JP2010516702A - 置換１，３−ジオキサンのプロドラッグおよびそれらの使用 - Google Patents

置換１，３−ジオキサンのプロドラッグおよびそれらの使用 Download PDF

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JP2010516702A
JP2010516702A JP2009546563A JP2009546563A JP2010516702A JP 2010516702 A JP2010516702 A JP 2010516702A JP 2009546563 A JP2009546563 A JP 2009546563A JP 2009546563 A JP2009546563 A JP 2009546563A JP 2010516702 A JP2010516702 A JP 2010516702A
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ppar
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JP2010516702A5 (enExample
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ペテリス アルバーツ，
アレクサンドラ サンタナ ソレンセン，
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Danstar Ferment AG
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Evolva AG
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Priority claimed from PCT/IB2007/002542 external-priority patent/WO2007138485A2/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
    • C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A61K31/36—Compounds containing methylenedioxyphenyl groups, e.g. sesamin
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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JP2009546563A 2007-01-18 2008-01-18 置換１，３−ジオキサンのプロドラッグおよびそれらの使用 Withdrawn JP2010516702A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
PCT/IB2007/002542 WO2007138485A2 (en) 2006-01-18 2007-01-18 Ppar modulators
US98980607P 2007-11-21 2007-11-21
US98980807P 2007-11-21 2007-11-21
US98980507P 2007-11-21 2007-11-21
PCT/US2008/051525 WO2008089464A1 (en) 2007-01-18 2008-01-18 Prodrugs of substituted 1,3-dioxanes and their uses

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