JP2013500977A5 - - Google Patents

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Publication number
JP2013500977A5
JP2013500977A5 JP2012523011A JP2012523011A JP2013500977A5 JP 2013500977 A5 JP2013500977 A5 JP 2013500977A5 JP 2012523011 A JP2012523011 A JP 2012523011A JP 2012523011 A JP2012523011 A JP 2012523011A JP 2013500977 A5 JP2013500977 A5 JP 2013500977A5
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JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
pharmaceutical composition
acceptable salt
salt form
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JP2012523011A
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English (en)
Japanese (ja)
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JP2013500977A (ja
JP5738292B2 (ja
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Priority claimed from PCT/US2010/043592 external-priority patent/WO2011017178A1/en
Publication of JP2013500977A publication Critical patent/JP2013500977A/ja
Publication of JP2013500977A5 publication Critical patent/JP2013500977A5/ja
Application granted granted Critical
Publication of JP5738292B2 publication Critical patent/JP5738292B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012523011A 2009-07-28 2010-07-28 Jak経路の阻害のための組成物および方法 Expired - Fee Related JP5738292B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22919109P 2009-07-28 2009-07-28
US61/229,191 2009-07-28
PCT/US2010/043592 WO2011017178A1 (en) 2009-07-28 2010-07-28 Compositions and methods for inhibition of the jak pathway

Publications (3)

Publication Number Publication Date
JP2013500977A JP2013500977A (ja) 2013-01-10
JP2013500977A5 true JP2013500977A5 (enExample) 2013-09-12
JP5738292B2 JP5738292B2 (ja) 2015-06-24

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ID=42676842

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012523011A Expired - Fee Related JP5738292B2 (ja) 2009-07-28 2010-07-28 Jak経路の阻害のための組成物および方法

Country Status (11)

Country Link
US (1) US20110028503A1 (enExample)
EP (1) EP2459195A1 (enExample)
JP (1) JP5738292B2 (enExample)
KR (1) KR101740076B1 (enExample)
CN (2) CN102470135A (enExample)
AU (3) AU2010281404A1 (enExample)
BR (1) BR112012002001A2 (enExample)
CA (1) CA2768543C (enExample)
MX (1) MX337849B (enExample)
RU (1) RU2557982C2 (enExample)
WO (1) WO2011017178A1 (enExample)

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JP6427497B2 (ja) * 2013-10-21 2018-11-21 日本たばこ産業株式会社 眼疾患の治療剤又は予防剤
KR20180073687A (ko) 2015-11-03 2018-07-02 세라밴스 바이오파마 알앤디 아이피, 엘엘씨 호흡기 질환의 치료를 위한 jak 키나제 저해제 화합물
SG11201909019SA (en) 2017-05-01 2019-10-30 Theravance Biopharma R&D Ip Llc Methods of treatment using a jak inhibitor compound
CN107805212B (zh) * 2017-11-03 2021-08-20 宿迁德威化工股份有限公司 一种2-甲基-5-氨基苯磺酰胺的制备方法
BR112022001418A2 (pt) 2019-08-08 2022-06-07 Rigel Pharmaceuticals Inc Compostos e método para tratar a síndrome de liberação de citocinas
CN111973599A (zh) * 2020-08-07 2020-11-24 杭州邦顺制药有限公司 用于眼部疾病治疗的化合物
TW202317550A (zh) 2021-06-25 2023-05-01 美商施萬生物製藥研發 Ip有限責任公司 作為jak抑制劑之咪唑吲唑化合物

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