JP2009542815A5 - - Google Patents

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Publication number
JP2009542815A5
JP2009542815A5 JP2009519604A JP2009519604A JP2009542815A5 JP 2009542815 A5 JP2009542815 A5 JP 2009542815A5 JP 2009519604 A JP2009519604 A JP 2009519604A JP 2009519604 A JP2009519604 A JP 2009519604A JP 2009542815 A5 JP2009542815 A5 JP 2009542815A5
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JP
Japan
Prior art keywords
ylamino
methoxyquinolin
group
dichloropyridin
cyclopentyloxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009519604A
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English (en)
Japanese (ja)
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JP2009542815A (ja
JP5280357B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2007/072919 external-priority patent/WO2008006050A2/en
Publication of JP2009542815A publication Critical patent/JP2009542815A/ja
Publication of JP2009542815A5 publication Critical patent/JP2009542815A5/ja
Application granted granted Critical
Publication of JP5280357B2 publication Critical patent/JP5280357B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009519604A 2006-07-07 2007-07-06 Ｐｄｅ４の二環式ヘテロアリール阻害剤 Expired - Fee Related JP5280357B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US81950906P 2006-07-07 2006-07-07
US60/819,509 2006-07-07
US88682507P 2007-01-26 2007-01-26
US60/886,825 2007-01-26
PCT/US2007/072919 WO2008006050A2 (en) 2006-07-07 2007-07-06 Bicyclic heteroaryl inhibitors of pde4

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013107844A Division JP5705269B2 (ja) 2006-07-07 2013-05-22 Ｐｄｅ４の二環式ヘテロアリール阻害剤

Publications (3)

Publication Number Publication Date
JP2009542815A JP2009542815A (ja) 2009-12-03
JP2009542815A5 true JP2009542815A5 (enExample) 2010-08-26
JP5280357B2 JP5280357B2 (ja) 2013-09-04

Family

ID=38739981

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009519604A Expired - Fee Related JP5280357B2 (ja) 2006-07-07 2007-07-06 Ｐｄｅ４の二環式ヘテロアリール阻害剤
JP2013107844A Expired - Fee Related JP5705269B2 (ja) 2006-07-07 2013-05-22 Ｐｄｅ４の二環式ヘテロアリール阻害剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2013107844A Expired - Fee Related JP5705269B2 (ja) 2006-07-07 2013-05-22 Ｐｄｅ４の二環式ヘテロアリール阻害剤

Country Status (11)

Country Link
US (5) US20090291950A1 (enExample)
EP (1) EP2037924A2 (enExample)
JP (2) JP5280357B2 (enExample)
KR (2) KR20090109527A (enExample)
CN (1) CN104606194A (enExample)
AU (1) AU2007269070B2 (enExample)
BR (1) BRPI0713253A2 (enExample)
CA (1) CA2657093A1 (enExample)
CO (1) CO6190532A2 (enExample)
MX (1) MX2009000148A (enExample)
WO (3) WO2008006050A2 (enExample)

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US9890173B2 (en) 2013-11-01 2018-02-13 Kala Pharmaceuticals, Inc. Crystalline forms of therapeutic compounds and uses thereof
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US10131669B2 (en) 2014-07-24 2018-11-20 Pfizer Inc. Pyrazolopyrimidine compounds
HUE044040T2 (hu) 2014-08-06 2019-09-30 Pfizer Imidazopiridazin vegyületek
JP6740354B2 (ja) 2015-10-05 2020-08-12 ザ トラスティーズ オブ コロンビア ユニバーシティー イン ザ シティー オブ ニューヨーク オートファジーの流れ及びホスホリパーゼｄ及びタウを含むタンパク質凝集体のクリアランスの活性化剤ならびにタンパク質症の治療方法
AU2016379444B2 (en) * 2015-12-24 2021-04-29 The Regents Of The University Of California CFTR regulators and methods of use thereof
US10253036B2 (en) 2016-09-08 2019-04-09 Kala Pharmaceuticals, Inc. Crystalline forms of therapeutic compounds and uses thereof
EP3509423A4 (en) 2016-09-08 2020-05-13 Kala Pharmaceuticals, Inc. CRYSTALLINE FORMS OF THERAPEUTIC COMPOUNDS AND USES THEREOF
EP3509421A4 (en) 2016-09-08 2020-05-20 Kala Pharmaceuticals, Inc. CRYSTALLINE FORMS OF THERAPEUTIC COMPOUNDS AND USES THEREOF
CN106916104B (zh) * 2017-02-28 2019-08-27 牡丹江医学院 用于治疗结肠炎的药物
BR112019025578A2 (pt) 2017-07-26 2020-06-16 Hg&H Pharmaceuticals (Pty) Ltd Mesembrenol e/ou mesembranol para profilaxia e tratamento de pacientes que sofrem de epilepsia e doenças associadas
KR20200044873A (ko) 2017-08-24 2020-04-29 더 리젠츠 오브 더 유니버시티 오브 캘리포니아 안구 제약학적 조성물
CN113490739A (zh) * 2019-01-23 2021-10-08 通路治疗公司 通过磷酸二酯酶4(pde4)抑制治疗癫痫的方法
US20220371990A1 (en) * 2019-09-08 2022-11-24 Hadasit Medical Research Services And Developmect Ltd. Anti-fibrotic compounds and use thereof
CN116507336A (zh) * 2020-09-10 2023-07-28 Vanda制药公司 治疗pdeiv介导的疾病或病症的方法

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