JP2008521827A - Ｓ１ｐ受容体アゴニストの投与レジメン - Google Patents
Ｓ１ｐ受容体アゴニストの投与レジメン Download PDFInfo
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- JP2008521827A JP2008521827A JP2007543584A JP2007543584A JP2008521827A JP 2008521827 A JP2008521827 A JP 2008521827A JP 2007543584 A JP2007543584 A JP 2007543584A JP 2007543584 A JP2007543584 A JP 2007543584A JP 2008521827 A JP2008521827 A JP 2008521827A
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- agonist
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Landscapes
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| JP2013043351A Division JP2013129664A (ja) | 2004-11-29 | 2013-03-05 | Ｓ１ｐ受容体アゴニストの投与レジメン |
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| JP2013043351A Withdrawn JP2013129664A (ja) | 2004-11-29 | 2013-03-05 | Ｓ１ｐ受容体アゴニストの投与レジメン |
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| JP2014266267A Pending JP2015061883A (ja) | 2004-11-29 | 2014-12-26 | Ｓ１ｐ受容体アゴニストの投与レジメン |
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| EP (3) | EP2384749A1 (https=) |
| JP (4) | JP2008521827A (https=) |
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Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012500247A (ja) * | 2008-08-18 | 2012-01-05 | ノバルティス アーゲー | 末梢神経障害の治療のための化合物 |
| JP2012512881A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | １−［４−［１−（４−シクロヘキシル−３−トリフルオロメチル−ベンジルオキシイミノ）−エチル］−２−エチル−ベンジル］−アゼチジン−３−カルボン酸ヘミフマル酸塩 |
| JP2012512885A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | 新規な塩 |
| JP2012107059A (ja) * | 2004-11-29 | 2012-06-07 | Novartis Ag | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2012513401A (ja) * | 2008-12-22 | 2012-06-14 | ノバルティス アーゲー | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2016155840A (ja) * | 2009-09-29 | 2016-09-01 | ノバルティス アーゲー | Ｓ１ｐ受容体モジュレーターの投与計画 |
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| MX2007001661A (es) | 2004-08-13 | 2007-04-23 | Praecis Pharm Inc | Metodos y composiciones para modular la actividad del receptor de esfingosina -1 fosfato (sip). |
| SI2295049T1 (sl) * | 2005-09-09 | 2015-03-31 | Novartis Ag | Zdravljenje avtoimunskih bolezni |
| GB0612721D0 (en) * | 2006-06-27 | 2006-08-09 | Novartis Ag | Organic compounds |
| ES2707576T3 (es) | 2007-05-04 | 2019-04-04 | Novartis Ag | Uso de modulador del receptor S1P |
| HUE033168T2 (en) * | 2008-03-17 | 2017-11-28 | Actelion Pharmaceuticals Ltd | Dosage regimen for selective SIP1 receptor agonist |
| NZ589412A (en) * | 2008-05-20 | 2012-11-30 | Kyorin Seiyaku Kk | Use of a sphingosine-1-phosphate (S1P) agonist for maintance of induced remission of autoimmune or inflammatory diseases after inital treatment |
| US9149459B2 (en) | 2008-07-23 | 2015-10-06 | Novartis Ag | Sphingosine 1 phosphate receptor modulators and their use to treat muscle inflammation |
| CN102256942B (zh) * | 2008-12-18 | 2013-07-24 | 诺瓦提斯公司 | 1-(4-{1-[(e)-4-环己基-3-三氟甲基-苄氧基亚氨基]-乙基}-2-乙基-苄基)-氮杂环丁烷-3-甲酸的多晶型物 |
| CN105213372A (zh) * | 2008-12-22 | 2016-01-06 | 诺华股份有限公司 | S1p受体激动剂的给药方案 |
| AU2015275246B2 (en) * | 2008-12-22 | 2018-02-01 | Novartis Ag | Dosage regimen for a S1P receptor agonist |
| US20110124605A1 (en) * | 2009-11-20 | 2011-05-26 | Shreeram Aradhye | Use of an S1P Receptor Agonist |
| US8791100B2 (en) | 2010-02-02 | 2014-07-29 | Novartis Ag | Aryl benzylamine compounds |
