JP2013525264A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2013525264A5 JP2013525264A5 JP2012549043A JP2012549043A JP2013525264A5 JP 2013525264 A5 JP2013525264 A5 JP 2013525264A5 JP 2012549043 A JP2012549043 A JP 2012549043A JP 2012549043 A JP2012549043 A JP 2012549043A JP 2013525264 A5 JP2013525264 A5 JP 2013525264A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound represented
- group
- manufacturing
- production method
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- YZDLKGSISFGIRU-UHFFFAOYSA-N C(C1C(C2)CCCC1)[N]2(CC1)CCN1c1n[s]c2ccccc12 Chemical compound C(C1C(C2)CCCC1)[N]2(CC1)CCN1c1n[s]c2ccccc12 YZDLKGSISFGIRU-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US32780910P | 2010-04-26 | 2010-04-26 | |
| US61/327,809 | 2010-04-26 | ||
| PCT/JP2011/060570 WO2011136383A1 (en) | 2010-04-26 | 2011-04-25 | A process of a quaternary ammonium salt |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013525264A JP2013525264A (ja) | 2013-06-20 |
| JP2013525264A5 true JP2013525264A5 (enExample) | 2014-05-22 |
| JP5820821B2 JP5820821B2 (ja) | 2015-11-24 |
Family
ID=44816340
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012549043A Active JP5820821B2 (ja) | 2010-04-26 | 2011-04-25 | 第四級アンモニウム塩の製造法 |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US8921551B2 (enExample) |
| EP (1) | EP2563790B1 (enExample) |
| JP (1) | JP5820821B2 (enExample) |
| DK (1) | DK2563790T3 (enExample) |
| ES (1) | ES2594709T3 (enExample) |
| HU (1) | HUE030294T2 (enExample) |
| WO (1) | WO2011136383A1 (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5820822B2 (ja) * | 2010-04-26 | 2015-11-24 | 大日本住友製薬株式会社 | リン酸塩を用いる第四級アンモニウム塩の製造法 |
| US9409899B2 (en) | 2012-02-13 | 2016-08-09 | Cadila Healthcare Limited | Process for preparing benzisothiazol-3-yl-piperazin-1-yl-methyl-cyclo hexylmethanisoindol-1,3-dione and its intermediates |
| CN103450172A (zh) * | 2012-05-30 | 2013-12-18 | 广州药源生物医药科技有限公司 | 一种抗精神病药物鲁拉西酮的制备方法 |
| CN102863437A (zh) * | 2012-09-04 | 2013-01-09 | 济南百诺医药科技开发有限公司 | 一种鲁拉西酮的制备方法 |
| CN102827157A (zh) * | 2012-09-20 | 2012-12-19 | 北京哈三联科技股份有限公司 | 一种制备鲁拉西酮的方法 |
| CN102936243B (zh) * | 2012-11-16 | 2015-08-05 | 上海伯倚化工科技有限公司 | 一种鲁拉西酮的合成方法 |
| CN103864774B (zh) * | 2012-12-14 | 2016-09-28 | 成都弘达药业有限公司 | 一种鲁拉西酮的制备方法 |
| ITMI20130262A1 (it) * | 2013-02-22 | 2014-08-23 | Edmond Pharma Srl | Procedimento per la preparazione di lurasidone cloridrato |
| ITMI20131737A1 (it) | 2013-10-17 | 2015-04-18 | Procos Spa | Processo per la sintesi industriale di lurasidone |
| JP6594351B2 (ja) | 2014-06-16 | 2019-10-23 | ジョンソン、マッセイ、パブリック、リミテッド、カンパニー | 新規中間体を含むアルキル化アリールピペラジン及びアルキル化アリールピペリジン化合物の製造方法 |
| US10426770B2 (en) | 2014-10-14 | 2019-10-01 | Jubilant Generics Limited | Process for the preparation of Lurasidone hydrochloride |
| EP3242876A4 (en) * | 2015-01-08 | 2019-01-02 | Piramal Enterprises Limited | An improved process for the preparation of lurasidone and its intermediate |
| CN113185508A (zh) * | 2015-04-21 | 2021-07-30 | 上海医药集团股份有限公司 | 一种制备高纯度高收率鲁拉西酮的方法 |
| CN106946872A (zh) * | 2017-03-20 | 2017-07-14 | 常州工程职业技术学院 | 一种制备鲁拉西酮关键中间体的方法 |
