JP2009537469A5 - - Google Patents
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- Publication number
- JP2009537469A5 JP2009537469A5 JP2009510362A JP2009510362A JP2009537469A5 JP 2009537469 A5 JP2009537469 A5 JP 2009537469A5 JP 2009510362 A JP2009510362 A JP 2009510362A JP 2009510362 A JP2009510362 A JP 2009510362A JP 2009537469 A5 JP2009537469 A5 JP 2009537469A5
- Authority
- JP
- Japan
- Prior art keywords
- halogen
- alkyl
- substituted
- hydrogen
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 229910052736 halogen Inorganic materials 0.000 claims 26
- 229910052739 hydrogen Inorganic materials 0.000 claims 24
- 239000001257 hydrogen Substances 0.000 claims 24
- 150000002367 halogens Chemical class 0.000 claims 20
- 125000001424 substituent group Chemical group 0.000 claims 17
- 150000002431 hydrogen Chemical class 0.000 claims 16
- 150000001875 compounds Chemical class 0.000 claims 15
- 125000004093 cyano group Chemical group *C#N 0.000 claims 14
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 9
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 9
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 7
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 5
- 125000000217 alkyl group Chemical group 0.000 claims 4
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 3
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 3
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 3
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 3
- 125000004438 haloalkoxy group Chemical group 0.000 claims 3
- 125000005843 halogen group Chemical group 0.000 claims 3
- 229910052760 oxygen Inorganic materials 0.000 claims 3
- 239000001301 oxygen Substances 0.000 claims 3
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 2
- -1 C 1 -C 6 alkyl Chemical group 0.000 claims 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 2
- 230000002401 inhibitory effect Effects 0.000 claims 2
- 244000005700 microbiome Species 0.000 claims 2
- 125000001624 naphthyl group Chemical group 0.000 claims 2
- 230000003032 phytopathogenic effect Effects 0.000 claims 2
- 125000002943 quinolinyl group Chemical group N1=C(C=CC2=CC=CC=C12)* 0.000 claims 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims 2
- 229910052717 sulfur Chemical group 0.000 claims 2
- 239000011593 sulfur Chemical group 0.000 claims 2
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 1
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims 1
- 206010061217 Infestation Diseases 0.000 claims 1
- 239000004480 active ingredient Substances 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 150000001602 bicycloalkyls Chemical group 0.000 claims 1
- 244000038559 crop plants Species 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 125000001188 haloalkyl group Chemical group 0.000 claims 1
- 125000001072 heteroaryl group Chemical group 0.000 claims 1
- 125000005842 heteroatom Chemical group 0.000 claims 1
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 1
- 229910052757 nitrogen Inorganic materials 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06010224 | 2006-05-18 | ||
| EP06010224.1 | 2006-05-18 | ||
| PCT/EP2007/004425 WO2007134799A1 (en) | 2006-05-18 | 2007-05-16 | Novel microbiocides |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009537469A JP2009537469A (ja) | 2009-10-29 |
| JP2009537469A5 true JP2009537469A5 (enExample) | 2010-05-27 |
| JP5155303B2 JP5155303B2 (ja) | 2013-03-06 |
Family
ID=38474462