| EP2566473B1 (en) * | 2010-05-06 | 2016-01-06 | Novartis AG | Dosage regimen of diaryl sulfide derivatives |
| BR112013017302B1 (pt) | 2011-01-07 | 2021-12-07 | Novartis Ag | Composição farmacêutica em fase sólida |
| PH12014500854A1 (en) * | 2011-10-21 | 2021-08-09 | Novartis Ag | Dosage regimen for an s1p receptor modulator or agonist |
| MX350891B (es) | 2012-08-17 | 2017-09-22 | Actelion Pharmaceuticals Ltd | Proceso para la preparacion de (2z,5z)-5-(3-cloro-4-((r)-2,3-dihid roxipropoxi) bencilideno)-2-(propilimino)-3-(o-tolil) tiazolidin-4-ona y el intermediario usado en dicho proceso. |
| CN102887829B (zh) * | 2012-09-05 | 2014-07-02 | 中国科学院上海药物研究所 | 芬戈莫德粘酸盐及其晶体的制备方法和用途 |
| US10675254B2 (en) | 2013-10-11 | 2020-06-09 | Teikoku Seiyaku Co., Ltd. | Sphingosine-1-phosphate receptor agonist iontophoretic devices and methods of using the same |
| JP6401257B2 (ja) | 2013-10-11 | 2018-10-10 | テイコク ファーマ ユーエスエー インコーポレーテッド | 局所用スフィンゴシン−１−リン酸受容体アゴニスト製剤及びその使用方法 |
| MA41139B1 (fr) | 2014-12-11 | 2026-02-27 | Laboratoires Juvise Pharmaceuticals | Combinaison pharmaceutique comprenant du ponesimod et son utilisation dans le traitement de la sclérose en plaque |
| EP4056179A1 (en) | 2014-12-11 | 2022-09-14 | Actelion Pharmaceuticals Ltd | Dosing regimen for ponesimod, a selective s1p1 receptor agonist |
| WO2016135644A1 (en) | 2015-02-26 | 2016-09-01 | Novartis Ag | Treatment of autoimmune disease in a patient receiving additionally a beta-blocker |
| US10250466B2 (en) * | 2016-03-29 | 2019-04-02 | Juniper Networks, Inc. | Application signature generation and distribution |
| US11629124B2 (en) | 2017-03-09 | 2023-04-18 | Novartis Ag | Solid forms comprising an oxime ether compound, compositions and methods of use thereof |
| AU2020372647B2 (en) | 2019-10-31 | 2026-02-05 | Idorsia Pharmaceuticals Ltd | Combination of a CXCR7 antagonist with an S1P1 receptor modulator |
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| ATE298740T1 (de) | 1997-04-04 | 2005-07-15 | Mitsubishi Pharma Corp | 2-aminopropan-1,3-diol-verbindungen, ihre medizinische anwendung und zwischenprodukte zu ihrer synthese |
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- 2005-11-28 RU RU2007124327/15A patent/RU2478384C2/ru not_active IP Right Cessation
- 2005-11-28 PL PL05826219T patent/PL1819326T3/pl unknown
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| JP2012107059A (ja) * | 2004-11-29 | 2012-06-07 | Novartis Ag | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2012500247A (ja) * | 2008-08-18 | 2012-01-05 | ノバルティス アーゲー | 末梢神経障害の治療のための化合物 |
| JP2012512881A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | １−［４−［１−（４−シクロヘキシル−３−トリフルオロメチル−ベンジルオキシイミノ）−エチル］−２−エチル−ベンジル］−アゼチジン−３−カルボン酸ヘミフマル酸塩 |
| JP2012512885A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | 新規な塩 |
| JP2012513401A (ja) * | 2008-12-22 | 2012-06-14 | ノバルティス アーゲー | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2014144970A (ja) * | 2008-12-22 | 2014-08-14 | Novartis Ag | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2017141238A (ja) * | 2008-12-22 | 2017-08-17 | ノバルティス アーゲー | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2019167360A (ja) * | 2008-12-22 | 2019-10-03 | ノバルティス アーゲー | Ｓ１ｐ受容体アゴニストの投与レジメン |
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