JP2013503901A5 - - Google Patents

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Publication number
JP2013503901A5
JP2013503901A5 JP2012528084A JP2012528084A JP2013503901A5 JP 2013503901 A5 JP2013503901 A5 JP 2013503901A5 JP 2012528084 A JP2012528084 A JP 2012528084A JP 2012528084 A JP2012528084 A JP 2012528084A JP 2013503901 A5 JP2013503901 A5 JP 2013503901A5
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JP
Japan
Prior art keywords
group
amino
pyridin
methyl
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2012528084A
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English (en)
Japanese (ja)
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JP2013503901A (ja
JP5868855B2 (ja
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Publication date
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Priority claimed from PCT/US2010/047800 external-priority patent/WO2011028995A1/en
Publication of JP2013503901A publication Critical patent/JP2013503901A/ja
Publication of JP2013503901A5 publication Critical patent/JP2013503901A5/ja
Application granted granted Critical
Publication of JP5868855B2 publication Critical patent/JP5868855B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012528084A 2009-09-03 2010-09-03 チロシンキナーゼ調節剤としての化合物 Expired - Fee Related JP5868855B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US23960309P 2009-09-03 2009-09-03
US61/239,603 2009-09-03
US30661610P 2010-02-22 2010-02-22
US61/306,616 2010-02-22
US35669910P 2010-06-21 2010-06-21
US61/356,699 2010-06-21
US36053110P 2010-07-01 2010-07-01
US61/360,531 2010-07-01
PCT/US2010/047800 WO2011028995A1 (en) 2009-09-03 2010-09-03 Compounds as tyrosine kinase modulators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016001387A Division JP6109974B2 (ja) 2009-09-03 2016-01-06 チロシンキナーゼ調節剤としての化合物

Publications (3)

Publication Number Publication Date
JP2013503901A JP2013503901A (ja) 2013-02-04
JP2013503901A5 true JP2013503901A5 (enExample) 2013-10-24
JP5868855B2 JP5868855B2 (ja) 2016-02-24

Family

ID=43086186

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2012528089A Pending JP2013503903A (ja) 2009-09-03 2010-09-03 チロシンキナーゼモジュレーターとしての化合物
JP2012528084A Expired - Fee Related JP5868855B2 (ja) 2009-09-03 2010-09-03 チロシンキナーゼ調節剤としての化合物
JP2016001387A Expired - Fee Related JP6109974B2 (ja) 2009-09-03 2016-01-06 チロシンキナーゼ調節剤としての化合物

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2012528089A Pending JP2013503903A (ja) 2009-09-03 2010-09-03 チロシンキナーゼモジュレーターとしての化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2016001387A Expired - Fee Related JP6109974B2 (ja) 2009-09-03 2016-01-06 チロシンキナーゼ調節剤としての化合物

Country Status (19)

Country Link
US (5) US8614234B2 (enExample)
EP (2) EP2473513B1 (enExample)
JP (3) JP2013503903A (enExample)
KR (2) KR20120047313A (enExample)
CN (2) CN102498114A (enExample)
AU (2) AU2010289359A1 (enExample)
BR (2) BR112012004718A2 (enExample)
CA (2) CA2772718C (enExample)
CL (2) CL2012000587A1 (enExample)
ES (1) ES2730086T3 (enExample)
IL (2) IL218332A0 (enExample)
IN (1) IN2012DN02493A (enExample)
MX (2) MX2012002591A (enExample)
NZ (2) NZ598455A (enExample)
PH (1) PH12014500281A1 (enExample)
RU (2) RU2012112151A (enExample)
SG (2) SG178963A1 (enExample)
WO (2) WO2011028995A1 (enExample)
ZA (2) ZA201201592B (enExample)

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WO2017040853A1 (en) 2015-09-02 2017-03-09 Glaukos Corporation Drug delivery implants with bi-directional delivery capacity
US11564833B2 (en) 2015-09-25 2023-01-31 Glaukos Corporation Punctal implants with controlled drug delivery features and methods of using same
CN107531679B (zh) * 2016-03-18 2021-07-02 江苏恒瑞医药股份有限公司 芳香酰胺类衍生物、其制备方法及其在医药上的应用
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CN107663202B (zh) * 2016-07-29 2020-09-04 西华大学 3-(脲基-甲基)-4-芳基-吡啶衍生物及其制备方法和作为抗肝癌药物的应用
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LT3860998T (lt) 2018-10-05 2024-06-25 Annapurna Bio Inc. Junginiai ir kompozicijos, skirti gydyti būkles, susijusias su apj receptoriaus aktyvumu
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9902709B2 (en) 2014-04-08 2018-02-27 Peking University Founder Group Co., Ltd. Polysubstituted pyridine compound, preparation method, use and pharmaceutical composition

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