JP2021528446A5 - - Google Patents

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Publication number
JP2021528446A5
JP2021528446A5 JP2020571690A JP2020571690A JP2021528446A5 JP 2021528446 A5 JP2021528446 A5 JP 2021528446A5 JP 2020571690 A JP2020571690 A JP 2020571690A JP 2020571690 A JP2020571690 A JP 2020571690A JP 2021528446 A5 JP2021528446 A5 JP 2021528446A5
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JP
Japan
Prior art keywords
oxa
azabicyclo
nonane
carboxylate
piperidine
Prior art date
Application number
JP2020571690A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021528446A (ja
JP7317054B2 (ja
JPWO2019243851A5 (https=
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Priority claimed from GBGB1810239.2A external-priority patent/GB201810239D0/en
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Publication of JP2021528446A publication Critical patent/JP2021528446A/ja
Publication of JPWO2019243851A5 publication Critical patent/JPWO2019243851A5/ja
Publication of JP2021528446A5 publication Critical patent/JP2021528446A5/ja
Application granted granted Critical
Publication of JP7317054B2 publication Critical patent/JP7317054B2/ja
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JP2020571690A 2018-06-22 2019-06-24 ムスカリンm1および/またはm4受容体のアゴニストとしての架橋化合物 Active JP7317054B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1810239.2A GB201810239D0 (en) 2018-06-22 2018-06-22 Pharmaceutical compounds
GB1810239.2 2018-06-22
PCT/GB2019/051780 WO2019243851A1 (en) 2018-06-22 2019-06-24 Bridged compounds as agonists of the muscarinic m1 and/or m4 receptor

Publications (4)

Publication Number Publication Date
JP2021528446A JP2021528446A (ja) 2021-10-21
JPWO2019243851A5 JPWO2019243851A5 (https=) 2022-06-30
JP2021528446A5 true JP2021528446A5 (https=) 2022-06-30
JP7317054B2 JP7317054B2 (ja) 2023-07-28

Family

ID=63042513

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020571690A Active JP7317054B2 (ja) 2018-06-22 2019-06-24 ムスカリンm1および/またはm4受容体のアゴニストとしての架橋化合物

Country Status (10)

Country Link
US (2) US10787447B2 (https=)
EP (1) EP3810614B1 (https=)
JP (1) JP7317054B2 (https=)
CN (1) CN112585143B (https=)
AU (1) AU2019289217B2 (https=)
CA (1) CA3104222A1 (https=)
ES (1) ES2984420T3 (https=)
GB (1) GB201810239D0 (https=)
TW (1) TWI822803B (https=)
WO (1) WO2019243851A1 (https=)

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GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds

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