JP2017528519A5 - - Google Patents
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- Publication number
- JP2017528519A5 JP2017528519A5 JP2017530971A JP2017530971A JP2017528519A5 JP 2017528519 A5 JP2017528519 A5 JP 2017528519A5 JP 2017530971 A JP2017530971 A JP 2017530971A JP 2017530971 A JP2017530971 A JP 2017530971A JP 2017528519 A5 JP2017528519 A5 JP 2017528519A5
- Authority
- JP
- Japan
- Prior art keywords
- pyridin
- methoxy
- benzoxazol
- methyl
- methoxypyridin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462043603P | 2014-08-29 | 2014-08-29 | |
| US62/043,603 | 2014-08-29 | ||
| PCT/US2015/047407 WO2016033445A1 (en) | 2014-08-29 | 2015-08-28 | Probes for imaging huntingtin protein |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020214504A Division JP7126541B2 (ja) | 2014-08-29 | 2020-12-24 | ハンチントンタンパク質のイメージング用プローブ |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017528519A JP2017528519A (ja) | 2017-09-28 |
| JP2017528519A5 true JP2017528519A5 (enExample) | 2018-10-04 |
| JP6817207B2 JP6817207B2 (ja) | 2021-01-20 |
Family
ID=55400648
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017530971A Active JP6817207B2 (ja) | 2014-08-29 | 2015-08-28 | ハンチントンタンパク質のイメージング用プローブ |
| JP2020214504A Active JP7126541B2 (ja) | 2014-08-29 | 2020-12-24 | ハンチントンタンパク質のイメージング用プローブ |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020214504A Active JP7126541B2 (ja) | 2014-08-29 | 2020-12-24 | ハンチントンタンパク質のイメージング用プローブ |
Country Status (20)
| Country | Link |
|---|---|
| US (3) | US10479802B2 (enExample) |
| EP (2) | EP4006016A3 (enExample) |
| JP (2) | JP6817207B2 (enExample) |
| KR (2) | KR102586736B1 (enExample) |
| CN (2) | CN107108534B (enExample) |
| AU (1) | AU2015308774B2 (enExample) |
| BR (1) | BR112017004141B8 (enExample) |
| CA (1) | CA2959501C (enExample) |
| DK (1) | DK3186233T3 (enExample) |
| EA (1) | EA035646B1 (enExample) |
| ES (1) | ES2898965T3 (enExample) |
| HR (1) | HRP20211778T1 (enExample) |
| HU (1) | HUE056957T2 (enExample) |
| IL (1) | IL250803B (enExample) |
| MX (2) | MX380810B (enExample) |
| PL (1) | PL3186233T3 (enExample) |
| PT (1) | PT3186233T (enExample) |
| SG (1) | SG11201701600QA (enExample) |
| SI (1) | SI3186233T1 (enExample) |
| WO (1) | WO2016033445A1 (enExample) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX386798B (es) | 2014-08-29 | 2025-03-19 | Chdi Foundation Inc | Sondas para la proyección de imagen de la proteína huntingtina. |
| US11071793B2 (en) | 2014-08-29 | 2021-07-27 | Chdi Foundation, Inc. | Probes for imaging huntingtin protein |
| KR102586736B1 (ko) * | 2014-08-29 | 2023-10-11 | 씨에이치디아이 파운데이션, 인코포레이티드 | 헌팅틴을 단백질 영상화하기 위한 프로브 |
| CA2959505A1 (en) | 2014-08-29 | 2016-03-03 | Chdi Foundation, Inc. | Probes for imaging huntingtin protein |
| EP3340796B1 (en) | 2015-08-28 | 2021-04-21 | CHDI Foundation, Inc. | Probes for imaging huntingtin protein |
| KR20240036709A (ko) | 2016-03-11 | 2024-03-20 | 에이씨 이뮨 에스에이 | 진단 및 치료를 위한 바이사이클릭 화합물 |
| CN107056723A (zh) * | 2017-04-21 | 2017-08-18 | 云南大学 | 一种具有抑制血管内皮生长因子受体信号传导的化合物 |
| DK3682881T3 (da) | 2017-09-14 | 2026-05-11 | Daiichi Sankyo Co Limited | Forbindelse med cyklisk struktur |
| CN111989328B (zh) | 2018-04-20 | 2023-04-18 | 拜耳公司 | 作为害虫防治剂的杂环衍生物 |
| ES2988770T3 (es) | 2018-06-08 | 2024-11-21 | Ac Immune Sa | Nuevos compuestos para diagnóstico |
| ES2974634T3 (es) | 2018-12-21 | 2024-06-28 | Celgene Corp | Inhibidores de tienopiridinas de RIPK2 |
| WO2020176424A1 (en) | 2019-02-25 | 2020-09-03 | Chdi Foundation, Inc. | Compounds for targeting mutant huntingtin protein and uses thereof |
| CN111635400A (zh) | 2019-03-02 | 2020-09-08 | 察略盛医药科技(上海)有限公司 | 吡唑并[1,5-a]吡啶类衍生物、及其制备方法和用途 |
| US11992535B2 (en) * | 2019-12-18 | 2024-05-28 | Chdi Foundation, Inc. | Compounds and probes for imaging huntingtin protein |
| CA3167339A1 (en) | 2020-01-13 | 2021-07-22 | Verge Analytics, Inc. | Substituted pyrazolo-pyrimidines and uses thereof |
| CA3175602A1 (en) | 2020-05-07 | 2021-11-11 | Jerome Molette | Novel compounds for diagnosis |
| AU2021322253A1 (en) * | 2020-08-06 | 2023-02-23 | Chdi Foundation, Inc. | Heterobiaryl compounds and imaging agents for imaging Huntingtin protein |
