JP2010535252A5 - - Google Patents
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- JP2010535252A5 JP2010535252A5 JP2010520219A JP2010520219A JP2010535252A5 JP 2010535252 A5 JP2010535252 A5 JP 2010535252A5 JP 2010520219 A JP2010520219 A JP 2010520219A JP 2010520219 A JP2010520219 A JP 2010520219A JP 2010535252 A5 JP2010535252 A5 JP 2010535252A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- diabetes
- type
- metabolic
- nachr agonist
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US95361307P | 2007-08-02 | 2007-08-02 | |
| US95361407P | 2007-08-02 | 2007-08-02 | |
| US95361007P | 2007-08-02 | 2007-08-02 | |
| US97165407P | 2007-09-12 | 2007-09-12 | |
| PCT/US2008/071893 WO2009018511A2 (en) | 2007-08-02 | 2008-08-01 | Alpha7 nachr agonists for treating or preventing metabolic disorders |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010535252A JP2010535252A (ja) | 2010-11-18 |
| JP2010535252A5 true JP2010535252A5 (OSRAM) | 2011-01-06 |
Family
ID=39945177
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010520219A Pending JP2010535252A (ja) | 2007-08-02 | 2008-08-01 | 代謝障害を治療または予防するためのα７ｎＡＣｈＲアゴニスト |
| JP2010520213A Active JP5358573B2 (ja) | 2007-08-02 | 2008-08-01 | （２ｓ，３ｒ）−ｎ−（２−（（３−ピリジニル）メチル）−１−アザビシクロ［２．２．２］オクタ−３−イル）ベンゾフラン−２−カルボキサミド、その新規塩形態およびその使用方法 |
| JP2013148087A Active JP5852611B2 (ja) | 2007-08-02 | 2013-07-17 | （２ｓ，３ｒ）−ｎ−（２−（（３−ピリジニル）メチル）−１−アザビシクロ［２．２．２］オクタ−３−イル）ベンゾフラン−２−カルボキサミド、その新規塩形態およびその使用方法 |
| JP2013148091A Active JP6106549B2 (ja) | 2007-08-02 | 2013-07-17 | （２ｓ，３ｒ）−ｎ−（２−（（３−ピリジニル）メチル）−１−アザビシクロ［２．２．２］オクタ−３−イル）ベンゾフラン−２−カルボキサミド、その新規塩形態およびその使用方法 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010520213A Active JP5358573B2 (ja) | 2007-08-02 | 2008-08-01 | （２ｓ，３ｒ）−ｎ−（２−（（３−ピリジニル）メチル）−１−アザビシクロ［２．２．２］オクタ−３−イル）ベンゾフラン−２−カルボキサミド、その新規塩形態およびその使用方法 |
| JP2013148087A Active JP5852611B2 (ja) | 2007-08-02 | 2013-07-17 | （２ｓ，３ｒ）−ｎ−（２−（（３−ピリジニル）メチル）−１−アザビシクロ［２．２．２］オクタ−３−イル）ベンゾフラン−２−カルボキサミド、その新規塩形態およびその使用方法 |
| JP2013148091A Active JP6106549B2 (ja) | 2007-08-02 | 2013-07-17 | （２ｓ，３ｒ）−ｎ−（２−（（３−ピリジニル）メチル）−１−アザビシクロ［２．２．２］オクタ−３−イル）ベンゾフラン−２−カルボキサミド、その新規塩形態およびその使用方法 |
Country Status (35)
| Country | Link |
|---|---|
| US (6) | US20110124678A1 (OSRAM) |
| EP (6) | EP2465501B1 (OSRAM) |
| JP (4) | JP2010535252A (OSRAM) |
| KR (2) | KR20100051684A (OSRAM) |
| CN (4) | CN101868237A (OSRAM) |
| AR (1) | AR067775A1 (OSRAM) |
| AU (3) | AU2008283813A1 (OSRAM) |
| BR (2) | BRPI0814889A2 (OSRAM) |
| CA (2) | CA2694510A1 (OSRAM) |
| CL (3) | CL2008002271A1 (OSRAM) |
| CO (2) | CO6260080A2 (OSRAM) |
| CY (1) | CY1113561T1 (OSRAM) |
| DK (2) | DK2182949T3 (OSRAM) |
| EC (2) | ECSP10010008A (OSRAM) |
| ES (3) | ES2606752T3 (OSRAM) |
| HR (1) | HRP20130286T1 (OSRAM) |
| HU (1) | HUE030387T2 (OSRAM) |
| IL (1) | IL218976A0 (OSRAM) |
| ME (1) | ME01508B (OSRAM) |
| MX (3) | MX2010001293A (OSRAM) |
| MY (1) | MY148002A (OSRAM) |
| NO (2) | NO20100077L (OSRAM) |
| NZ (2) | NZ582828A (OSRAM) |
| PE (3) | PE20121820A1 (OSRAM) |
| PH (2) | PH12012501513A1 (OSRAM) |
| PL (1) | PL2182949T3 (OSRAM) |
| PT (1) | PT2182949E (OSRAM) |
| RS (1) | RS52743B (OSRAM) |
| RU (2) | RU2012140148A (OSRAM) |
| SA (2) | SA08290475B1 (OSRAM) |
| SI (1) | SI2182949T1 (OSRAM) |
| TW (3) | TW201402116A (OSRAM) |
| UY (1) | UY31265A (OSRAM) |
| WO (2) | WO2009018505A1 (OSRAM) |
| ZA (1) | ZA201000719B (OSRAM) |
Families Citing this family (38)
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| SA08290475B1 (ar) * | 2007-08-02 | 2013-06-22 | Targacept Inc | (2s، 3r)-n-(2-((3-بيردينيل)ميثيل)-1-آزا بيسيكلو[2، 2، 2]أوكت-3-يل)بنزو فيوران-2-كربوكساميد، وصور أملاحه الجديدة وطرق استخدامه |
| US20110098312A1 (en) * | 2008-05-12 | 2011-04-28 | Targacept ,Inc | Methods for preventing the development of retinopathy by the oral administration of nnr ligands |
