JP2010507602A5 - - Google Patents

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Publication number
JP2010507602A5
JP2010507602A5 JP2009533691A JP2009533691A JP2010507602A5 JP 2010507602 A5 JP2010507602 A5 JP 2010507602A5 JP 2009533691 A JP2009533691 A JP 2009533691A JP 2009533691 A JP2009533691 A JP 2009533691A JP 2010507602 A5 JP2010507602 A5 JP 2010507602A5
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JP
Japan
Prior art keywords
formula
alkylamino
alkoxy
alkyl
hydroxycarbonyl
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JP2009533691A
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English (en)
Japanese (ja)
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JP5247712B2 (ja
JP2010507602A (ja
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Priority claimed from DE102006050516A external-priority patent/DE102006050516A1/de
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Publication of JP2010507602A publication Critical patent/JP2010507602A/ja
Publication of JP2010507602A5 publication Critical patent/JP2010507602A5/ja
Application granted granted Critical
Publication of JP5247712B2 publication Critical patent/JP5247712B2/ja
Active legal-status Critical Current
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JP2009533691A 2006-10-26 2007-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類 Active JP5247712B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102006050516.6 2006-10-26
DE102006050516A DE102006050516A1 (de) 2006-10-26 2006-10-26 Substituierte Dihydropyrazolone und ihre Verwendung
PCT/EP2007/008877 WO2008067871A1 (de) 2006-10-26 2007-10-12 Substituierte dihydropyrazolone zur behandlung kardiovaskulärer und hämatologischer erkrankungen

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010229627A Division JP5300813B2 (ja) 2006-10-26 2010-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類

Publications (3)

Publication Number Publication Date
JP2010507602A JP2010507602A (ja) 2010-03-11
JP2010507602A5 true JP2010507602A5 (enExample) 2010-11-25
JP5247712B2 JP5247712B2 (ja) 2013-07-24

Family

ID=38734870

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009533691A Active JP5247712B2 (ja) 2006-10-26 2007-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類
JP2010229627A Active JP5300813B2 (ja) 2006-10-26 2010-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010229627A Active JP5300813B2 (ja) 2006-10-26 2010-10-12 心血管および血液の疾患の処置用の置換ジヒドロピラゾロン類

Country Status (40)

Country Link
US (5) US8389520B2 (enExample)
EP (3) EP2546253B1 (enExample)
JP (2) JP5247712B2 (enExample)
KR (1) KR101455879B1 (enExample)
CN (2) CN103342696B (enExample)
AR (1) AR063392A1 (enExample)
AU (1) AU2007328052B2 (enExample)
BR (1) BRPI0717367B8 (enExample)
CA (1) CA2667382C (enExample)
CO (1) CO6170359A2 (enExample)
CR (2) CR10750A (enExample)
CU (2) CU23743B7 (enExample)
CY (1) CY1114272T1 (enExample)
DE (1) DE102006050516A1 (enExample)
DK (2) DK2546253T3 (enExample)
ES (3) ES2421454T3 (enExample)
GT (1) GT200900095A (enExample)
HN (1) HN2009000784A (enExample)
HR (2) HRP20130779T1 (enExample)
IL (2) IL198289A (enExample)
MA (1) MA30914B1 (enExample)
MX (1) MX2009004324A (enExample)
MY (1) MY169564A (enExample)
NO (1) NO343308B1 (enExample)
NZ (2) NZ576458A (enExample)
PE (3) PE20080895A1 (enExample)
PH (1) PH12013500578B1 (enExample)
PL (2) PL2546253T3 (enExample)
PT (2) PT2084151E (enExample)
RS (1) RS52924B (enExample)
RU (2) RU2469031C2 (enExample)
SG (1) SG176421A1 (enExample)
SI (1) SI2084151T1 (enExample)
SV (1) SV2009003236A (enExample)
TN (1) TN2009000132A1 (enExample)
TW (3) TWI437991B (enExample)
UA (1) UA98125C2 (enExample)
UY (1) UY30663A1 (enExample)
WO (1) WO2008067871A1 (enExample)
ZA (1) ZA200902705B (enExample)

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CA2927437C (en) * 2013-10-17 2022-06-28 Bayer Pharma Aktiengesellschaft Pharmaceutical dosage forms containing sodium-1-[6-(morpholin-4-yl)pyrimidin-4-yl]-4-(1h-1,2,3-triazol-1-yl)-1h-pyrazol-5-olate
US10065928B2 (en) 2014-09-02 2018-09-04 Sunshine Lake Pharma Co., Ltd. Quinolinone compound and use thereof
CN107778262A (zh) * 2016-08-24 2018-03-09 尹玉新 1,5‑双取代四氮唑类化合物及其制备方法和应用
CN109694380B (zh) * 2017-10-23 2022-09-27 中国医药研究开发中心有限公司 二氢吡唑啉酮类化合物及其制备方法和医药用途
CN111825690B (zh) * 2019-04-17 2022-09-27 中国医药研究开发中心有限公司 一种phd抑制剂的新晶型及其制备方法
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US10702525B1 (en) 2019-09-04 2020-07-07 United Arab Emirates University Pyrimidine derivatives as anti-diabetic agents
US20230135152A1 (en) * 2020-02-11 2023-05-04 AcuraStem Incorporated Pikfyve kinase inhibitors
JP2023513624A (ja) 2020-02-18 2023-03-31 バイエル・アクチエンゲゼルシヤフト 殺有害生物剤としてのヘテロアリール－トリアゾール化合物
CN115605467B (zh) * 2020-03-20 2025-06-13 阿克比治疗有限公司 Phd抑制剂化合物、组合物和其用途
EP3888684A1 (en) 2020-03-31 2021-10-06 Bayer Animal Health GmbH Composition having improved voluntary acceptance
EP4138825A1 (en) 2020-04-20 2023-03-01 Akebia Therapeutics Inc. Treatment of viral infections, of organ injury, and of related conditions using a hif prolyl hydroxylase inhibitor or a hif-alpha stabilizer
WO2022150623A1 (en) 2021-01-08 2022-07-14 Akebia Therapeutics, Inc. Compounds and composition for the treatment of anemia
WO2022251563A1 (en) 2021-05-27 2022-12-01 Keryx Biopharmaceuticals, Inc. Pediatric formulations of ferric citrate
DE102021206771B4 (de) 2021-06-29 2025-12-24 Volkswagen Aktiengesellschaft Verfahren zum Ausgeben eines Startbereichs für einen Parkvorgang eines Kraftfahrzeugs, elektronische Recheneinrichtung sowie Kraftfahrzeug
CN116120340B (zh) * 2021-11-15 2023-10-31 艾立康药业股份有限公司 一种吡啶并噁嗪类化合物及其制备方法、组合物和用途
CN116063233B (zh) * 2022-10-31 2025-08-15 广州市联瑞制药有限公司 一种1h-咪唑-1-乙酸烃酯的制备方法
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