JP2016516815A5 - - Google Patents

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JP2016516815A5
JP2016516815A5 JP2016509049A JP2016509049A JP2016516815A5 JP 2016516815 A5 JP2016516815 A5 JP 2016516815A5 JP 2016509049 A JP2016509049 A JP 2016509049A JP 2016509049 A JP2016509049 A JP 2016509049A JP 2016516815 A5 JP2016516815 A5 JP 2016516815A5
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compound
formula
mixture
base
producing
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JP2016509049A
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JP2016516815A (ja
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Priority claimed from PCT/US2014/034301 external-priority patent/WO2014172423A1/en
Publication of JP2016516815A publication Critical patent/JP2016516815A/ja
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JP2016509049A 2013-04-17 2014-04-16 1−エチル−7−(2−メチル−6−(1H−1,2,4−トリアゾール−3−イル)ピリジン−3−イル)−3,4−ジヒドロピラジノ[2,3−b]ピラジン−2(1H)−オンに関する医薬製剤、プロセス、固形形態、及び使用方法 Pending JP2016516815A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361813064P 2013-04-17 2013-04-17
US61/813,064 2013-04-17
US201361911201P 2013-12-03 2013-12-03
US61/911,201 2013-12-03
PCT/US2014/034301 WO2014172423A1 (en) 2013-04-17 2014-04-16 Pharmaceutical formulations, processes, solid forms and methods of use relating to 1-ethyl-7-(2-methyl-6-(1h-1,2,4-triazol-3-yl) pyridin-3-yl) -3,4-dihydropyrazino[2,3-b]pyrazin-2(1h)-one

Related Child Applications (1)

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JP2018103448A Division JP6517979B2 (ja) 2013-04-17 2018-05-30 1−エチル−7−(2−メチル−6−(1H−1,2,4−トリアゾール−3−イル)ピリジン−3−イル)−3,4−ジヒドロピラジノ[2,3−b]ピラジン−2(1H)−オンに関する医薬製剤、プロセス、固形形態、及び使用方法

Publications (2)

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JP2016516815A JP2016516815A (ja) 2016-06-09
JP2016516815A5 true JP2016516815A5 (enExample) 2017-05-18

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JP2016509049A Pending JP2016516815A (ja) 2013-04-17 2014-04-16 1−エチル−7−(2−メチル−6−(1H−1,2,4−トリアゾール−3−イル)ピリジン−3−イル)−3,4−ジヒドロピラジノ[2,3−b]ピラジン−2(1H)−オンに関する医薬製剤、プロセス、固形形態、及び使用方法
JP2018103448A Active JP6517979B2 (ja) 2013-04-17 2018-05-30 1−エチル−7−(2−メチル−6−(1H−1,2,4−トリアゾール−3−イル)ピリジン−3−イル)−3,4−ジヒドロピラジノ[2,3−b]ピラジン−2(1H)−オンに関する医薬製剤、プロセス、固形形態、及び使用方法

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JP2018103448A Active JP6517979B2 (ja) 2013-04-17 2018-05-30 1−エチル−7−(2−メチル−6−(1H−1,2,4−トリアゾール−3−イル)ピリジン−3−イル)−3,4−ジヒドロピラジノ[2,3−b]ピラジン−2(1H)−オンに関する医薬製剤、プロセス、固形形態、及び使用方法

Country Status (24)

Country Link
US (3) US9359364B2 (enExample)
EP (2) EP2986609B1 (enExample)
JP (2) JP2016516815A (enExample)
KR (2) KR102459285B1 (enExample)
CN (2) CN105324381A (enExample)
AU (1) AU2014254050B2 (enExample)
BR (1) BR112015026300A2 (enExample)
CA (1) CA2909629C (enExample)
CL (1) CL2015003068A1 (enExample)
CR (1) CR20150577A (enExample)
EA (2) EA030726B1 (enExample)
ES (1) ES2744198T3 (enExample)
HK (1) HK1221951A1 (enExample)
IL (1) IL242102B (enExample)
MX (2) MX393164B (enExample)
NI (1) NI201500152A (enExample)
NZ (2) NZ730189A (enExample)
PE (1) PE20160041A1 (enExample)
PH (2) PH12015502394A1 (enExample)
SA (1) SA515370014B1 (enExample)
SG (1) SG11201508527VA (enExample)
TW (1) TW201527300A (enExample)
WO (1) WO2014172423A1 (enExample)
ZA (1) ZA201507737B (enExample)

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NZ629486A (en) 2013-05-29 2017-11-24 Signal Pharm Llc Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1h)-one, a solid form thereof and methods of their use
NZ714742A (en) 2014-04-16 2017-04-28 Signal Pharm Llc Solid forms of 1-ethyl-7-(2-methyl-6-(1h-1,2,4-triazol-3-yl)pyridin-3-yl)-3,4-dihydropyrazino[2,3-b]pyrazin-2(1h)-one, compositions thereof and methods of their use
EP3131551A4 (en) * 2014-04-16 2017-09-20 Signal Pharmaceuticals, LLC SOLID FORMS COMPRISING 1-ETHYL-7-(2-METHYL-6-(1H-1,2,4-TRIAZOL-3-YL) PYRIDIN-3-YL)-3,4-DIHYDROPYRAZINO(2,3-b)PYRAZIN-2(1H)-ONE, AND A COFORMER, COMPOSITIONS AND METHODS OF USE THEREOF
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