JP2013526596A5 - - Google Patents

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Publication number
JP2013526596A5
JP2013526596A5 JP2013511631A JP2013511631A JP2013526596A5 JP 2013526596 A5 JP2013526596 A5 JP 2013526596A5 JP 2013511631 A JP2013511631 A JP 2013511631A JP 2013511631 A JP2013511631 A JP 2013511631A JP 2013526596 A5 JP2013526596 A5 JP 2013526596A5
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treatment
pain
hereinafter
diseases
found
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JP2013511631A
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Japanese (ja)
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JP5636094B2 (ja
JP2013526596A (ja
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Priority claimed from PCT/EP2011/058355 external-priority patent/WO2011147772A1/en
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Publication of JP2013526596A5 publication Critical patent/JP2013526596A5/ja
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JP2013511631A 2010-05-25 2011-05-23 Ccr2受容体アンタゴニスト Active JP5636094B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10163848 2010-05-25
EP10163848.4 2010-05-25
PCT/EP2011/058355 WO2011147772A1 (en) 2010-05-25 2011-05-23 Ccr2 receptor antagonists

Publications (3)

Publication Number Publication Date
JP2013526596A JP2013526596A (ja) 2013-06-24
JP2013526596A5 true JP2013526596A5 (enExample) 2014-10-30
JP5636094B2 JP5636094B2 (ja) 2014-12-03

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ID=43216431

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JP2013511631A Active JP5636094B2 (ja) 2010-05-25 2011-05-23 Ccr2受容体アンタゴニスト

Country Status (4)

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US (1) US9018212B2 (enExample)
EP (1) EP2576542B1 (enExample)
JP (1) JP5636094B2 (enExample)
WO (1) WO2011147772A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5603770B2 (ja) 2007-05-31 2014-10-08 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ccr2受容体拮抗薬およびその使用
CN102256963B (zh) 2008-12-19 2014-06-11 贝林格尔.英格海姆国际有限公司 作为ccr2受体拮抗剂用于治疗炎症、哮喘和copd的环状嘧啶-4-甲酰胺
ES2674275T3 (es) 2009-12-17 2018-06-28 Centrexion Therapeutics Corporation Antagonistas del receptor CCR2 y usos de los mismos
JP5646736B2 (ja) 2010-05-12 2014-12-24 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ccr2受容体アンタゴニスト、これらの製造方法、及び薬物としてのこれらの使用
WO2011141474A1 (en) 2010-05-12 2011-11-17 Boehringer Ingelheim International Gmbh Novel ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments
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WO2011147772A1 (en) 2010-05-25 2011-12-01 Boehringer Ingelheim International Gmbh Ccr2 receptor antagonists
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EP2731941B1 (en) 2011-07-15 2019-05-08 Boehringer Ingelheim International GmbH Novel and selective ccr2 antagonists
PT3317270T (pt) 2015-07-02 2020-08-24 Centrexion Therapeutics Corp (4-((3r,4r)-3-metoxitetrahidro-pirano-4-ilamino)piperidina-1-il)(5-metil-6-(((2r,6s)-6-(p-tolil)tetrahidro-2h-pirano-2-il)metilamino)pirimidina-4-il)citrato de metanona

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JP5646736B2 (ja) 2010-05-12 2014-12-24 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ccr2受容体アンタゴニスト、これらの製造方法、及び薬物としてのこれらの使用
WO2011144501A1 (en) 2010-05-17 2011-11-24 Boehringer Ingelheim International Gmbh Ccr2 antagonists and uses thereof
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WO2012171863A1 (en) 2011-06-16 2012-12-20 Boehringer Ingelheim International Gmbh New selective ccr2 antagonists
EP2731941B1 (en) 2011-07-15 2019-05-08 Boehringer Ingelheim International GmbH Novel and selective ccr2 antagonists

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