JP2010507602A5 - - Google Patents

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Publication number
JP2010507602A5
JP2010507602A5 JP2009533691A JP2009533691A JP2010507602A5 JP 2010507602 A5 JP2010507602 A5 JP 2010507602A5 JP 2009533691 A JP2009533691 A JP 2009533691A JP 2009533691 A JP2009533691 A JP 2009533691A JP 2010507602 A5 JP2010507602 A5 JP 2010507602A5
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JP
Japan
Prior art keywords
formula
alkylamino
alkoxy
alkyl
hydroxycarbonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009533691A
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English (en)
Japanese (ja)
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JP5247712B2 (ja
JP2010507602A (ja
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Publication date
Priority claimed from DE102006050516A external-priority patent/DE102006050516A1/de
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Publication of JP2010507602A publication Critical patent/JP2010507602A/ja
Publication of JP2010507602A5 publication Critical patent/JP2010507602A5/ja
Application granted granted Critical
Publication of JP5247712B2 publication Critical patent/JP5247712B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009533691A 2006-10-26 2007-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類 Active JP5247712B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102006050516A DE102006050516A1 (de) 2006-10-26 2006-10-26 Substituierte Dihydropyrazolone und ihre Verwendung
DE102006050516.6 2006-10-26
PCT/EP2007/008877 WO2008067871A1 (de) 2006-10-26 2007-10-12 Substituierte dihydropyrazolone zur behandlung kardiovaskulärer und hämatologischer erkrankungen

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010229627A Division JP5300813B2 (ja) 2006-10-26 2010-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類

Publications (3)

Publication Number Publication Date
JP2010507602A JP2010507602A (ja) 2010-03-11
JP2010507602A5 true JP2010507602A5 (enExample) 2010-11-25
JP5247712B2 JP5247712B2 (ja) 2013-07-24

Family

ID=38734870

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009533691A Active JP5247712B2 (ja) 2006-10-26 2007-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類
JP2010229627A Active JP5300813B2 (ja) 2006-10-26 2010-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010229627A Active JP5300813B2 (ja) 2006-10-26 2010-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類

Country Status (40)

Country Link
US (5) US8389520B2 (enExample)
EP (3) EP2084151B1 (enExample)
JP (2) JP5247712B2 (enExample)
KR (1) KR101455879B1 (enExample)
CN (2) CN101631785B (enExample)
AR (1) AR063392A1 (enExample)
AU (1) AU2007328052B2 (enExample)
BR (1) BRPI0717367B8 (enExample)
CA (1) CA2667382C (enExample)
CO (1) CO6170359A2 (enExample)
CR (2) CR10750A (enExample)
CU (2) CU23743B7 (enExample)
CY (1) CY1114272T1 (enExample)
DE (1) DE102006050516A1 (enExample)
DK (2) DK2084151T3 (enExample)
ES (3) ES2421454T3 (enExample)
GT (1) GT200900095A (enExample)
HN (1) HN2009000784A (enExample)
HR (2) HRP20130779T1 (enExample)
IL (2) IL198289A (enExample)
MA (1) MA30914B1 (enExample)
MX (1) MX2009004324A (enExample)
MY (1) MY169564A (enExample)
NO (1) NO343308B1 (enExample)
NZ (2) NZ576458A (enExample)
PE (3) PE20080895A1 (enExample)
PH (1) PH12013500578B1 (enExample)
PL (2) PL2084151T3 (enExample)
PT (2) PT2546253E (enExample)
RS (1) RS52924B (enExample)
RU (2) RU2469031C2 (enExample)
SG (1) SG176421A1 (enExample)
SI (1) SI2084151T1 (enExample)
SV (1) SV2009003236A (enExample)
TN (1) TN2009000132A1 (enExample)
TW (3) TWI437991B (enExample)
UA (1) UA98125C2 (enExample)
UY (1) UY30663A1 (enExample)
WO (1) WO2008067871A1 (enExample)
ZA (1) ZA200902705B (enExample)

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AU2009334570B2 (en) 2008-12-29 2016-06-09 Sanofi Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof
IT1393337B1 (it) 2009-03-06 2012-04-20 Italiana Sint Spa Sintesi di (4as, 7as)-ottaidro-1h-pirrolo[3,4-b]piridina
DE102010044131A1 (de) 2010-11-18 2012-05-24 Bayer Schering Pharma Aktiengesellschaft Substituiertes Natrium-1H-pyrazol-5-olat
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RS56255B1 (sr) * 2012-05-08 2017-11-30 Bayern Pharma Ag Postupak proizvodnje jedinjenja triazola
WO2013181136A1 (en) 2012-05-29 2013-12-05 Momentive Performance Materials Gmbh Preparation of isocyanato silanes
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SI3057580T1 (sl) 2013-10-17 2021-07-30 Bayer Pharma Aktiengesellschaft Farmacevtske dozirne oblike, ki vsebujejo natrijev 1-(6-(morfolin-4-il)pirimidin-4-il)-4-(1H-1,2,3-triazol-1-il)-1H- pirazol-5-olat
WO2016034108A1 (zh) 2014-09-02 2016-03-10 广东东阳光药业有限公司 喹啉酮类化合物及其应用
CN107778262A (zh) * 2016-08-24 2018-03-09 尹玉新 1,5‑双取代四氮唑类化合物及其制备方法和应用
CN109694380B (zh) * 2017-10-23 2022-09-27 中国医药研究开发中心有限公司 二氢吡唑啉酮类化合物及其制备方法和医药用途
CN111825690B (zh) * 2019-04-17 2022-09-27 中国医药研究开发中心有限公司 一种phd抑制剂的新晶型及其制备方法
US11579118B2 (en) 2019-06-03 2023-02-14 Tdw Delaware, Inc. Single point contact triaxial sensor head for an inline inspection tool
US10702525B1 (en) 2019-09-04 2020-07-07 United Arab Emirates University Pyrimidine derivatives as anti-diabetic agents
EP4103281A1 (en) * 2020-02-11 2022-12-21 Acurastem Inc. Pikfyve kinase inhibitors
US20230148601A1 (en) 2020-02-18 2023-05-18 Bayer Aktiengesellschaft Novel heteroaryl-triazole compounds as pesticides
EP4121424A1 (en) * 2020-03-20 2023-01-25 Akebia Therapeutics Inc. Phd inhibitor compounds, compositions, and their use
EP3888684A1 (en) 2020-03-31 2021-10-06 Bayer Animal Health GmbH Composition having improved voluntary acceptance
EP4138825A1 (en) 2020-04-20 2023-03-01 Akebia Therapeutics Inc. Treatment of viral infections, of organ injury, and of related conditions using a hif prolyl hydroxylase inhibitor or a hif-alpha stabilizer
WO2022150623A1 (en) 2021-01-08 2022-07-14 Akebia Therapeutics, Inc. Compounds and composition for the treatment of anemia
TW202313072A (zh) 2021-05-27 2023-04-01 美商凱立克斯生物製藥股份有限公司 檸檬酸鐵之兒科調配物
DE102021206771A1 (de) 2021-06-29 2022-12-29 Volkswagen Aktiengesellschaft Verfahren zum Ausgeben eines Startbereichs für einen Parkvorgang eines Kraftfahrzeugs, elektronische Recheneinrichtung sowie Kraftfahrzeug
CN116120340B (zh) * 2021-11-15 2023-10-31 艾立康药业股份有限公司 一种吡啶并噁嗪类化合物及其制备方法、组合物和用途
CN116063233B (zh) * 2022-10-31 2025-08-15 广州市联瑞制药有限公司 一种1h-咪唑-1-乙酸烃酯的制备方法
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