JP2021501805A5 - - Google Patents

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Publication number
JP2021501805A5
JP2021501805A5 JP2020544334A JP2020544334A JP2021501805A5 JP 2021501805 A5 JP2021501805 A5 JP 2021501805A5 JP 2020544334 A JP2020544334 A JP 2020544334A JP 2020544334 A JP2020544334 A JP 2020544334A JP 2021501805 A5 JP2021501805 A5 JP 2021501805A5
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JP
Japan
Prior art keywords
cyclopropyl
vinyl
isoxazole
carboxylic acid
azabicyclo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020544334A
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English (en)
Japanese (ja)
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JP2021501805A (ja
JP7264906B2 (ja
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Publication date
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Priority claimed from PCT/US2018/058323 external-priority patent/WO2019089670A1/en
Publication of JP2021501805A publication Critical patent/JP2021501805A/ja
Publication of JP2021501805A5 publication Critical patent/JP2021501805A5/ja
Application granted granted Critical
Publication of JP7264906B2 publication Critical patent/JP7264906B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020544334A 2017-11-01 2018-10-31 ファルネソイドx受容体モジュレーターとしてのアルケン化合物 Active JP7264906B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762580060P 2017-11-01 2017-11-01
US62/580,060 2017-11-01
PCT/US2018/058323 WO2019089670A1 (en) 2017-11-01 2018-10-31 Alkene compounds as farnesoid x receptor modulators

Publications (3)

Publication Number Publication Date
JP2021501805A JP2021501805A (ja) 2021-01-21
JP2021501805A5 true JP2021501805A5 (enExample) 2022-03-18
JP7264906B2 JP7264906B2 (ja) 2023-04-25

Family

ID=64332184

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020544334A Active JP7264906B2 (ja) 2017-11-01 2018-10-31 ファルネソイドx受容体モジュレーターとしてのアルケン化合物

Country Status (7)

Country Link
US (1) US11168079B2 (enExample)
EP (1) EP3704106B1 (enExample)
JP (1) JP7264906B2 (enExample)
KR (1) KR102732404B1 (enExample)
CN (1) CN111511731B (enExample)
ES (1) ES2944657T3 (enExample)
WO (1) WO2019089670A1 (enExample)

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TW202308629A (zh) 2021-04-28 2023-03-01 法商Enyo製藥公司 使用fxr激動劑作為組合治療以增強tlr3激動劑之療效
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