JP2012505235A5 - - Google Patents

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Publication number
JP2012505235A5
JP2012505235A5 JP2011531168A JP2011531168A JP2012505235A5 JP 2012505235 A5 JP2012505235 A5 JP 2012505235A5 JP 2011531168 A JP2011531168 A JP 2011531168A JP 2011531168 A JP2011531168 A JP 2011531168A JP 2012505235 A5 JP2012505235 A5 JP 2012505235A5
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JP
Japan
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independently
heterocyclyl
nhc
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JP2011531168A
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Japanese (ja)
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JP2012505235A (ja
JP5560278B2 (ja
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Priority claimed from PCT/US2009/059968 external-priority patent/WO2010042699A1/en
Publication of JP2012505235A publication Critical patent/JP2012505235A/ja
Publication of JP2012505235A5 publication Critical patent/JP2012505235A5/ja
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Expired - Fee Related legal-status Critical Current
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JP2011531168A 2008-10-09 2009-10-08 キナーゼ阻害剤として有用なイミダゾピリダジンカルボニトリル Expired - Fee Related JP5560278B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10404508P 2008-10-09 2008-10-09
US61/104,045 2008-10-09
PCT/US2009/059968 WO2010042699A1 (en) 2008-10-09 2009-10-08 Imidazopyridazinecarbonitriles useful as kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2012505235A JP2012505235A (ja) 2012-03-01
JP2012505235A5 true JP2012505235A5 (enExample) 2012-08-09
JP5560278B2 JP5560278B2 (ja) 2014-07-23

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Family Applications (1)

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JP2011531168A Expired - Fee Related JP5560278B2 (ja) 2008-10-09 2009-10-08 キナーゼ阻害剤として有用なイミダゾピリダジンカルボニトリル

Country Status (27)

Country Link
US (3) US8252795B2 (enExample)
EP (1) EP2350081B1 (enExample)
JP (1) JP5560278B2 (enExample)
KR (1) KR20110075010A (enExample)
CN (1) CN102245609B (enExample)
AR (1) AR073818A1 (enExample)
AU (1) AU2009302360B2 (enExample)
BR (1) BRPI0920135A2 (enExample)
CA (1) CA2739782A1 (enExample)
CL (1) CL2011000777A1 (enExample)
CO (1) CO6361936A2 (enExample)
CY (1) CY1114539T1 (enExample)
DK (1) DK2350081T3 (enExample)
EA (1) EA018163B1 (enExample)
ES (1) ES2426951T3 (enExample)
HR (1) HRP20130787T1 (enExample)
IL (1) IL211693A (enExample)
MX (1) MX2011003304A (enExample)
NZ (1) NZ591712A (enExample)
PE (1) PE20110411A1 (enExample)
PL (1) PL2350081T3 (enExample)
PT (1) PT2350081E (enExample)
SI (1) SI2350081T1 (enExample)
SM (1) SMT201300109B (enExample)
TW (1) TWI491610B (enExample)
WO (1) WO2010042699A1 (enExample)
ZA (1) ZA201102423B (enExample)

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WO2017223432A1 (en) 2016-06-24 2017-12-28 Polaris Pharmaceuticals Ck2 inhibitors, compositions and methods thereof
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US11299494B2 (en) 2016-11-17 2022-04-12 Bristol-Myers Squibb Company Substituted imidazo[1,2-b]pyridazines as interleukin-23 and interferon-α modulators
SG11201908940UA (en) 2017-03-30 2019-10-30 Hoffmann La Roche Isoquinolines as inhibitors of hpk1
CA3079786A1 (en) 2017-10-24 2019-05-02 The Broad Institute, Inc. 4h-pyrrolo[3,2-c]pyridin-4-one derivatives
WO2019128871A1 (zh) 2017-12-29 2019-07-04 江苏中旗科技股份有限公司 N-烷基-n-氰基烷基苯甲酰胺类化合物及其应用
WO2019128872A1 (zh) 2017-12-29 2019-07-04 江苏中旗科技股份有限公司 一种具有杀虫活性的吡唑酰胺类化合物及其应用
CN109988150B (zh) 2017-12-29 2022-04-12 江苏中旗科技股份有限公司 N-烷基-n-氰基烷基苯甲酰胺类化合物及其应用
JP7377207B2 (ja) * 2018-01-29 2023-11-09 メルク パテント ゲーエムベーハー Gcn2阻害剤およびその使用
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JP7637630B2 (ja) 2019-03-19 2025-02-28 ベーリンガー インゲルハイム フェトメディカ ゲーエムベーハー 駆虫性アザベンゾチオフェンおよびアザベンゾフラン化合物
US20240307362A1 (en) 2019-04-24 2024-09-19 Bayer Aktiengesellschaft 4H-PYRROLO[3,2-c]PYRIDIN-4-ONE COMPOUNDS
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JP2024505284A (ja) 2021-02-03 2024-02-05 サノフイ イミダゾ[4,5-d]ピリダジンの誘導体、それらの製造およびそれらの治療用途
AR127495A1 (es) 2021-11-01 2024-01-31 Boehringer Ingelheim Vetmedica Gmbh Compuestos de pirrolopiridazina como antihelmínticos
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TWI491610B (zh) * 2008-10-09 2015-07-11 必治妥美雅史谷比公司 作為激酶抑制劑之咪唑并嗒腈

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