JP2010519243A5 - - Google Patents

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JP2010519243A5
JP2010519243A5 JP2009550278A JP2009550278A JP2010519243A5 JP 2010519243 A5 JP2010519243 A5 JP 2010519243A5 JP 2009550278 A JP2009550278 A JP 2009550278A JP 2009550278 A JP2009550278 A JP 2009550278A JP 2010519243 A5 JP2010519243 A5 JP 2010519243A5
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Japan
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compound
mixture
hydroxy
pharmaceutically acceptable
salt
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JP2009550278A
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JP5243455B2 (ja
JP2010519243A (ja
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Priority claimed from PCT/EP2008/051971 external-priority patent/WO2008101914A2/en
Publication of JP2010519243A publication Critical patent/JP2010519243A/ja
Publication of JP2010519243A5 publication Critical patent/JP2010519243A5/ja
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Publication of JP5243455B2 publication Critical patent/JP5243455B2/ja
Expired - Fee Related legal-status Critical Current
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JP2009550278A 2007-02-23 2008-02-19 新規化合物 Expired - Fee Related JP5243455B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07102956 2007-02-23
EP07102956.5 2007-02-23
PCT/EP2008/051971 WO2008101914A2 (en) 2007-02-23 2008-02-19 N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase

Publications (3)

Publication Number Publication Date
JP2010519243A JP2010519243A (ja) 2010-06-03
JP2010519243A5 true JP2010519243A5 (OSRAM) 2011-03-10
JP5243455B2 JP5243455B2 (ja) 2013-07-24

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JP2009550278A Expired - Fee Related JP5243455B2 (ja) 2007-02-23 2008-02-19 新規化合物

Country Status (13)

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US (3) US8383820B2 (OSRAM)
EP (1) EP2150526B1 (OSRAM)
JP (1) JP5243455B2 (OSRAM)
KR (1) KR101487813B1 (OSRAM)
CN (1) CN101679217A (OSRAM)
AU (1) AU2008219326B2 (OSRAM)
BR (1) BRPI0806847A2 (OSRAM)
CA (1) CA2675669C (OSRAM)
EA (1) EA016951B1 (OSRAM)
IL (1) IL199853A (OSRAM)
MX (1) MX2009008228A (OSRAM)
WO (1) WO2008101914A2 (OSRAM)
ZA (1) ZA200904916B (OSRAM)

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US8053447B2 (en) 2006-04-07 2011-11-08 High Point Pharmaceuticals, Llc 11β-hydroxysteroid dehydrogenase type 1 active compounds
CA2655282A1 (en) * 2006-06-16 2007-12-21 High Point Pharmaceuticals, Llc Pharmaceutical use of substituted piperidine carboxamides
CA2657078A1 (en) * 2006-07-13 2008-01-17 High Point Pharmaceuticals, Llc 11beta-hydroxysteroid dehydrogenase type 1 active compounds
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EP2125704A1 (en) * 2007-02-23 2009-12-02 High Point Pharmaceuticals, LLC N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
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JP5764133B2 (ja) * 2010-09-03 2015-08-12 大日本住友製薬株式会社 環状アミド誘導体
KR101332805B1 (ko) 2011-03-31 2013-11-27 한국화학연구원 아다만틸기를 갖는 설파마이드 유도체 및 이의 약제학적으로 허용 가능한 염
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
CN104529858A (zh) * 2015-01-13 2015-04-22 佛山市赛维斯医药科技有限公司 含卤代金刚烷和酰胺类衍生物、其制备方法和用途
CN104529856A (zh) * 2015-01-13 2015-04-22 佛山市赛维斯医药科技有限公司 一种硝基金刚烷酰胺衍生物、其制备方法和用途
CN104974084A (zh) * 2015-07-19 2015-10-14 佛山市赛维斯医药科技有限公司 一类胺基二吡啶叔醇结构的11β-HSD1抑制剂及其用途
CN104974080A (zh) * 2015-07-19 2015-10-14 佛山市赛维斯医药科技有限公司 二吡啶叔醇结构的11β-HSD1抑制剂、制备方法及其用途
CN110291383B (zh) * 2017-02-23 2021-12-28 株式会社Ihi Oh自由基检测探测器、oh自由基测定装置以及oh自由基测定方法

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JP2010519242A (ja) 2007-02-23 2010-06-03 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー 新規化合物
JP2010519239A (ja) 2007-02-23 2010-06-03 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー １１−ベータ−ヒドロキシステロイドデヒドロゲナーゼの阻害因子としてのｎ−アドマンチルベンザミド
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JP2010522766A (ja) 2007-03-28 2010-07-08 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー １１ベータ−ｈｓｄ１活性化合物
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EP2362730A4 (en) 2008-11-21 2012-08-29 High Point Pharmaceuticals Llc Adamantyl BENZAMIDE CONNECTIONS

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