2017-08-14 2024-01-01 美商雲杉生物科技股份有限公司 促皮質素釋放因子受體拮抗劑

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