JP2019530725A5 - - Google Patents

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Publication number
JP2019530725A5
JP2019530725A5 JP2019520420A JP2019520420A JP2019530725A5 JP 2019530725 A5 JP2019530725 A5 JP 2019530725A5 JP 2019520420 A JP2019520420 A JP 2019520420A JP 2019520420 A JP2019520420 A JP 2019520420A JP 2019530725 A5 JP2019530725 A5 JP 2019530725A5
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JP
Japan
Prior art keywords
ethyl
cyclohexane
cyano
diazepan
dihydrospiro
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JP2019520420A
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English (en)
Japanese (ja)
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JP7100634B2 (ja
JP2019530725A (ja
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Priority claimed from GBGB1617454.2A external-priority patent/GB201617454D0/en
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Publication of JP2019530725A5 publication Critical patent/JP2019530725A5/ja
Application granted granted Critical
Publication of JP7100634B2 publication Critical patent/JP7100634B2/ja
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JP2019520420A 2016-10-14 2017-10-16 Cns疾患及び疼痛の治療におけるムスカリンm1及び/又はm4受容体の調節因子として活性を有する複素環式化合物。 Active JP7100634B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662408468P 2016-10-14 2016-10-14
US62/408,468 2016-10-14
GBGB1617454.2A GB201617454D0 (en) 2016-10-14 2016-10-14 Pharmaceutical compounds
GB1617454.2 2016-10-14
PCT/GB2017/053115 WO2018069732A1 (en) 2016-10-14 2017-10-16 Heterocyclic compounds having activity as modulators of muscarinic m1 and/or m4 receptors in the treatment of cns diseases and pains.

Publications (3)

Publication Number Publication Date
JP2019530725A JP2019530725A (ja) 2019-10-24
JP2019530725A5 true JP2019530725A5 (enExample) 2020-11-26
JP7100634B2 JP7100634B2 (ja) 2022-07-13

Family

ID=57680777

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019520420A Active JP7100634B2 (ja) 2016-10-14 2017-10-16 Cns疾患及び疼痛の治療におけるムスカリンm1及び/又はm4受容体の調節因子として活性を有する複素環式化合物。

Country Status (8)

Country Link
US (1) US11834407B2 (enExample)
EP (1) EP3526207B1 (enExample)
JP (1) JP7100634B2 (enExample)
CN (1) CN109996792B (enExample)
DK (1) DK3526207T3 (enExample)
ES (1) ES2898206T3 (enExample)
GB (1) GB201617454D0 (enExample)
WO (1) WO2018069732A1 (enExample)

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GB201519352D0 (en) 2015-11-02 2015-12-16 Heptares Therapeutics Ltd Pharmaceutical compounds
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GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202103211D0 (en) 2021-03-08 2021-04-21 Heptares Therapeutics Ltd Pharmaceutical compounds for use in therapy

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