JP2014505035A5 - - Google Patents

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JP2014505035A5
JP2014505035A5 JP2013543478A JP2013543478A JP2014505035A5 JP 2014505035 A5 JP2014505035 A5 JP 2014505035A5 JP 2013543478 A JP2013543478 A JP 2013543478A JP 2013543478 A JP2013543478 A JP 2013543478A JP 2014505035 A5 JP2014505035 A5 JP 2014505035A5
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disease
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injury
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JP6144627B2 (ja
JP2014505035A (ja
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Priority claimed from PCT/CA2011/050773 external-priority patent/WO2012079172A1/en
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JP2013543478A 2010-12-15 2011-12-14 アミノ酸1および3で修飾されたシクロスポリン類似体分子 Active JP6144627B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US42357610P 2010-12-15 2010-12-15
US61/423,576 2010-12-15
PCT/CA2011/050773 WO2012079172A1 (en) 2010-12-15 2011-12-14 Cyclosporine analogue molecules modified at amino acid 1 and 3

Related Child Applications (1)

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JP2017024484A Division JP6831259B2 (ja) 2010-12-15 2017-02-13 アミノ酸1および3で修飾されたシクロスポリン類似体分子

Publications (3)

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JP2014505035A JP2014505035A (ja) 2014-02-27
JP2014505035A5 true JP2014505035A5 (enExample) 2015-07-09
JP6144627B2 JP6144627B2 (ja) 2017-06-07

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Application Number Title Priority Date Filing Date
JP2013543478A Active JP6144627B2 (ja) 2010-12-15 2011-12-14 アミノ酸1および3で修飾されたシクロスポリン類似体分子
JP2017024484A Active JP6831259B2 (ja) 2010-12-15 2017-02-13 アミノ酸1および3で修飾されたシクロスポリン類似体分子
JP2019018182A Pending JP2019123712A (ja) 2010-12-15 2019-02-04 アミノ酸1および3で修飾されたシクロスポリン類似体分子

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JP2017024484A Active JP6831259B2 (ja) 2010-12-15 2017-02-13 アミノ酸1および3で修飾されたシクロスポリン類似体分子
JP2019018182A Pending JP2019123712A (ja) 2010-12-15 2019-02-04 アミノ酸1および3で修飾されたシクロスポリン類似体分子

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US (2) US9200038B2 (enExample)
EP (2) EP3461835A1 (enExample)
JP (3) JP6144627B2 (enExample)
KR (3) KR102011339B1 (enExample)
CN (2) CN107496902B (enExample)
AU (1) AU2011342284C1 (enExample)
BR (1) BR112013014890B1 (enExample)
CA (1) CA2821009C (enExample)
DK (1) DK2651965T3 (enExample)
ES (1) ES2705750T3 (enExample)
HR (1) HRP20190096T1 (enExample)
HU (1) HUE042490T2 (enExample)
IL (1) IL226792A (enExample)
LT (1) LT2651965T (enExample)
MX (1) MX353720B (enExample)
MY (2) MY192981A (enExample)
NZ (1) NZ611620A (enExample)
PH (1) PH12013501213A1 (enExample)
PL (1) PL2651965T3 (enExample)
PT (1) PT2651965T (enExample)
RU (1) RU2630690C9 (enExample)
SG (2) SG191069A1 (enExample)
SI (1) SI2651965T1 (enExample)
TR (1) TR201900128T4 (enExample)
WO (1) WO2012079172A1 (enExample)

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TW201639873A (zh) 2015-01-08 2016-11-16 歐樂根公司 Mebmt側鏈已環化之環孢菌素衍生物
CN118324867A (zh) * 2016-05-17 2024-07-12 美国科技环球有限公司 新型环孢菌素衍生物及其用途
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WO2019246312A1 (en) 2018-06-20 2019-12-26 Progenity, Inc. Treatment of a disease of the gastrointestinal tract with an immunomodulator
ES2990218T3 (es) * 2018-08-22 2024-11-29 Bacainn Biotherapeutics Ltd Composiciones de ciclosporina y métodos de uso
US12409206B2 (en) 2020-02-19 2025-09-09 Hepion Pharmaceuticals, Inc. Use of cyclosporine analogues for treating fibrosis
AR121404A1 (es) * 2020-02-25 2022-06-01 Hepion Pharmaceuticals Inc Uso de análogos de ciclosporina para tratar cáncer
WO2021190603A1 (en) * 2020-03-26 2021-09-30 Farsight Medical Technology (Shanghai) Co., Ltd. Cyclophilin inhibitors and uses thereof
TW202144379A (zh) 2020-03-26 2021-12-01 大陸商睿諾醫療科技(上海)有限公司 親環蛋白抑制劑及其用途
CN116829168A (zh) * 2020-11-29 2023-09-29 海必恩制药公司 环孢菌素类似物作为抗血栓形成剂的用途
CN113173974B (zh) 2021-03-18 2024-09-06 北京大学深圳研究生院 环孢素衍生物的合成方法
CN115677533B (zh) * 2021-07-30 2023-12-05 沈阳化工研究院有限公司 一种4-庚基苯甲腈的制备方法
IT202300001116A1 (it) * 2023-01-25 2024-07-25 Indena Spa Processo per la preparazione di un intermedio utile per la sintesi di voclosporina
CN121219307A (zh) * 2023-06-02 2025-12-26 睿诺医疗科技(上海)有限公司 亲环蛋白抑制剂及其用途
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