JP2020507566A5 - - Google Patents

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Publication number
JP2020507566A5
JP2020507566A5 JP2019542672A JP2019542672A JP2020507566A5 JP 2020507566 A5 JP2020507566 A5 JP 2020507566A5 JP 2019542672 A JP2019542672 A JP 2019542672A JP 2019542672 A JP2019542672 A JP 2019542672A JP 2020507566 A5 JP2020507566 A5 JP 2020507566A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound according
membered
cancer
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Withdrawn
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JP2019542672A
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English (en)
Japanese (ja)
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JP2020507566A (ja
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Priority claimed from PCT/US2018/017668 external-priority patent/WO2018148576A1/en
Publication of JP2020507566A publication Critical patent/JP2020507566A/ja
Publication of JP2020507566A5 publication Critical patent/JP2020507566A5/ja
Withdrawn legal-status Critical Current

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JP2019542672A 2017-02-10 2018-02-09 ベンゾチオフェンエストロゲン受容体モジュレーター Withdrawn JP2020507566A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201762457643P 2017-02-10 2017-02-10
US62/457,643 2017-02-10
US201762460358P 2017-02-17 2017-02-17
US62/460,358 2017-02-17
US201862614279P 2018-01-05 2018-01-05
US62/614,279 2018-01-05
PCT/US2018/017668 WO2018148576A1 (en) 2017-02-10 2018-02-09 Benzothiophene estrogen receptor modulators

Publications (2)

Publication Number Publication Date
JP2020507566A JP2020507566A (ja) 2020-03-12
JP2020507566A5 true JP2020507566A5 (enExample) 2021-03-25

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ID=63106724

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JP2019542672A Withdrawn JP2020507566A (ja) 2017-02-10 2018-02-09 ベンゾチオフェンエストロゲン受容体モジュレーター

Country Status (10)

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US (3) US10208011B2 (enExample)
EP (1) EP3580223A4 (enExample)
JP (1) JP2020507566A (enExample)
KR (1) KR20190117582A (enExample)
CN (1) CN110461853A (enExample)
AU (1) AU2018217809A1 (enExample)
CA (1) CA3052810A1 (enExample)
IL (1) IL268319A (enExample)
TW (1) TW201835064A (enExample)
WO (1) WO2018148576A1 (enExample)

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KR102765922B1 (ko) * 2018-02-06 2025-02-11 더 보오드 오브 트러스티스 오브 더 유니버시티 오브 일리노이즈 선택적인 에스트로겐 수용체 분해제로서의 치환된 벤조티오펜 유사체
CN108203404A (zh) * 2018-03-02 2018-06-26 上海博邦医药科技有限公司 (r)-3-苯基哌啶或/和(s)-3-苯基哌啶以及尼拉帕尼的手性中间体的合成方法
JP2021534177A (ja) * 2018-08-16 2021-12-09 ジー1 セラピューティクス, インコーポレイテッド 医学的障害を治療するためのベンゾチオフェンエストロゲン受容体モジュレーター
WO2021065898A1 (ja) 2019-09-30 2021-04-08 日本ケミファ株式会社 アゼパン誘導体
JP7853532B2 (ja) 2020-05-19 2026-04-30 ファーマコスモス ホールディング エー/エス 医学的障害を治療するためのサイクリン依存性キナーゼ阻害化合物
CN113816892A (zh) * 2021-08-27 2021-12-21 安徽鼎旺医药有限公司 一种醋酸巴多昔芬的合成方法
CN113801094A (zh) * 2021-10-29 2021-12-17 中国药科大学 一种2-羰基苯并噻吩类化合物及其制备方法和用途
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