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009510362A Expired - Fee Related JP5155303B2 (ja) | 2006-05-18 | 2007-05-16 | 新規な殺微生物剤 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US8618023B2 (enExample) |
| EP (1) | EP2018367B1 (enExample) |
| JP (1) | JP5155303B2 (enExample) |
| KR (1) | KR101380139B1 (enExample) |
| CN (1) | CN101466671B (enExample) |
| AR (1) | AR061021A1 (enExample) |
| AT (1) | ATE449068T1 (enExample) |
| BR (1) | BRPI0712027B1 (enExample) |
| CA (1) | CA2650795A1 (enExample) |
| DE (1) | DE602007003343D1 (enExample) |
| ES (1) | ES2335319T3 (enExample) |
| GT (1) | GT200700041A (enExample) |
| MX (1) | MX2008014534A (enExample) |
| TW (1) | TWI388547B (enExample) |
| WO (1) | WO2007134799A1 (enExample) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009043784A1 (en) * | 2007-10-04 | 2009-04-09 | F. Hoffmann-La Roche Ag | Cyclopropyl aryl amide derivatives and uses thereof |
| US8993808B2 (en) | 2009-01-21 | 2015-03-31 | Oryzon Genomics, S.A. | Phenylcyclopropylamine derivatives and their medical use |
| EP2398770B1 (en) * | 2009-02-17 | 2016-12-28 | Bayer Intellectual Property GmbH | Fungicidal n-(phenylcycloalkyl)carboxamide, n-(benzylcycloalkyl)carboxamide and thiocarboxamide derivatives |
| US8859555B2 (en) | 2009-09-25 | 2014-10-14 | Oryzon Genomics S.A. | Lysine Specific Demethylase-1 inhibitors and their use |
| EP2486002B1 (en) | 2009-10-09 | 2019-03-27 | Oryzon Genomics, S.A. | Substituted heteroaryl- and aryl- cyclopropylamine acetamides and their use |
| CN102574808A (zh) * | 2009-10-16 | 2012-07-11 | 先正达参股股份有限公司 | 新型杀微生物剂 |
| WO2011106573A2 (en) | 2010-02-24 | 2011-09-01 | Oryzon Genomics, S.A. | Lysine demethylase inhibitors for diseases and disorders associated with hepadnaviridae |
| US9616058B2 (en) | 2010-02-24 | 2017-04-11 | Oryzon Genomics, S.A. | Potent selective LSD1 inhibitors and dual LSD1/MAO-B inhibitors for antiviral use |
| RU2424660C1 (ru) * | 2010-03-25 | 2011-07-27 | Валерий Федорович Швец | Композиция для обработки растений и плодов и способы повышения урожая плодоовощной и растениеводческой продукции и увеличение срока его хранения |
| MX2012012111A (es) | 2010-04-19 | 2013-05-30 | Oryzon Genomics Sa | Inhibidores de demetilasa-1 especifica de lisina y su uso. |
| ES2533026T3 (es) | 2010-06-03 | 2015-04-07 | Bayer Intellectual Property Gmbh | N-[(het)arilalquil)]pirazol (tio)carboxamidas y sus análogos heterosustituidos |
| SI2598482T1 (sl) | 2010-07-29 | 2018-09-28 | Oryzon Genomics, S.A. | Inhibitorji demetilaze lsd1 na osnovi arilciklopropilamina in njihova medicinska uporaba |
| WO2012013727A1 (en) | 2010-07-29 | 2012-02-02 | Oryzon Genomics S.A. | Cyclopropylamine derivatives useful as lsd1 inhibitors |
| WO2012045883A1 (en) | 2010-10-08 | 2012-04-12 | Oryzon Genomics S.A. | Cyclopropylamine inhibitors of oxidases |
| WO2012072713A2 (en) | 2010-11-30 | 2012-06-07 | Oryzon Genomics, S.A. | Lysine demethylase inhibitors for diseases and disorders associated with flaviviridae |
| WO2012107498A1 (en) | 2011-02-08 | 2012-08-16 | Oryzon Genomics S.A. | Lysine demethylase inhibitors for myeloproliferative disorders |
| RS58475B1 (sr) | 2011-10-20 | 2019-04-30 | Oryzon Genomics Sa | Jedinjenja (hetero)aril ciklopropilamina kao lsd1 inhibitori |
| CN107266345B (zh) | 2011-10-20 | 2021-08-17 | 奥瑞泽恩基因组学股份有限公司 | 作为lsd1抑制剂的(杂)芳基环丙胺化合物 |
| WO2013120940A2 (en) | 2012-02-14 | 2013-08-22 | Syngenta Participations Ag | Novel compounds |
| EP2740474A1 (en) | 2012-12-05 | 2014-06-11 | Instituto Europeo di Oncologia S.r.l. | Cyclopropylamine derivatives useful as inhibitors of histone demethylases kdm1a |
