JP2013508456A5 - - Google Patents
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- Publication number
- JP2013508456A5 JP2013508456A5 JP2012536897A JP2012536897A JP2013508456A5 JP 2013508456 A5 JP2013508456 A5 JP 2013508456A5 JP 2012536897 A JP2012536897 A JP 2012536897A JP 2012536897 A JP2012536897 A JP 2012536897A JP 2013508456 A5 JP2013508456 A5 JP 2013508456A5
- Authority
- JP
- Japan
- Prior art keywords
- dihydropyrazino
- pyrazin
- methyl
- triazol
- pyridin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25491709P | 2009-10-26 | 2009-10-26 | |
| US61/254,917 | 2009-10-26 | ||
| US32848010P | 2010-04-27 | 2010-04-27 | |
| US61/328,480 | 2010-04-27 | ||
| PCT/US2010/053678 WO2011053518A1 (en) | 2009-10-26 | 2010-10-22 | Methods of synthesis and purification of heteroaryl compounds |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016148782A Division JP6338622B2 (ja) | 2009-10-26 | 2016-07-28 | ヘテロアリール化合物の合成方法および精製方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013508456A JP2013508456A (ja) | 2013-03-07 |
| JP2013508456A5 true JP2013508456A5 (https=) | 2013-11-07 |
Family
ID=43922466
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012536897A Pending JP2013508456A (ja) | 2009-10-26 | 2010-10-22 | ヘテロアリール化合物の合成方法および精製方法 |
| JP2016148782A Active JP6338622B2 (ja) | 2009-10-26 | 2016-07-28 | ヘテロアリール化合物の合成方法および精製方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016148782A Active JP6338622B2 (ja) | 2009-10-26 | 2016-07-28 | ヘテロアリール化合物の合成方法および精製方法 |
Country Status (23)
| Country | Link |
|---|---|
| US (3) | US8569494B2 (https=) |
| EP (2) | EP2493472B1 (https=) |
| JP (2) | JP2013508456A (https=) |
| KR (2) | KR101903925B1 (https=) |
| CN (2) | CN106117213B (https=) |
| AR (1) | AR078788A1 (https=) |
| AU (1) | AU2010313585B2 (https=) |
| BR (1) | BR112012009751A2 (https=) |
| CA (1) | CA2778615C (https=) |
| CO (1) | CO6541598A2 (https=) |
| CR (1) | CR20120211A (https=) |
| EC (1) | ECSP12011831A (https=) |
| ES (2) | ES2751705T3 (https=) |
| IL (1) | IL219368A (https=) |
| MX (1) | MX341704B (https=) |
| MY (1) | MY177695A (https=) |
| NI (1) | NI201200066A (https=) |
| NZ (2) | NZ618135A (https=) |
| PH (2) | PH12012500825A1 (https=) |
| RU (1) | RU2557242C2 (https=) |
| SG (1) | SG10201500511TA (https=) |
| WO (1) | WO2011053518A1 (https=) |
| ZA (1) | ZA201202959B (https=) |
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| CN115135636B (zh) * | 2020-04-29 | 2024-08-23 | 北京泰德制药股份有限公司 | 喹喔啉酮衍生物作为kras g12c突变蛋白的不可逆抑制剂 |
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