JP2007504174A5 - - Google Patents

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Publication number
JP2007504174A5
JP2007504174A5 JP2006525016A JP2006525016A JP2007504174A5 JP 2007504174 A5 JP2007504174 A5 JP 2007504174A5 JP 2006525016 A JP2006525016 A JP 2006525016A JP 2006525016 A JP2006525016 A JP 2006525016A JP 2007504174 A5 JP2007504174 A5 JP 2007504174A5
Authority
JP
Japan
Prior art keywords
disorders
epilepsy
pharmaceutical composition
pain
depression
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006525016A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007504174A (ja
Filing date
Publication date
Priority claimed from US10/655,393 external-priority patent/US7186726B2/en
Application filed filed Critical
Publication of JP2007504174A publication Critical patent/JP2007504174A/ja
Publication of JP2007504174A5 publication Critical patent/JP2007504174A5/ja
Pending legal-status Critical Current

Links

JP2006525016A 2003-09-03 2004-09-03 カルシウムチャネル遮断薬として使用されるピペラジン置換化合物 Pending JP2007504174A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/655,393 US7186726B2 (en) 1998-06-30 2003-09-03 Preferentially substituted calcium channel blockers
PCT/CA2004/001629 WO2005021523A1 (en) 2003-09-03 2004-09-03 Piperazine substituted compounds used as calcium channel blockers

Publications (2)

Publication Number Publication Date
JP2007504174A JP2007504174A (ja) 2007-03-01
JP2007504174A5 true JP2007504174A5 (OSRAM) 2007-10-18

Family

ID=34273458

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006525016A Pending JP2007504174A (ja) 2003-09-03 2004-09-03 カルシウムチャネル遮断薬として使用されるピペラジン置換化合物

Country Status (12)

Country Link
US (2) US7186726B2 (OSRAM)
EP (1) EP1670775A4 (OSRAM)
JP (1) JP2007504174A (OSRAM)
CN (1) CN1871225A (OSRAM)
AU (1) AU2004268711A1 (OSRAM)
BR (1) BRPI0414094A (OSRAM)
CA (1) CA2537487A1 (OSRAM)
IL (1) IL174025A0 (OSRAM)
MX (1) MXPA06002467A (OSRAM)
NZ (1) NZ546254A (OSRAM)
WO (1) WO2005021523A1 (OSRAM)
ZA (1) ZA200602684B (OSRAM)

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US7511077B2 (en) * 2005-02-09 2009-03-31 Neuromed Pharmaceuticals Ltd. Diamine calcium channel blockers
JP2008534630A (ja) * 2005-04-08 2008-08-28 ニューロメッド ファーマシューティカルズ リミテッド 疼痛の軽減のためのｎ型カルシウムチャネルブロッカーを含む組み合わせ治療の方法
US7705002B2 (en) 2005-05-19 2010-04-27 Vertex Pharmaceuticals Incorporated Biaryls useful as modulators of ion channels
JP5388574B2 (ja) 2005-05-31 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド イオンチャネルのモジュレーターとして有用なヘテロ環式類
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WO2008031227A1 (en) * 2006-09-14 2008-03-20 Neuromed Pharmaceuticals Ltd. Diaryl piperidine compounds as calcium channel blockers
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TWI404716B (zh) * 2006-10-17 2013-08-11 Kudos Pharm Ltd 酞嗪酮（ｐｈｔｈａｌａｚｉｎｏｎｅ）衍生物
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EP2149560B1 (en) 2007-05-22 2015-05-13 Astellas Pharma Inc. 1-substituted tetrahydroisoquinoline compound
KR101598231B1 (ko) * 2007-10-17 2016-02-26 쿠도스 파마슈티칼스 리미티드 4-[3-(4-시클로프로판카르보닐-피페라진-1-카르보닐)-4-플루오로-벤질]-2ｈ-프탈라진-1-온
WO2009132454A1 (en) * 2008-04-28 2009-11-05 Neuromed Pharmaceuticals Ltd. Di-t-butylphenyl piperazines as calcium channel blockers
US20090270338A1 (en) * 2008-04-28 2009-10-29 Galemmo Jr Robert Diaryl-cyclylalkyl derivatives as calcium channel blockers
CA2737400C (en) * 2008-10-07 2016-11-22 Astrazeneca Uk Limited Pharmaceutical formulation 514
PT3002008T (pt) 2010-03-11 2018-12-24 Univ New York Compostos de amido como moduladores roryt e suas utilizações
US8591944B2 (en) 2011-03-08 2013-11-26 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
US8409560B2 (en) 2011-03-08 2013-04-02 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
EP2753327A4 (en) * 2011-09-09 2015-04-08 Univ New York AMIDOVER BINDINGS AS RORYT MODULATORS AND ITS USE
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