JP2012527442A5 - - Google Patents

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Publication number
JP2012527442A5
JP2012527442A5 JP2012511355A JP2012511355A JP2012527442A5 JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5 JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012511355 A JP2012511355 A JP 2012511355A JP 2012527442 A5 JP2012527442 A5 JP 2012527442A5
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JP
Japan
Prior art keywords
salt
diffraction pattern
pharmaceutical composition
powder diffraction
ray powder
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JP2012511355A
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English (en)
Japanese (ja)
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JP5717727B2 (ja
JP2012527442A (ja
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Priority claimed from GBGB0908772.7A external-priority patent/GB0908772D0/en
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Publication of JP2012527442A publication Critical patent/JP2012527442A/ja
Publication of JP2012527442A5 publication Critical patent/JP2012527442A5/ja
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Publication of JP5717727B2 publication Critical patent/JP5717727B2/ja
Expired - Fee Related legal-status Critical Current
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JP2012511355A 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩 Expired - Fee Related JP5717727B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0908772.7 2009-05-21
GBGB0908772.7A GB0908772D0 (en) 2009-05-21 2009-05-21 New salts 756
PCT/GB2010/050822 WO2010133882A1 (en) 2009-05-21 2010-05-20 Disaccharin, difumaric acid, di-l-hydroxy-2-naphthoic acid and mono-benzoic acid salts of 4- (dimethylamin0)butyl 2- (4- ( (2-amino-4-methyl-6- (pentylamino) pyrimidin- 5 -yl) methyl) phenyl)acetate

Publications (3)

Publication Number Publication Date
JP2012527442A JP2012527442A (ja) 2012-11-08
JP2012527442A5 true JP2012527442A5 (https=) 2013-07-04
JP5717727B2 JP5717727B2 (ja) 2015-05-13

Family

ID=40862774

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012511355A Expired - Fee Related JP5717727B2 (ja) 2009-05-21 2010-05-20 ２−（４−（（２−アミノ−４−メチル−６−（ペンチルアミノ）ピリミジン−５−イル）メチル）フェニル）酢酸４−（ジメチルアミノ）ブチルの二サッカリン塩、二フマル酸塩、二ｌ−ヒドロキシ−２−ナフトエ酸塩および一安息香酸塩

Country Status (30)

Country Link
US (1) US8476288B2 (https=)
EP (1) EP2435412B1 (https=)
JP (1) JP5717727B2 (https=)
KR (1) KR101709363B1 (https=)
CN (1) CN102596917B (https=)
AR (1) AR076597A1 (https=)
AU (1) AU2010250920B2 (https=)
BR (1) BRPI1012198A8 (https=)
CA (1) CA2760765A1 (https=)
CL (1) CL2011002941A1 (https=)
CO (1) CO6440532A2 (https=)
CR (1) CR20110611A (https=)
CU (1) CU24053B1 (https=)
DO (1) DOP2011000360A (https=)
EA (1) EA021854B1 (https=)
EC (1) ECSP11011469A (https=)
ES (1) ES2566912T3 (https=)
GB (1) GB0908772D0 (https=)
HN (1) HN2011003072A (https=)
IL (1) IL216280A0 (https=)
MX (1) MX2011012344A (https=)
NI (1) NI201100205A (https=)
NZ (1) NZ596118A (https=)
PE (1) PE20120989A1 (https=)
SA (1) SA110310402B1 (https=)
SG (1) SG175322A1 (https=)
TW (1) TW201100389A (https=)
UY (1) UY32649A (https=)
WO (1) WO2010133882A1 (https=)
ZA (1) ZA201109383B (https=)

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TWI619704B (zh) 2012-05-18 2018-04-01 大日本住友製藥股份有限公司 羧酸化合物
PT3166607T (pt) 2014-07-11 2022-12-07 Gilead Sciences Inc Moduladores de receptores de tipo toll para o tratamento do vih
CA2960436C (en) 2014-09-16 2021-01-05 Gilead Sciences, Inc. Solid forms of a toll-like receptor modulator
RU2748833C2 (ru) 2016-11-28 2021-05-31 Цзянсу Хэнжуй Медсин Ко., Лтд. Производное пиразоло-гетероарила, способ его получения и медицинское применение
EP3636646A4 (en) 2017-05-18 2020-12-09 Jiangsu Hengrui Medicine Co., Ltd. HETEROARYL PYRAZOL DERIVATIVE AND MANUFACTURING METHOD FOR IT AND MEDICAL USES THEREOF
CN111819178B (zh) 2018-05-25 2022-04-12 江苏恒瑞医药股份有限公司 一种吡唑并杂芳基类衍生物盐酸盐的晶型及制备方法

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