| TW201031664A (en) | 2009-01-26 | 2010-09-01 | Targacept Inc | Preparation and therapeutic applications of (2S,3R)-N-2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)-3,5-difluorobenzamide |
| JO3250B1 (ar) | 2009-09-22 | 2018-09-16 | Novartis Ag | إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 |
| CN103221411B (zh) | 2010-05-17 | 2016-05-11 | 富瑞姆制药公司 | (R)-7-氯-N-(奎宁环-3-基)苯并[b]噻吩-2-甲酰胺盐酸盐单水合物的晶型 |
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| CN106074548A (zh) | 2010-09-23 | 2016-11-09 | 艾伯维巴哈马有限公司 | 氮杂金刚烷衍生物的一水合物 |
| JP2014502996A (ja) * | 2011-01-18 | 2014-02-06 | ターガセプト，インコーポレイテッド | 統合失調症における認知障害の治療 |
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| PL2685979T3 (pl) | 2011-03-18 | 2017-02-28 | Alkermes Pharma Ireland Limited | Kompozycje farmaceutyczne do wstrzykiwania zawierające środek nierozpuszczalny w wodzie, środek przeciwpsychotyczny, laurynian sorbitanu i polisorbat 20 |
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| EP2727604A4 (en) | 2011-06-30 | 2015-03-18 | Toray Industries | ANTIPRURIGINOUS AGENT |
| TW201311698A (zh) * | 2011-08-22 | 2013-03-16 | Targacept Inc | 作為神經元菸鹼乙醯膽鹼受體配位體之１，４－二氮雜雙環［３．２．２］壬烷 |
| CA3083244C (en) | 2011-10-20 | 2023-01-03 | Novartis Ag | Biomarkers predictive of responsiveness to alpha 7 nicotinic acetylcholine receptor activator treatment |
| US9993556B2 (en) * | 2012-03-19 | 2018-06-12 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising fatty glycerol esters |
| AU2013235519C1 (en) | 2012-03-19 | 2018-04-26 | Alkermes Pharma Ireland Limited | Pharmaaceutical compositions comprising fatty acid esters |
| CA2867137C (en) | 2012-03-19 | 2020-12-08 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol |
| AU2013259871A1 (en) | 2012-05-08 | 2014-11-20 | Forum Pharmaceuticals Inc. | Methods of maintaining, treating or improving cognitive function |
| NZ730571A (en) | 2012-09-19 | 2018-12-21 | Alkermes Pharma Ireland Ltd | Pharmaceutical compositions having improved storage stability |
| JP6114951B2 (ja) | 2012-12-11 | 2017-04-19 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体アクチベーターによる処置に対する応答性を予測するバイオマーカー |
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| ES2883232T3 (es) | 2013-01-15 | 2021-12-07 | Novartis Ag | Uso de agonistas del receptor nicotínico de acetilcolina alfa 7 |
| WO2014111837A1 (en) | 2013-01-15 | 2014-07-24 | Novartis Ag | Use of alpha 7 nicotinic acetylcholine receptor agonists |
| WO2014111751A1 (en) | 2013-01-15 | 2014-07-24 | Novartis Ag | Use of alpha 7 nicotinic receptor agonists for the treatment of narcolepsy |
| WO2014153424A1 (en) * | 2013-03-19 | 2014-09-25 | La Jolla Institute For Allergy And Immunology | Reducing diabetes in patients receiving hmg-coa reductase inhibitors (statins) |
| BR112016021535A8 (pt) | 2014-03-20 | 2021-07-20 | Alkermes Pharma Ireland Ltd | kit compreendendo formulações de aripiprazol tendo velocidades de injeção aumentadas útil para o tratamento de uma desordem do sistema nervoso central e uso |
| WO2015154064A2 (en) | 2014-04-04 | 2015-10-08 | Del Mar Pharmaceuticals | Use of dianhydrogalactitol and analogs or derivatives thereof to treat non-small-cell carcinoma of the lung and ovarian cancer |
| CN104288771B (zh) * | 2014-09-30 | 2017-03-15 | 郑州大学第五附属医院 | α7nAChR激动剂的新用途 |
| US10857140B2 (en) | 2015-05-06 | 2020-12-08 | The Regents Of The University Of California | K-Ras modulators |
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| RU2675111C2 (ru) * | 2017-03-31 | 2018-12-17 | Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт фундаментальной и клинической иммунологии" | Способ стимуляции нейрогенеза в гиппокампе |
| EP3612526A2 (en) | 2017-04-20 | 2020-02-26 | The Regents of the University of California | K-ras modulators |
| AU2019230014B2 (en) | 2018-03-05 | 2024-11-28 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
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