JP2010535233A5 - - Google Patents

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Publication number
JP2010535233A5
JP2010535233A5 JP2010520122A JP2010520122A JP2010535233A5 JP 2010535233 A5 JP2010535233 A5 JP 2010535233A5 JP 2010520122 A JP2010520122 A JP 2010520122A JP 2010520122 A JP2010520122 A JP 2010520122A JP 2010535233 A5 JP2010535233 A5 JP 2010535233A5
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JP
Japan
Prior art keywords
protein kinase
kinase inhibitor
combination
alkyl
mek
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
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JP2010520122A
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English (en)
Japanese (ja)
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JP2010535233A (ja
JP5479337B2 (ja
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Publication date
Priority claimed from US11/830,733 external-priority patent/US8101799B2/en
Priority claimed from US12/016,897 external-priority patent/US7820664B2/en
Application filed filed Critical
Priority claimed from PCT/US2008/071397 external-priority patent/WO2009018238A1/en
Publication of JP2010535233A publication Critical patent/JP2010535233A/ja
Publication of JP2010535233A5 publication Critical patent/JP2010535233A5/ja
Application granted granted Critical
Publication of JP5479337B2 publication Critical patent/JP5479337B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2010520122A 2007-07-30 2008-07-28 Ｍｅｋ阻害剤およびｒａｆキナーゼ阻害剤の組み合わせ、ならびにその使用 Expired - Fee Related JP5479337B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US11/830,733 US8101799B2 (en) 2005-07-21 2007-07-30 Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK
US11/830,733 2007-07-30
US12/016,897 2008-01-18
US12/016,897 US7820664B2 (en) 2007-01-19 2008-01-18 Inhibitors of MEK
PCT/US2008/071397 WO2009018238A1 (en) 2007-07-30 2008-07-28 Combinations of mek inhibitors and raf kinase inhibitors and uses thereof

Publications (3)

Publication Number Publication Date
JP2010535233A JP2010535233A (ja) 2010-11-18
JP2010535233A5 true JP2010535233A5 (enExample) 2011-09-22
JP5479337B2 JP5479337B2 (ja) 2014-04-23

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010520122A Expired - Fee Related JP5479337B2 (ja) 2007-07-30 2008-07-28 Ｍｅｋ阻害剤およびｒａｆキナーゼ阻害剤の組み合わせ、ならびにその使用

Country Status (6)

Country Link
US (1) US8648116B2 (enExample)
EP (1) EP2175885B1 (enExample)
JP (1) JP5479337B2 (enExample)
CA (3) CA2694646C (enExample)
UA (1) UA99731C2 (enExample)
WO (1) WO2009018238A1 (enExample)

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