JP2013508456A5 - - Google Patents

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Publication number
JP2013508456A5
JP2013508456A5 JP2012536897A JP2012536897A JP2013508456A5 JP 2013508456 A5 JP2013508456 A5 JP 2013508456A5 JP 2012536897 A JP2012536897 A JP 2012536897A JP 2012536897 A JP2012536897 A JP 2012536897A JP 2013508456 A5 JP2013508456 A5 JP 2013508456A5
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JP
Japan
Prior art keywords
dihydropyrazino
pyrazin
methyl
triazol
pyridin
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012536897A
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English (en)
Japanese (ja)
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JP2013508456A (ja
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Priority claimed from PCT/US2010/053678 external-priority patent/WO2011053518A1/en
Publication of JP2013508456A publication Critical patent/JP2013508456A/ja
Publication of JP2013508456A5 publication Critical patent/JP2013508456A5/ja
Pending legal-status Critical Current

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JP2012536897A 2009-10-26 2010-10-22 ヘテロアリール化合物の合成方法および精製方法 Pending JP2013508456A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US25491709P 2009-10-26 2009-10-26
US61/254,917 2009-10-26
US32848010P 2010-04-27 2010-04-27
US61/328,480 2010-04-27
PCT/US2010/053678 WO2011053518A1 (en) 2009-10-26 2010-10-22 Methods of synthesis and purification of heteroaryl compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016148782A Division JP6338622B2 (ja) 2009-10-26 2016-07-28 ヘテロアリール化合物の合成方法および精製方法

Publications (2)

Publication Number Publication Date
JP2013508456A JP2013508456A (ja) 2013-03-07
JP2013508456A5 true JP2013508456A5 (https=) 2013-11-07

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JP2012536897A Pending JP2013508456A (ja) 2009-10-26 2010-10-22 ヘテロアリール化合物の合成方法および精製方法
JP2016148782A Active JP6338622B2 (ja) 2009-10-26 2016-07-28 ヘテロアリール化合物の合成方法および精製方法

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JP2016148782A Active JP6338622B2 (ja) 2009-10-26 2016-07-28 ヘテロアリール化合物の合成方法および精製方法

Country Status (23)

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US (3) US8569494B2 (https=)
EP (2) EP2493472B1 (https=)
JP (2) JP2013508456A (https=)
KR (2) KR101903925B1 (https=)
CN (2) CN106117213B (https=)
AR (1) AR078788A1 (https=)
AU (1) AU2010313585B2 (https=)
BR (1) BR112012009751A2 (https=)
CA (1) CA2778615C (https=)
CO (1) CO6541598A2 (https=)
CR (1) CR20120211A (https=)
EC (1) ECSP12011831A (https=)
ES (2) ES2751705T3 (https=)
IL (1) IL219368A (https=)
MX (1) MX341704B (https=)
MY (1) MY177695A (https=)
NI (1) NI201200066A (https=)
NZ (2) NZ618135A (https=)
PH (2) PH12012500825A1 (https=)
RU (1) RU2557242C2 (https=)
SG (1) SG10201500511TA (https=)
WO (1) WO2011053518A1 (https=)
ZA (1) ZA201202959B (https=)

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CA2744498C (en) 2008-11-25 2017-10-24 University Of Rochester Mlk inhibitors and methods of use

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