JP2014505035A5 - - Google Patents

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JP2014505035A5
JP2014505035A5 JP2013543478A JP2013543478A JP2014505035A5 JP 2014505035 A5 JP2014505035 A5 JP 2014505035A5 JP 2013543478 A JP2013543478 A JP 2013543478A JP 2013543478 A JP2013543478 A JP 2013543478A JP 2014505035 A5 JP2014505035 A5 JP 2014505035A5
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disease
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injury
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JP6144627B2 (ja
JP2014505035A (ja
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Priority claimed from PCT/CA2011/050773 external-priority patent/WO2012079172A1/en
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JP2013543478A 2010-12-15 2011-12-14 アミノ酸１および３で修飾されたシクロスポリン類似体分子 Active JP6144627B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US42357610P 2010-12-15 2010-12-15
US61/423,576 2010-12-15
PCT/CA2011/050773 WO2012079172A1 (en) 2010-12-15 2011-12-14 Cyclosporine analogue molecules modified at amino acid 1 and 3

Related Child Applications (1)

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JP2017024484A Division JP6831259B2 (ja) 2010-12-15 2017-02-13 アミノ酸１および３で修飾されたシクロスポリン類似体分子

Publications (3)

Publication Number Publication Date
JP2014505035A JP2014505035A (ja) 2014-02-27
JP2014505035A5 true JP2014505035A5 (enExample) 2015-07-09
JP6144627B2 JP6144627B2 (ja) 2017-06-07

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Application Number Title Priority Date Filing Date
JP2013543478A Active JP6144627B2 (ja) 2010-12-15 2011-12-14 アミノ酸１および３で修飾されたシクロスポリン類似体分子
JP2017024484A Active JP6831259B2 (ja) 2010-12-15 2017-02-13 アミノ酸１および３で修飾されたシクロスポリン類似体分子
JP2019018182A Pending JP2019123712A (ja) 2010-12-15 2019-02-04 アミノ酸１および３で修飾されたシクロスポリン類似体分子

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JP2017024484A Active JP6831259B2 (ja) 2010-12-15 2017-02-13 アミノ酸１および３で修飾されたシクロスポリン類似体分子
JP2019018182A Pending JP2019123712A (ja) 2010-12-15 2019-02-04 アミノ酸１および３で修飾されたシクロスポリン類似体分子

Country Status (25)

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US (2) US9200038B2 (enExample)
EP (2) EP2651965B1 (enExample)
JP (3) JP6144627B2 (enExample)
KR (3) KR102305423B1 (enExample)
CN (2) CN103443119B (enExample)
AU (1) AU2011342284C1 (enExample)
BR (1) BR112013014890B1 (enExample)
CA (1) CA2821009C (enExample)
DK (1) DK2651965T3 (enExample)
ES (1) ES2705750T3 (enExample)
HR (1) HRP20190096T1 (enExample)
HU (1) HUE042490T2 (enExample)
IL (1) IL226792A (enExample)
LT (1) LT2651965T (enExample)
MX (1) MX353720B (enExample)
MY (2) MY165152A (enExample)
NZ (1) NZ611620A (enExample)
PH (1) PH12013501213A1 (enExample)
PL (1) PL2651965T3 (enExample)
PT (1) PT2651965T (enExample)
RU (1) RU2630690C9 (enExample)
SG (2) SG191069A1 (enExample)
SI (1) SI2651965T1 (enExample)
TR (1) TR201900128T4 (enExample)
WO (1) WO2012079172A1 (enExample)

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CN121554542A (zh) 2018-08-22 2026-02-24 贝凯恩生物医疗技术有限公司 环孢菌素组合物及使用方法
US12594275B2 (en) 2019-02-07 2026-04-07 The Regents Of The University Of California Immunophilin binding agents and uses thereof
TW202143994A (zh) 2020-02-19 2021-12-01 美商希皮恩製藥公司 環孢素類似物於治療纖維化之用途
CN115484961A (zh) * 2020-02-25 2022-12-16 海必恩制药公司 环孢菌素类似物用于治疗癌症的用途
CA3172535A1 (en) 2020-03-26 2021-09-30 Ching-Pong Mak Cyclophilin inhibitors and uses thereof
WO2021190603A1 (en) * 2020-03-26 2021-09-30 Farsight Medical Technology (Shanghai) Co., Ltd. Cyclophilin inhibitors and uses thereof
EP4251189A1 (en) * 2020-11-29 2023-10-04 Hepion Pharmaceuticals, Inc. Use of cyclosporine analogues as antithrombotic agents
CN113173974B (zh) 2021-03-18 2024-09-06 北京大学深圳研究生院 环孢素衍生物的合成方法
CN115677533B (zh) * 2021-07-30 2023-12-05 沈阳化工研究院有限公司 一种4-庚基苯甲腈的制备方法
IT202300001116A1 (it) * 2023-01-25 2024-07-25 Indena Spa Processo per la preparazione di un intermedio utile per la sintesi di voclosporina
WO2024245384A1 (en) * 2023-06-02 2024-12-05 Farsight Medical Technology (Shanghai) Co., Ltd. Cyclophilin inhibitors and uses thereof
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