| TW201507722A (zh) | 2013-04-30 | 2015-03-01 | Bayer Cropscience Ag | 做為殺線蟲劑及殺體內寄生蟲劑的ｎ－（２－鹵素－２－苯乙基）－羧醯胺類 |
| JP7421479B2 (ja) * | 2017-12-20 | 2024-01-24 | シンジェンタ パーティシペーションズ アーゲー | 植物病原性微生物による野菜、トマト及びジャガイモ植物の被害を防除又は防止する方法 |
| PY1999323A (es) * | 2018-11-28 | 2020-10-29 | Bayer Ag | (tio)amidas de piridazina como compuestos fungicidas |
| CN115915941B (zh) | 2020-05-06 | 2025-07-15 | 拜耳公司 | 作为杀真菌化合物的吡啶（硫代）酰胺 |
| BR112022023012A2 (pt) | 2020-05-12 | 2022-12-20 | Bayer Ag | (tio)amidas de triazina e pirimidina como compostos fungicidas |
| BR112022023550A2 (pt) * | 2020-05-19 | 2023-01-03 | Bayer Cropscience Ag | (tio)amidas azabicíclicas como compostos fungicidas |
| CN115697059A (zh) | 2020-05-27 | 2023-02-03 | 拜耳公司 | 活性化合物组合 |
| CN118541353A (zh) | 2021-11-03 | 2024-08-23 | 拜耳公司 | 作为杀真菌化合物的双(杂)芳基硫醚(硫代)酰胺 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5849769A (en) | 1994-08-24 | 1998-12-15 | Medivir Ab | N-arylalkyl-N-heteroarylurea and guandine compounds and methods of treating HIV infection |
| JP3844533B2 (ja) | 1995-12-15 | 2006-11-15 | 日本曹達株式会社 | ２，６−ジクロロイソニコチン酸フェネチルアミド誘導体及び植物病害防除剤 |
| FR2784375B1 (fr) | 1998-10-12 | 2000-11-24 | Adir | Nouveaux derives cycliques a chaine cycloalkylenique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| KR100676987B1 (ko) | 1998-11-04 | 2007-01-31 | 메이지 세이카 가부시키가이샤 | 피콜린산아미드 유도체, 그 것을 유효성분으로서 함유하는유해생물 방제제 |
| EP1388535A1 (en) * | 2002-08-07 | 2004-02-11 | Aventis Pharma Deutschland GmbH | Acylated arylcycloalkylamines and their use as pharmaceuticals |
| US7186735B2 (en) * | 2002-08-07 | 2007-03-06 | Sanofi-Aventis Deutschland Gmbh | Acylated arylcycloalkylamines and their use as pharmaceuticals |
| KR101276929B1 (ko) * | 2004-04-26 | 2013-06-19 | 바이엘 크롭사이언스 아게 | 살진균제로서 유용한 2-피리디닐시클로알킬카르복사미드유도체 |
| EP1591442A1 (en) * | 2004-04-26 | 2005-11-02 | Bayer CropScience S.A. | 2-Pyridinycycloalkylbenzamide derivatives and their use as fungicides |
| US7932396B2 (en) * | 2005-05-18 | 2011-04-26 | Bayer Cropscience Ag | 2-pyridinylcycloalkylbenzamide derivatives and their use as fungicides |
| EP1885712B1 (en) * | 2005-05-18 | 2011-02-23 | Bayer CropScience AG | New 2-pyridinylcycloalkylcarboxamide derivatives as fungicides. |
-
2007
- 2007-05-16 KR KR1020087030887A patent/KR101380139B1/ko not_active Expired - Fee Related
- 2007-05-16 DE DE602007003343T patent/DE602007003343D1/de active Active
- 2007-05-16 EP EP07764538A patent/EP2018367B1/en not_active Not-in-force
- 2007-05-16 BR BRPI0712027A patent/BRPI0712027B1/pt not_active IP Right Cessation
- 2007-05-16 ES ES07764538T patent/ES2335319T3/es active Active
- 2007-05-16 WO PCT/EP2007/004425 patent/WO2007134799A1/en not_active Ceased
- 2007-05-16 US US12/301,080 patent/US8618023B2/en not_active Expired - Fee Related
- 2007-05-16 CN CN2007800211443A patent/CN101466671B/zh not_active Expired - Fee Related
- 2007-05-16 CA CA002650795A patent/CA2650795A1/en not_active Abandoned
- 2007-05-16 MX MX2008014534A patent/MX2008014534A/es active IP Right Grant
- 2007-05-16 GT GT200700041A patent/GT200700041A/es unknown
- 2007-05-16 JP JP2009510362A patent/JP5155303B2/ja not_active Expired - Fee Related
- 2007-05-16 AT AT07764538T patent/ATE449068T1/de not_active IP Right Cessation
- 2007-05-16 TW TW096117375A patent/TWI388547B/zh not_active IP Right Cessation
- 2007-05-18 AR ARP070102155A patent/AR061021A1/es not_active Application Discontinuation
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