JP2012519160A - Ｐｄｅ４阻害剤及びｎｓａｉｄを含有する組み合わせ薬 - Google Patents
Ｐｄｅ４阻害剤及びｎｓａｉｄを含有する組み合わせ薬 Download PDFInfo
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- JP2012519160A JP2012519160A JP2011551465A JP2011551465A JP2012519160A JP 2012519160 A JP2012519160 A JP 2012519160A JP 2011551465 A JP2011551465 A JP 2011551465A JP 2011551465 A JP2011551465 A JP 2011551465A JP 2012519160 A JP2012519160 A JP 2012519160A
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- methyl
- ethyl
- oxo
- hetaryl
- methylene
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- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 claims description 14
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| PCT/EP2010/052079 WO2010097334A1 (de) | 2009-02-27 | 2010-02-18 | Arzneimittelkombinationen enthaltend pde4-inhibitoren und nsaids |
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012519159A (ja) * | 2009-02-27 | 2012-08-23 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｐｄｅ４阻害剤及びｎｓａｉｄを含有する複合薬 |
| JP2016505512A (ja) * | 2012-10-25 | 2016-02-25 | テトラ ディスカバリー パートナーズ エルエルシー | Ｐｄｅ４のヘテロアリール阻害剤 |
| JP2018507236A (ja) * | 2015-03-04 | 2018-03-15 | エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ | トリアゾロピリジン化合物及びその使用法 |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1847543A1 (de) | 2006-04-19 | 2007-10-24 | Boehringer Ingelheim Pharma GmbH & Co. KG | Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen |
| RU2500681C2 (ru) | 2007-10-19 | 2013-12-10 | Берингер Ингельхайм Интернациональ Гмбх | Замещенные гетероциклом пиперазинодигидротиенопиримидины |
| EP2215093B1 (de) | 2007-10-19 | 2011-12-14 | Boehringer Ingelheim International GmbH | Neue piperazino-dihydrothienopyrimidin-derivate |
| SI2610258T1 (sl) * | 2007-10-19 | 2014-12-31 | Boehringer Ingelheim International Gmbh | Substituirani piperidino-dihidrotienopirimidini |
| ES2523169T3 (es) | 2008-01-25 | 2014-11-21 | High Point Pharmaceuticals, Llc | Compuestos tricíclicos como moduladores de la síntesis de TNF y como inhibidores de PDE4 |
| GB2477590A (en) * | 2010-02-05 | 2011-08-10 | Biocopea Ltd | A non-steroidal anti-inflammatory drug (NSAID) formulation comprising a lipid carrier |
| US11730709B2 (en) | 2010-10-29 | 2023-08-22 | Infirst Healthcare Limited | Compositions and methods for treating severe pain |
| US11202831B2 (en) | 2010-10-29 | 2021-12-21 | Infirst Healthcare Limited | Solid solution compositions and use in cardiovascular disease |
| US9737500B2 (en) | 2010-10-29 | 2017-08-22 | Infirst Healthcare Limited | Compositions and methods for treating severe pain |
| US9271950B2 (en) | 2010-10-29 | 2016-03-01 | Infirst Healthcare Limited | Compositions for treating chronic inflammation and inflammatory diseases |
| US10695432B2 (en) | 2010-10-29 | 2020-06-30 | Infirst Healthcare Limited | Solid solution compositions and use in severe pain |
| US9308213B2 (en) | 2010-10-29 | 2016-04-12 | Infirst Healthcare Limited | Solid solution compositions and use in chronic inflammation |
| US9744132B2 (en) | 2010-10-29 | 2017-08-29 | Infirst Healthcare Limited | Solid solution compositions and use in chronic inflammation |
| US11224659B2 (en) | 2010-10-29 | 2022-01-18 | Infirst Healthcare Limited | Solid solution compositions and use in severe pain |
| US8895537B2 (en) | 2010-10-29 | 2014-11-25 | Infirst Healthcare Ltd. | Compositions and methods for treating cardiovascular diseases |
| US9504664B2 (en) | 2010-10-29 | 2016-11-29 | Infirst Healthcare Limited | Compositions and methods for treating severe pain |
| US10695431B2 (en) | 2010-10-29 | 2020-06-30 | Infirst Healthcare Limited | Solid solution compositions and use in cardiovascular disease |
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| US10626129B2 (en) | 2012-10-25 | 2020-04-21 | Tetra Discovery Partners, LLC | Heteroaryl inhibitors of PDE4 |
| JP2018507236A (ja) * | 2015-03-04 | 2018-03-15 | エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ | トリアゾロピリジン化合物及びその使用法 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2400962B1 (de) | 2017-11-08 |
| WO2010097334A1 (de) | 2010-09-02 |
| US9161927B2 (en) | 2015-10-20 |
| US20120035143A1 (en) | 2012-02-09 |
| EP2400962A1 (de) | 2012-01-04 |
| CA2753604A1 (en) | 2010-09-02 |
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