| WO2022216947A1 (en) * | 2021-04-08 | 2022-10-13 | Chdi Foundation, Inc. | Isoindolinone compounds and imaging agents for imaging huntingtin protein |
| KR20240001208A (ko) * | 2021-04-27 | 2024-01-03 | 씨에이치디아이 파운데이션, 인코포레이티드 | 헌팅틴 단백질 영상화를 위한 중수소화 화합물 및 영상화제 |
| MX2024000313A (es) | 2021-07-09 | 2024-03-06 | Plexium Inc | Compuestos de arilo y composiciones farmaceuticas que modulan la ikzf2. |
| WO2023084000A1 (en) | 2021-11-10 | 2023-05-19 | Ac Immune Sa | 4h-imidazo[1,5-b]pyrazole derivatives for diagnosis |
| US20250034149A1 (en) | 2021-11-10 | 2025-01-30 | Ac Immune Sa | Dihydropyrrolo[3,4c]-pyrazole derivatives and their use in diagnosis |
| EP4430044A1 (en) | 2021-11-10 | 2024-09-18 | AC Immune SA | Dihydropyrrolo[3,4-c]pyrazole derivatives and their use in diagnosis |
| TW202425965A (zh) | 2022-09-30 | 2024-07-01 | 日商科研製藥股份有限公司 | 縮環化合物及含有其之醫藥 |
| EP4634191A1 (en) | 2022-12-16 | 2025-10-22 | AC Immune SA | Novel compounds for diagnosis |
| JP2026500311A (ja) | 2022-12-16 | 2026-01-06 | エーシー・イミューン・エス・アー | 診断のための新規化合物 |
| KR20260027149A (ko) * | 2023-05-18 | 2026-02-27 | 엔베다 테라퓨틱스, 인크. | G 단백질 결합 수용체 길항제 |
| WO2025037013A1 (en) | 2023-08-16 | 2025-02-20 | Ac Immune Sa | Diagnostic compounds that bind to alpha-synuclein |
| WO2025106920A1 (en) * | 2023-11-15 | 2025-05-22 | Yale University | Parp pet imaging agents and methods of using the same |
| CN119264072B (zh) * | 2024-12-06 | 2025-05-02 | 国科大杭州高等研究院 | 对细胞成像的荧光探针及其合成方法和应用 |
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| CA2959505A1 (en) | 2014-08-29 | 2016-03-03 | Chdi Foundation, Inc. | Probes for imaging huntingtin protein |
| KR102586736B1 (ko) | 2014-08-29 | 2023-10-11 | 씨에이치디아이 파운데이션, 인코포레이티드 | 헌팅틴을 단백질 영상화하기 위한 프로브 |
| US11071793B2 (en) | 2014-08-29 | 2021-07-27 | Chdi Foundation, Inc. | Probes for imaging huntingtin protein |
| MX386798B (es) | 2014-08-29 | 2025-03-19 | Chdi Foundation Inc | Sondas para la proyección de imagen de la proteína huntingtina. |
| EP3340796B1 (en) | 2015-08-28 | 2021-04-21 | CHDI Foundation, Inc. | Probes for imaging huntingtin protein |
-
2015
- 2015-08-28 KR KR1020227035965A patent/KR102586736B1/ko active Active
- 2015-08-28 PL PL15836321T patent/PL3186233T3/pl unknown
- 2015-08-28 JP JP2017530971A patent/JP6817207B2/ja active Active
- 2015-08-28 MX MX2017002703A patent/MX380810B/es unknown
- 2015-08-28 KR KR1020177008383A patent/KR102456946B1/ko active Active
- 2015-08-28 DK DK15836321.8T patent/DK3186233T3/da active
- 2015-08-28 EA EA201790407A patent/EA035646B1/ru unknown
- 2015-08-28 HR HRP20211778TT patent/HRP20211778T1/hr unknown
- 2015-08-28 SG SG11201701600QA patent/SG11201701600QA/en unknown
- 2015-08-28 EP EP21192872.6A patent/EP4006016A3/en not_active Withdrawn
- 2015-08-28 BR BR112017004141A patent/BR112017004141B8/pt active IP Right Grant
- 2015-08-28 US US15/507,208 patent/US10479802B2/en active Active
- 2015-08-28 HU HUE15836321A patent/HUE056957T2/hu unknown
- 2015-08-28 CN CN201580058282.3A patent/CN107108534B/zh active Active
- 2015-08-28 AU AU2015308774A patent/AU2015308774B2/en active Active
- 2015-08-28 SI SI201531751T patent/SI3186233T1/sl unknown
- 2015-08-28 WO PCT/US2015/047407 patent/WO2016033445A1/en not_active Ceased
- 2015-08-28 PT PT158363218T patent/PT3186233T/pt unknown
- 2015-08-28 CN CN202310475134.8A patent/CN116655618B/zh active Active
- 2015-08-28 ES ES15836321T patent/ES2898965T3/es active Active
- 2015-08-28 CA CA2959501A patent/CA2959501C/en active Active
- 2015-08-28 EP EP15836321.8A patent/EP3186233B8/en active Active
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2017
- 2017-02-27 IL IL250803A patent/IL250803B/en active IP Right Grant
- 2017-02-28 MX MX2021003311A patent/MX2021003311A/es unknown
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2019
- 2019-08-02 US US16/530,594 patent/US11059836B2/en active Active
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2020
- 2020-12-24 JP JP2020214504A patent/JP7126541B2/ja active Active
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2022
- 2022-08-05 US US17/881,895 patent/US12258355B2/en active Active