JP2020510617A5 - - Google Patents
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- Publication number
- JP2020510617A5 JP2020510617A5 JP2019529473A JP2019529473A JP2020510617A5 JP 2020510617 A5 JP2020510617 A5 JP 2020510617A5 JP 2019529473 A JP2019529473 A JP 2019529473A JP 2019529473 A JP2019529473 A JP 2019529473A JP 2020510617 A5 JP2020510617 A5 JP 2020510617A5
- Authority
- JP
- Japan
- Prior art keywords
- benzyl
- pyrazine
- phenyl
- oxo
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662428997P | 2016-12-01 | 2016-12-01 | |
| US62/428,997 | 2016-12-01 | ||
| US201762477512P | 2017-03-28 | 2017-03-28 | |
| US62/477,512 | 2017-03-28 | ||
| PCT/US2017/064229 WO2018102693A1 (en) | 2016-12-01 | 2017-12-01 | Cell impermeable coelenterazine analogues |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020510617A JP2020510617A (ja) | 2020-04-09 |
| JP2020510617A5 true JP2020510617A5 (https=) | 2021-01-21 |
| JP7139330B2 JP7139330B2 (ja) | 2022-09-20 |
Family
ID=60972321
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019529473A Active JP7139330B2 (ja) | 2016-12-01 | 2017-12-01 | 細胞不透過性セレンテラジンアナログ |
Country Status (5)
| Country | Link |
|---|---|
| US (2) | US10577370B2 (https=) |
| EP (2) | EP3548492B1 (https=) |
| JP (1) | JP7139330B2 (https=) |
| DK (1) | DK3548492T5 (https=) |
| WO (1) | WO2018102693A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3548492B1 (en) * | 2016-12-01 | 2023-07-05 | Promega Corporation | Cell impermeable coelenterazine analogues |
| JP7036343B2 (ja) * | 2017-03-28 | 2022-03-15 | 国立大学法人電気通信大学 | 新規セレンテラジン誘導体 |
| JP7419260B2 (ja) * | 2018-05-01 | 2024-01-22 | プロメガ コーポレイション | ＮａｎｏＬｕｃ自殺基質としてのセレンテラジン化合物 |
| WO2020041579A1 (en) * | 2018-08-23 | 2020-02-27 | Promega Corporation | Coelenterazine analogues |
| CA3114424A1 (en) | 2018-10-03 | 2020-04-09 | Promega Corporation | Compositions and methods for stabilizing coelenterazine and analogs and derivatives thereof |
| CN111116594B (zh) * | 2019-12-03 | 2021-05-28 | 山东大学 | 一种C-6位改造NanoLuc类型类似物及其制备方法与应用 |
| KR102940072B1 (ko) * | 2022-01-10 | 2026-03-17 | 주식회사 엘지화학 | 환상 술폰산에스테르 유도체 화합물의 제조방법 |
| CN116082185B (zh) * | 2023-04-06 | 2023-07-21 | 佛山职业技术学院 | 虫酰肼类半抗原、抗原、抗体、检测装置及其制备与应用 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7268229B2 (en) | 2001-11-02 | 2007-09-11 | Promega Corporation | Compounds to co-localize luminophores with luminescent proteins |
| US8883486B2 (en) | 2004-05-04 | 2014-11-11 | Universite De Montreal | Arrestin biosensor |
| WO2008118445A1 (en) | 2007-03-26 | 2008-10-02 | Promega Corporation | Methods to quench light from optical reactions |
| ES2795287T3 (es) | 2009-05-01 | 2020-11-23 | Promega Corp | Luciferasas de Oplophorus sintéticas con mayor emisión de luz |
| SG10202103336SA (en) | 2010-11-02 | 2021-04-29 | Promega Corp | Novel coelenterazine substrates and methods of use |
| CN103180324A (zh) | 2010-11-02 | 2013-06-26 | 普罗美加公司 | 腔肠素衍生物及其使用方法 |
| JP6067019B2 (ja) | 2011-09-02 | 2017-01-25 | プロメガ コーポレイションＰｒｏｍｅｇａ Ｃｏｒｐｏｒａｔｉｏｎ | 代謝的に活性な細胞の酸化還元状態を評価するための化合物及び方法、ならびにｎａｄ（ｐ）／ｎａｄ（ｐ）ｈを測定するための方法 |
| WO2013078244A1 (en) | 2011-11-21 | 2013-05-30 | Promega Corporation | Carboxy x rhodamine analogs |
| CN104395306B (zh) * | 2012-03-02 | 2019-04-23 | 皮尔斯生物科技有限公司 | 作为生物分子的标记染料的吲哚衍生物 |
| EP3099691B1 (en) | 2014-01-29 | 2019-11-20 | Promega Corporation | Pro-substrates for live cell applications |
| US9790537B2 (en) | 2014-01-29 | 2017-10-17 | Promega Corporation | Quinone-masked probes as labeling reagents for cell uptake measurements |
| WO2016210294A1 (en) | 2015-06-25 | 2016-12-29 | Promega Corporation | Thienopyrrole compounds and uses thereof as inhibitors of oplophorus-derived luciferases |
| JP7092677B2 (ja) | 2016-02-15 | 2022-06-28 | プロメガ コーポレイション | セレンテラジン類似体 |
| CN105968114B (zh) * | 2016-05-27 | 2018-11-09 | 山东大学 | 一种腔肠素类似物及其制备方法与应用 |
| JP7212612B2 (ja) * | 2016-07-28 | 2023-01-25 | プロメガ コーポレイション | セレンテラジン類縁体 |
| JP7200102B2 (ja) * | 2016-11-01 | 2023-01-06 | プロメガ コーポレイション | エネルギー受容体に係留されたセレンテラジン類縁体 |
| EP3548492B1 (en) * | 2016-12-01 | 2023-07-05 | Promega Corporation | Cell impermeable coelenterazine analogues |
-
2017
- 2017-12-01 EP EP17829356.9A patent/EP3548492B1/en active Active
- 2017-12-01 US US15/829,262 patent/US10577370B2/en active Active
- 2017-12-01 DK DK17829356.9T patent/DK3548492T5/da active
- 2017-12-01 EP EP23175129.8A patent/EP4279490A3/en active Pending
- 2017-12-01 JP JP2019529473A patent/JP7139330B2/ja active Active
- 2017-12-01 WO PCT/US2017/064229 patent/WO2018102693A1/en not_active Ceased
-
2019
- 2019-12-23 US US16/725,602 patent/US11192894B2/en active Active
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