JP2011518190A5 - - Google Patents
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- JP2011518190A5 JP2011518190A5 JP2011505258A JP2011505258A JP2011518190A5 JP 2011518190 A5 JP2011518190 A5 JP 2011518190A5 JP 2011505258 A JP2011505258 A JP 2011505258A JP 2011505258 A JP2011505258 A JP 2011505258A JP 2011518190 A5 JP2011518190 A5 JP 2011518190A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- hydroxy
- alkyl
- alkylamino
- heteroaryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 CC(C)(C(CC[C@](C)(C1CC2)[C@](C)(CC[C@@]3(C4CC(C)(C)CC3)C(*3*)=O)[C@]43C2=O)[C@]1(C)C=*(S)[Zn])C=O Chemical compound CC(C)(C(CC[C@](C)(C1CC2)[C@](C)(CC[C@@]3(C4CC(C)(C)CC3)C(*3*)=O)[C@]43C2=O)[C@]1(C)C=*(S)[Zn])C=O 0.000 description 4
- RMYWYZJDSBWZHH-DWIAEPJOSA-N CC(C)(CC1)CC(C([C@@](C)(CC2)[C@](C)(CCC3C(C)(C)C4=O)C(C5)[C@@]3(C)C=C4C#N)C5=O)[C@]12C(NCC(F)(F)F)=O Chemical compound CC(C)(CC1)CC(C([C@@](C)(CC2)[C@](C)(CCC3C(C)(C)C4=O)C(C5)[C@@]3(C)C=C4C#N)C5=O)[C@]12C(NCC(F)(F)F)=O RMYWYZJDSBWZHH-DWIAEPJOSA-N 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US4633208P | 2008-04-18 | 2008-04-18 | |
| US61/046,332 | 2008-04-18 | ||
| US11133308P | 2008-11-04 | 2008-11-04 | |
| US61/111,333 | 2008-11-04 | ||
| PCT/US2009/041170 WO2009129545A1 (en) | 2008-04-18 | 2009-04-20 | Antioxidant inflammation modulators: oleanolic acid derivatives with saturation in the c-ring |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011518190A JP2011518190A (ja) | 2011-06-23 |
| JP2011518190A5 true JP2011518190A5 (enExample) | 2012-06-07 |
| JP5529850B2 JP5529850B2 (ja) | 2014-06-25 |
Family
ID=41726396
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011505258A Active JP5529850B2 (ja) | 2008-04-18 | 2009-04-20 | 抗酸化炎症モジュレーター:c環中に飽和を有するオレアノール酸誘導体 |
Country Status (15)
| Country | Link |
|---|---|
| US (6) | US7915402B2 (enExample) |
| EP (1) | EP2279197B1 (enExample) |
| JP (1) | JP5529850B2 (enExample) |
| KR (1) | KR101713140B1 (enExample) |
| CN (1) | CN102164941B (enExample) |
| AU (1) | AU2009237578C1 (enExample) |
| BR (1) | BRPI0911208B1 (enExample) |
| CO (1) | CO6311106A2 (enExample) |
| EA (1) | EA022588B1 (enExample) |
| IL (1) | IL208714A (enExample) |
| MX (1) | MX2010011437A (enExample) |
| NZ (1) | NZ588709A (enExample) |
| TW (1) | TWI442925B (enExample) |
| WO (1) | WO2009129545A1 (enExample) |
| ZA (1) | ZA201007590B (enExample) |
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| BRPI0911208B1 (pt) | 2008-04-18 | 2021-05-25 | Reata Pharmaceuticals, Inc | Compostos moduladores inflamatórios antioxidantes, seu uso, e composição farmacêutica |
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| CN102499925B (zh) * | 2011-10-21 | 2015-11-11 | 上海中医药大学 | 一种中性粒细胞弹性蛋白酶抑制剂 |
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| JP6211527B2 (ja) | 2011-12-01 | 2017-10-11 | ハンジョウ ベンシェン ファーマシューティカル シーオー., エルティーディー.Hangzhou Bensheng Pharmaceutical Co., Ltd. | 2−置換オレアノール酸誘導体、その調製方法及びその用途 |
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