JP2009539984A5 - - Google Patents

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Publication number
JP2009539984A5
JP2009539984A5 JP2009515443A JP2009515443A JP2009539984A5 JP 2009539984 A5 JP2009539984 A5 JP 2009539984A5 JP 2009515443 A JP2009515443 A JP 2009515443A JP 2009515443 A JP2009515443 A JP 2009515443A JP 2009539984 A5 JP2009539984 A5 JP 2009539984A5
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JP
Japan
Prior art keywords
pharmaceutical composition
pharmaceutically acceptable
carboxamide
dihydro
chloro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2009515443A
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English (en)
Japanese (ja)
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JP5226678B2 (ja
JP2009539984A (ja
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Priority claimed from PCT/US2007/013721 external-priority patent/WO2007146248A2/en
Publication of JP2009539984A publication Critical patent/JP2009539984A/ja
Publication of JP2009539984A5 publication Critical patent/JP2009539984A5/ja
Application granted granted Critical
Publication of JP5226678B2 publication Critical patent/JP5226678B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009515443A 2006-06-12 2007-06-12 安定性ラキニモド製剤 Expired - Fee Related JP5226678B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81324706P 2006-06-12 2006-06-12
US60/813,247 2006-06-12
PCT/US2007/013721 WO2007146248A2 (en) 2006-06-12 2007-06-12 Stable laquinimod preparations

Publications (3)

Publication Number Publication Date
JP2009539984A JP2009539984A (ja) 2009-11-19
JP2009539984A5 true JP2009539984A5 (enExample) 2012-03-08
JP5226678B2 JP5226678B2 (ja) 2013-07-03

Family

ID=38832466

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009515443A Expired - Fee Related JP5226678B2 (ja) 2006-06-12 2007-06-12 安定性ラキニモド製剤

Country Status (27)

Country Link
US (3) US7989473B2 (enExample)
EP (1) EP2035001B1 (enExample)
JP (1) JP5226678B2 (enExample)
KR (4) KR20140091778A (enExample)
CN (1) CN101466379B (enExample)
AR (1) AR061348A1 (enExample)
AT (1) ATE532515T1 (enExample)
AU (1) AU2007258366B2 (enExample)
BR (1) BRPI0713694A2 (enExample)
CA (2) CA2899472C (enExample)
CY (1) CY1113003T1 (enExample)
DK (1) DK2035001T3 (enExample)
EA (1) EA018031B1 (enExample)
ES (1) ES2377149T3 (enExample)
HR (1) HRP20120093T1 (enExample)
IL (1) IL195724A (enExample)
MX (1) MX2008015808A (enExample)
NO (1) NO342485B1 (enExample)
NZ (1) NZ573846A (enExample)
PL (1) PL2035001T3 (enExample)
PT (1) PT2035001E (enExample)
RS (1) RS52169B (enExample)
SI (1) SI2035001T1 (enExample)
TW (1) TWI400073B (enExample)
UA (1) UA96449C2 (enExample)
WO (1) WO2007146248A2 (enExample)
ZA (1) ZA200810790B (enExample)

