JP2018530595A5 - - Google Patents

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Publication number
JP2018530595A5
JP2018530595A5 JP2018519749A JP2018519749A JP2018530595A5 JP 2018530595 A5 JP2018530595 A5 JP 2018530595A5 JP 2018519749 A JP2018519749 A JP 2018519749A JP 2018519749 A JP2018519749 A JP 2018519749A JP 2018530595 A5 JP2018530595 A5 JP 2018530595A5
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JP
Japan
Prior art keywords
trifluoromethyl
ethyl
imidazo
pyrazole
dihydro
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JP2018519749A
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English (en)
Japanese (ja)
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JP6860559B2 (ja
JP2018530595A (ja
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Priority claimed from PCT/US2016/057135 external-priority patent/WO2017066633A1/en
Publication of JP2018530595A publication Critical patent/JP2018530595A/ja
Publication of JP2018530595A5 publication Critical patent/JP2018530595A5/ja
Priority to JP2021053182A priority Critical patent/JP7090770B2/ja
Application granted granted Critical
Publication of JP6860559B2 publication Critical patent/JP6860559B2/ja
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JP2018519749A 2015-10-16 2016-10-14 Ep4アンタゴニスト Active JP6860559B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021053182A JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201562242734P 2015-10-16 2015-10-16
US201562242748P 2015-10-16 2015-10-16
US62/242,734 2015-10-16
US62/242,748 2015-10-16
BD252/2016 2016-10-13
BD2522016 2016-10-13
PCT/US2016/057135 WO2017066633A1 (en) 2015-10-16 2016-10-14 Ep4 antagonists

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021053182A Division JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Publications (3)

Publication Number Publication Date
JP2018530595A JP2018530595A (ja) 2018-10-18
JP2018530595A5 true JP2018530595A5 (cg-RX-API-DMAC7.html) 2019-11-28
JP6860559B2 JP6860559B2 (ja) 2021-04-14

Family

ID=58518017

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JP2018519749A Active JP6860559B2 (ja) 2015-10-16 2016-10-14 Ep4アンタゴニスト
JP2021053182A Active JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021053182A Active JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Country Status (11)

Country Link
US (3) US10316040B2 (cg-RX-API-DMAC7.html)
EP (1) EP3362454B1 (cg-RX-API-DMAC7.html)
JP (2) JP6860559B2 (cg-RX-API-DMAC7.html)
KR (1) KR102684436B1 (cg-RX-API-DMAC7.html)
CN (1) CN108473497B (cg-RX-API-DMAC7.html)
AU (1) AU2016338679B2 (cg-RX-API-DMAC7.html)
BR (1) BR112018007664B1 (cg-RX-API-DMAC7.html)
CA (1) CA3002144C (cg-RX-API-DMAC7.html)
IL (1) IL258737A (cg-RX-API-DMAC7.html)
MX (1) MX390051B (cg-RX-API-DMAC7.html)
WO (1) WO2017066633A1 (cg-RX-API-DMAC7.html)

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EP3625227B1 (en) 2017-05-18 2022-09-14 Idorsia Pharmaceuticals Ltd Benzofurane and benzothiophene derivatives as pge2 receptor modulators
AR111808A1 (es) 2017-05-18 2019-08-21 Idorsia Pharmaceuticals Ltd Derivados de pirimidina como moduladores del receptor de pge2
SI3625222T1 (sl) 2017-05-18 2021-11-30 Idorsia Pharmaceuticals Ltd Derivati fenila kot modulatorji receptorja pge2
TWI768043B (zh) 2017-05-18 2022-06-21 瑞士商愛杜西亞製藥有限公司 N-取代吲哚衍生物
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EP4245301A4 (en) 2020-11-13 2024-08-21 ONO Pharmaceutical Co., Ltd. TREATMENT OF CANCER BY COMBINED USE OF AN EP4 ANTAGONIST AND AN IMMUNE CHECKPOINT INHIBITOR

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