JP2009533393A5 - - Google Patents

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Publication number
JP2009533393A5
JP2009533393A5 JP2009504750A JP2009504750A JP2009533393A5 JP 2009533393 A5 JP2009533393 A5 JP 2009533393A5 JP 2009504750 A JP2009504750 A JP 2009504750A JP 2009504750 A JP2009504750 A JP 2009504750A JP 2009533393 A5 JP2009533393 A5 JP 2009533393A5
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JP
Japan
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alkyl
heteroaryl
aryl
alkynyl
alkenyl
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Abandoned
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JP2009504750A
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English (en)
Japanese (ja)
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JP2009533393A (ja
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Priority claimed from PCT/EP2007/053560 external-priority patent/WO2007116092A1/en
Publication of JP2009533393A publication Critical patent/JP2009533393A/ja
Publication of JP2009533393A5 publication Critical patent/JP2009533393A5/ja
Abandoned legal-status Critical Current

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JP2009504750A 2006-04-12 2007-04-12 酵素阻害薬 Abandoned JP2009533393A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79130206P 2006-04-12 2006-04-12
US87016506P 2006-12-15 2006-12-15
PCT/EP2007/053560 WO2007116092A1 (en) 2006-04-12 2007-04-12 Enzyme inhibitors

Publications (2)

Publication Number Publication Date
JP2009533393A JP2009533393A (ja) 2009-09-17
JP2009533393A5 true JP2009533393A5 (https=) 2010-05-27

Family

ID=38256669

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009504750A Abandoned JP2009533393A (ja) 2006-04-12 2007-04-12 酵素阻害薬

Country Status (12)

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US (2) US7728146B2 (https=)
EP (1) EP2007734A1 (https=)
JP (1) JP2009533393A (https=)
KR (1) KR20090004950A (https=)
AU (1) AU2007235876A1 (https=)
BR (1) BRPI0709984A2 (https=)
CA (1) CA2649209A1 (https=)
EA (1) EA200802054A1 (https=)
IL (1) IL194339A0 (https=)
MX (1) MX2008013130A (https=)
NZ (1) NZ571761A (https=)
WO (1) WO2007116092A1 (https=)

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EP2582709B1 (de) 2010-06-18 2018-01-24 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
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EP2766349B1 (de) 2011-03-08 2016-06-01 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2683699B1 (de) 2011-03-08 2015-06-24 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120056A1 (de) 2011-03-08 2012-09-13 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683704B1 (de) 2011-03-08 2014-12-17 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
US20150297573A1 (en) 2012-10-24 2015-10-22 INSERM (Institut National de la Santé et de la Recherche Médicale) TPL2 KINASE INHIBITORS FOR PREVENTING OR TREATING DIABETES AND FOR PROMOTING Beta-CELL SURVIVAL
PT3598971T (pt) 2013-01-22 2024-06-20 Vistagen Therapeutics Inc ¿formas de dosagem e utilizações terapêuticas de l-4 cloroquinurenina
US10426818B2 (en) 2015-03-24 2019-10-01 Inserm (Institut National De La Sante Et De La Recherche Medicale) Method and pharmaceutical composition for use in the treatment of diabetes
JP2018521007A (ja) * 2015-05-22 2018-08-02 ヴィスタゲン セラピューティクス、インコーポレイテッド Ｌ−４−クロロキヌレニンの治療的使用
JP2019089710A (ja) * 2016-03-22 2019-06-13 国立研究開発法人科学技術振興機構 イミダゾール化合物及びこれを含有する医薬
RU2614737C1 (ru) * 2016-04-12 2017-03-28 Общество с ограниченной ответственностью "Нормофарм" Способ улучшения памяти

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