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NZ573846A (en) 2006-06-12 2012-01-12 Teva Pharma Stable laquinimod preparations
EP2682120B1 (en) 2007-12-20 2016-08-03 Teva Pharmaceutical Industries, Ltd. Stable laquinimod preparations
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US20100322900A1 (en) 2009-06-19 2010-12-23 Teva Pharmaceutical Industries, Ltd. Treatment of multiple sclerosis with laquinimod
BR112012002124A2 (pt) * 2009-07-30 2015-09-15 Teva Pharma tratamento da doença de crohn com laquinimode.
DK2467372T3 (en) 2009-08-10 2016-08-22 Teva Pharma TREATMENT OF BDNF-RELATED DISEASES USING LAQUINIMOD
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BR112012022187A2 (pt) * 2010-03-03 2015-09-22 Teva Pharma tratamento de artrite reumatóide com a combinação de laquinimod e metotrexato
BR112012021905A2 (pt) * 2010-03-03 2015-09-29 Teva Pharma tratamento de nefrite lúpica usando laquinimod
KR20130092558A (ko) 2010-07-09 2013-08-20 테바 파마슈티컬 인더스트리즈 리미티드 중수소화된 n-에틸-n-페닐-1,2-다이하이드로-4-하이드록시-5-클로로-1-메틸-2-옥소퀴놀린-3-카복스아마이드, 그의 염 및 용도
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WO2013016686A1 (en) * 2011-07-28 2013-01-31 Teva Pharmaceutical Industries Ltd. Treatment of multiple sclerosis with combination of laquinimod and interferon-beta
EP2736335A4 (en) * 2011-07-28 2015-01-07 Teva Pharma TREATMENT OF MULTIPLE SCLEROSIS USING A COMBINATION OF LAQUINIMOD AND GLATIRAMERATE ACETATE
US8889627B2 (en) * 2011-10-12 2014-11-18 Teva Pharmaceutical Industries, Ltd. Treatment of multiple sclerosis with combination of laquinimod and fingolimod
CN106063787A (zh) 2012-02-03 2016-11-02 泰华制药工业有限公司 拉喹莫德用于治疗一线抗TNFα疗法失败的克罗恩氏病患者的用途
AU2013221304B2 (en) 2012-02-16 2017-12-21 Teva Pharmaceutical Industries Ltd. N-ethyl-N-phenyl-1,2-dihydro-4,5-di-hydroxy-1-methyl-2-oxo-3-quinoline carboxamide, preparation and uses thereof
US20130259856A1 (en) * 2012-03-27 2013-10-03 Teva Pharmaceutical Industries, Ltd. Treatment of multiple sclerosis with combination of laquinimod and dimethyl fumarate
TW201350467A (zh) * 2012-05-08 2013-12-16 Teva Pharma Ｎ－乙基－４－羥基－１－甲基－５－（甲基（２，３，４，５，６－五羥基己基）胺基）－２－側氧－ｎ－苯基－１，２－二氫喹啉－３－甲醯胺
TW201400117A (zh) 2012-06-05 2014-01-01 Teva Pharma 使用拉喹莫德治療眼發炎疾病
US20130345257A1 (en) * 2012-06-26 2013-12-26 The Regents Of The University Of California Composition for lupus nephritis and methods of making and using the same
AR091706A1 (es) * 2012-07-11 2015-02-25 Teva Pharma Formulaciones de laquinimod sin agentes alcalinizantes
TW201410243A (zh) * 2012-08-13 2014-03-16 Teva Pharma 用於治療大麻素受體型１（ｃｂ１）媒介之疾病之拉喹莫德（ｌａｑｕｉｎｉｍｏｄ）
TW201410244A (zh) 2012-08-13 2014-03-16 Teva Pharma 用於治療ｇａｂａ媒介之疾病之拉喹莫德（ｌａｑｕｉｎｉｍｏｄ）
EA201590788A1 (ru) 2012-11-07 2015-12-30 Тева Фармасьютикал Индастриз Лтд. Аминные соли лахинимода
CA2900503A1 (en) * 2013-02-15 2014-08-21 Teva Pharmaceutical Industries Ltd. Treatment of multiple sclerosis with laquinimod
AU2014236232A1 (en) * 2013-03-14 2015-11-05 Teva Pharmaceutical Industries Ltd. Crystals of laquinimod sodium and improved process for the manufacture thereof
MX2015010967A (es) 2013-03-14 2015-10-26 Teva Pharma Formulaciones transdermicas de laquinimod.
UY35748A (es) * 2013-09-27 2015-04-30 Teva Pharma Terapia combinada con laquinimod para el tratamiento de la esclerosis múltiple
AU2014364447A1 (en) * 2013-12-20 2016-08-04 Teva Pharmaceutical Industries Ltd. Use of laquinimod to delay Huntington's disease progression
EP3094330A4 (en) * 2014-01-17 2017-09-27 Teva Pharmaceutical Industries Ltd Treatment of crohn's disease using low doses of laquinimod
JP2017514824A (ja) 2014-04-29 2017-06-08 テバ ファーマシューティカル インダストリーズ リミティド 能力障害度が高い再発寛解型多発性硬化症（ｒｒｍｓ）患者の処置のためのラキニモド
CN110193014B (zh) * 2019-06-06 2021-05-11 温州医科大学 一种注射用拉喹莫德胶束冻干制剂及制备方法、拉喹莫德注射制剂

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BR112012002124A2 (pt) 2009-07-30 2015-09-15 Teva Pharma tratamento da doença de crohn com laquinimode.
DK2467372T3 (en) 2009-08-10 2016-08-22 Teva Pharma TREATMENT OF BDNF-RELATED DISEASES USING LAQUINIMOD
BR112012021905A2 (pt) 2010-03-03 2015-09-29 Teva Pharma tratamento de nefrite lúpica usando laquinimod
KR20130036217A (ko) 2010-03-03 2013-04-11 테바 파마슈티컬 인더스트리즈 리미티드 라퀴니모드를 이용한 루푸스 관절염의 치료
BR112012022187A2 (pt) 2010-03-03 2015-09-22 Teva Pharma tratamento de artrite reumatóide com a combinação de laquinimod e metotrexato
JP5934202B2 (ja) 2010-07-09 2016-06-15 テバ ファーマシューティカル インダストリーズ リミティド ５−クロロ−４−ヒドロキシ−１−メチル−２−オキソ−ｎ−フェニル−１，２−ジヒドロキノリン−３−カルボキサミドと、その塩及びその使用
KR20130092558A (ko) 2010-07-09 2013-08-20 테바 파마슈티컬 인더스트리즈 리미티드 중수소화된 n-에틸-n-페닐-1,2-다이하이드로-4-하이드록시-5-클로로-1-메틸-2-옥소퀴놀린-3-카복스아마이드, 그의 염 및 용도

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