| CN107936007B (zh) * | 2017-11-28 | 2021-05-25 | 常州寅盛药业有限公司 | 一种盐酸鲁拉西酮的合成方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4351939A (en) * | 1980-10-16 | 1982-09-28 | Mead Johnson & Company | Spiro-quaternary ammonium halides and N-(2-pyrimidinyl)piperazinylalkylazaspiroalkanedione process |
| JP2800953B2 (ja) * | 1990-07-06 | 1998-09-21 | 住友製薬株式会社 | 新規なイミド誘導体 |
| JP3775823B2 (ja) * | 1995-06-09 | 2006-05-17 | 大日本住友製薬株式会社 | 新規なイミド誘導体 |
| JP4175800B2 (ja) * | 2001-11-27 | 2008-11-05 | 住友化学株式会社 | イミド誘導体の製造方法 |
| KR101085806B1 (ko) | 2003-07-29 | 2011-11-22 | 다이닛본 스미토모 세이야꾸 가부시끼가이샤 | 이미드 화합물의 제조 방법 |
| JP2006169154A (ja) * | 2004-12-15 | 2006-06-29 | Sumitomo Chemical Co Ltd | 第四級アンモニウム塩の製造方法 |
| JP4708012B2 (ja) * | 2004-12-15 | 2011-06-22 | 大日本住友製薬株式会社 | 第四級アンモニウム塩の製造法 |
| EP1919922B1 (en) | 2005-08-30 | 2011-04-20 | Honeywell International Inc. | Method for synthesizing spiro quaternary ammonium systems |
| US20110003994A1 (en) * | 2009-07-02 | 2011-01-06 | Dainippon Sumitomo Pharma Co., Ltd. | Cycloalkane derivative |
| JP5820822B2 (ja) * | 2010-04-26 | 2015-11-24 | 大日本住友製薬株式会社 | リン酸塩を用いる第四級アンモニウム塩の製造法 |
-
2011
- 2011-04-25 ES ES11775164.4T patent/ES2594709T3/es active Active
- 2011-04-25 JP JP2012549043A patent/JP5820821B2/ja active Active
- 2011-04-25 DK DK11775164.4T patent/DK2563790T3/en active
- 2011-04-25 EP EP11775164.4A patent/EP2563790B1/en active Active
- 2011-04-25 HU HUE11775164A patent/HUE030294T2/en unknown
- 2011-04-25 WO PCT/JP2011/060570 patent/WO2011136383A1/en not_active Ceased
- 2011-04-26 US US13/093,927 patent/US8921551B2/en active Active
-
2014
- 2014-11-07 US US14/536,118 patent/US9309255B2/en active Active
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2013525264A5 (enExample) | ||
| JP2013525265A5 (enExample) | ||
| RU2012138259A (ru) | Способ получения ривароксабана | |
| CN102675101B (zh) | 2-(4-卤乙基)苯基-2-甲基丙酸酯的制备方法及合成比拉斯汀的方法 | |
| JP2018528182A5 (enExample) | ||
| JP2014521744A5 (enExample) | ||
| EA201170096A1 (ru) | Замещенные производные пиримидона | |
| WO2010146176A3 (en) | Process for hydrogenation of halogenoalkenes without dehalogenation | |
| JP2014094926A5 (enExample) | ||
| JP2014520901A (ja) | ４−置換イミダゾールの新規な調製プロセス | |
| Xu et al. | K2S2O8-mediated hydroxyalkylation of benzothiazoles with alcohols in aqueous solution | |
| JP2010505861A5 (enExample) | ||
| Murauski et al. | A Cooperative Ternary Catalysis System for Asymmetric Lactonizations of α‐Ketoesters | |
| RU2014129937A (ru) | Способы и промежуточные соединения для получения фармацевтических агентов | |
| EA201490998A1 (ru) | Способ получения сложных эфиров (5-фтор-2-метил-3-хинолин-2-илметил-индол-1-ил)-уксусной кислоты | |
| CN109020919B (zh) | 一种制备药用活性化合物n-取代苯并噻嗪-4-酮的方法 | |
| CN105198841B (zh) | 一种药物中间体多取代呋喃类化合物的合成方法 | |
| JP2016138105A5 (enExample) | ||
| RU2013148907A (ru) | Способ | |
| RU2016146552A (ru) | Раствор галогенида магния и способ его получения и его применение | |
| JP2018115129A5 (enExample) | ||
| JP2018505179A5 (enExample) | ||
| CN105152827A (zh) | 芳基磺酸酯类底物与有机钛的交叉偶联反应 | |
| CY1117612T1 (el) | Μια μεθοδος για την παρασκευη του εστερα της σκοπινης του δι-(2-θειενυλο)γλυκολικου οξεος, μιας ενδιαμεσης ενωσης στη συνθεση του βρωμιουχου τιοτροπιου | |
| JP2016150950A5 (enExample) |