JP2020059759A5 - - Google Patents

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Publication number
JP2020059759A5
JP2020059759A5 JP2020000332A JP2020000332A JP2020059759A5 JP 2020059759 A5 JP2020059759 A5 JP 2020059759A5 JP 2020000332 A JP2020000332 A JP 2020000332A JP 2020000332 A JP2020000332 A JP 2020000332A JP 2020059759 A5 JP2020059759 A5 JP 2020059759A5
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JP
Japan
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crystal
morpholinophenylamino
cyanomethyl
pyrimidin
benzamide
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JP2020000332A
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English (en)
Japanese (ja)
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JP2020059759A (ja
JP6840909B2 (ja
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Publication of JP2020059759A5 publication Critical patent/JP2020059759A5/ja
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JP2020000332A 2014-06-12 2020-01-06 Ｎ−（シアノメチル）−４−（２−（４−モルホリノフェニルアミノ）ピリミジン−４−イル）ベンズアミド塩酸塩 Active JP6840909B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462011315P 2014-06-12 2014-06-12
US62/011,315 2014-06-12

Related Parent Applications (1)

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JP2018164680A Division JP6883560B2 (ja) 2014-06-12 2018-09-03 Ｎ−（シアノメチル）−４−（２−（４−モルホリノフェニルアミノ）ピリミジン−４−イル）ベンズアミド塩酸塩

Publications (3)

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JP2020059759A JP2020059759A (ja) 2020-04-16
JP2020059759A5 true JP2020059759A5 (enExample) 2020-12-24
JP6840909B2 JP6840909B2 (ja) 2021-03-10

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JP2016572271A Active JP6600649B2 (ja) 2014-06-12 2015-06-11 Ｎ−（シアノメチル）−４−（２−（４−モルホリノフェニルアミノ）ピリミジン−４−イル）ベンズアミド塩酸塩
JP2018164680A Active JP6883560B2 (ja) 2014-06-12 2018-09-03 Ｎ−（シアノメチル）−４−（２−（４−モルホリノフェニルアミノ）ピリミジン−４−イル）ベンズアミド塩酸塩
JP2020000332A Active JP6840909B2 (ja) 2014-06-12 2020-01-06 Ｎ−（シアノメチル）−４−（２−（４−モルホリノフェニルアミノ）ピリミジン−４−イル）ベンズアミド塩酸塩
JP2021079700A Active JP7198867B2 (ja) 2014-06-12 2021-05-10 Ｎ－（シアノメチル）－４－（２－（４－モルホリノフェニルアミノ）ピリミジン－４－イル）ベンズアミド塩酸塩
JP2022202374A Active JP7550205B2 (ja) 2014-06-12 2022-12-19 Ｎ－（シアノメチル）－４－（２－（４－モルホリノフェニルアミノ）ピリミジン－４－イル）ベンズアミド塩酸塩

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JP2016572271A Active JP6600649B2 (ja) 2014-06-12 2015-06-11 Ｎ−（シアノメチル）−４−（２−（４−モルホリノフェニルアミノ）ピリミジン−４−イル）ベンズアミド塩酸塩
JP2018164680A Active JP6883560B2 (ja) 2014-06-12 2018-09-03 Ｎ−（シアノメチル）−４−（２−（４−モルホリノフェニルアミノ）ピリミジン−４−イル）ベンズアミド塩酸塩

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JP2021079700A Active JP7198867B2 (ja) 2014-06-12 2021-05-10 Ｎ－（シアノメチル）－４－（２－（４－モルホリノフェニルアミノ）ピリミジン－４－イル）ベンズアミド塩酸塩
JP2022202374A Active JP7550205B2 (ja) 2014-06-12 2022-12-19 Ｎ－（シアノメチル）－４－（２－（４－モルホリノフェニルアミノ）ピリミジン－４－イル）ベンズアミド塩酸塩

Country Status (37)

Country Link
US (5) US9469613B2 (enExample)
EP (3) EP3154950B1 (enExample)
JP (5) JP6600649B2 (enExample)
KR (1) KR101928225B1 (enExample)
CN (2) CN106458929A (enExample)
AP (1) AP2016009551A0 (enExample)
AR (1) AR100818A1 (enExample)
AU (1) AU2015274554B9 (enExample)
BR (1) BR112016028749A2 (enExample)
CA (1) CA2951883C (enExample)
CR (1) CR20160575A (enExample)
CU (1) CU20160183A7 (enExample)
CY (2) CY1123604T1 (enExample)
DK (1) DK3154950T3 (enExample)
EA (1) EA032639B1 (enExample)
EC (1) ECSP16093323A (enExample)
ES (1) ES2822773T3 (enExample)
FI (1) FIC20240025I1 (enExample)
FR (1) FR24C1030I2 (enExample)
HR (1) HRP20201492T1 (enExample)
HU (2) HUE051360T2 (enExample)
IL (3) IL249038B (enExample)
LT (2) LT3154950T (enExample)
LU (1) LUC00353I2 (enExample)
MA (1) MA40067A (enExample)
MX (3) MX374541B (enExample)
NL (1) NL301282I2 (enExample)
NZ (1) NZ725966A (enExample)
PH (1) PH12016502461A1 (enExample)
PL (1) PL3154950T3 (enExample)
PT (1) PT3154950T (enExample)
RS (1) RS61065B1 (enExample)
SG (2) SG11201610079VA (enExample)
SI (1) SI3154950T1 (enExample)
TW (3) TWI681954B (enExample)
UY (1) UY36166A (enExample)
WO (1) WO2015191846A1 (enExample)

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CN106316963B (zh) * 2015-06-26 2021-06-08 苏州泽璟生物制药股份有限公司 吗啡啉苯基氨基嘧啶化合物或其盐的多晶型物
CN106316964B (zh) * 2015-06-26 2019-06-25 苏州泽璟生物制药股份有限公司 苯基氨基嘧啶化合物或其盐的多晶型物
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TWI808055B (zh) 2016-05-11 2023-07-11 美商滬亞生物國際有限公司 Hdac 抑制劑與 pd-1 抑制劑之組合治療
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AU2021273014A1 (en) 2020-05-13 2022-11-17 AbbVie Deutschland GmbH & Co. KG Anti-hemojuvelin (HJV) antibodies for treating anemia of chronic disease
ES3075793T3 (en) 2020-05-13 2026-08-07 Disc Medicine Inc Anti-hemojuvelin (hjv) antibodies for treating myelofibrosis
CN117794545A (zh) 2021-07-30 2024-03-29 葛兰素史密斯克莱有限责任公司 骨髓纤维化的治疗中的生物标志物和患者选择
WO2023019095A2 (en) 2021-08-10 2023-02-16 Sierra Oncology, Inc. Momelotinib combination therapy
WO2023023473A1 (en) 2021-08-16 2023-02-23 Sierra Oncology, Inc. Methods of using momelotinib to treat chronic kidney disease
CN115957221B (zh) * 2021-10-09 2026-01-06 广东东阳光药业股份有限公司 抗纤维化组合物
WO2023152773A1 (en) * 2022-02-14 2023-08-17 Dr. Reddy's Institute Of Life Sciences Solid forms of momelotinib salts and improved processes for the preparation of momelotinib
CN119704552B (zh) * 2025-02-08 2025-06-13 泰州南洋塑料制品有限公司 一种电池槽注塑模具及边缘毛刺废料处理回收装置

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TWI681954B (zh) 2014-06-12 2020-01-11 美商西爾拉癌症醫學公司 Ｎ-（氰基甲基）-４-（２-（４-𠰌啉基苯基胺基）嘧啶-４-基）苯甲醯胺
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