JP2008521827A - Ｓ１ｐ受容体アゴニストの投与レジメン - Google Patents
Ｓ１ｐ受容体アゴニストの投与レジメン Download PDFInfo
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- JP2008521827A JP2008521827A JP2007543584A JP2007543584A JP2008521827A JP 2008521827 A JP2008521827 A JP 2008521827A JP 2007543584 A JP2007543584 A JP 2007543584A JP 2007543584 A JP2007543584 A JP 2007543584A JP 2008521827 A JP2008521827 A JP 2008521827A
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- agonist
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Landscapes
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Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012500247A (ja) * | 2008-08-18 | 2012-01-05 | ノバルティス アーゲー | 末梢神経障害の治療のための化合物 |
| JP2012512881A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | １−［４−［１−（４−シクロヘキシル−３−トリフルオロメチル−ベンジルオキシイミノ）−エチル］−２−エチル−ベンジル］−アゼチジン−３−カルボン酸ヘミフマル酸塩 |
| JP2012107059A (ja) * | 2004-11-29 | 2012-06-07 | Novartis Ag | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2012512885A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | 新規な塩 |
| JP2012513401A (ja) * | 2008-12-22 | 2012-06-14 | ノバルティス アーゲー | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2016155840A (ja) * | 2009-09-29 | 2016-09-01 | ノバルティス アーゲー | Ｓ１ｐ受容体モジュレーターの投与計画 |
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| US7241812B2 (en) | 2004-08-13 | 2007-07-10 | Praecis Pharmaceuticals, Inc. | Methods and compositions for modulating sphingosine-1-phosphate (S1P) receptor activity |
| ES2357426T3 (es) * | 2005-09-09 | 2011-04-26 | Novartis Ag | Tratamiento de enfermedades autoinmunes. |
| GB0612721D0 (en) * | 2006-06-27 | 2006-08-09 | Novartis Ag | Organic compounds |
| CN104337808A (zh) | 2007-05-04 | 2015-02-11 | 诺华股份有限公司 | S1p受体调节剂的用途 |
| LT2278960T (lt) * | 2008-03-17 | 2017-02-10 | Actelion Pharmaceuticals Ltd. | S1p1 receptoriaus selektyvaus agonisto dozavimo režimas |
| CA2724592A1 (en) * | 2008-05-20 | 2009-11-26 | Kyorin Pharmaceutical Co., Ltd. | Agent for maintenance of induced remission |
| KR101608108B1 (ko) * | 2008-07-23 | 2016-03-31 | 노파르티스 아게 | 스핑고신 1 포스페이트 수용체 조절제 및 근육 염증을 치료하기 위한 그의 용도 |
| BRPI0922457A2 (pt) * | 2008-12-18 | 2015-12-15 | Novartis Ag | forma polimórfica de ácido 1-(4-{1-[(e)-4-ciclo-hexil-3-trifluormetil-benziloxi-imino]-etil)-2-etil-benzil)-azetidino-3-carboxílico" |
| CA2747992C (en) * | 2008-12-22 | 2017-11-07 | Novartis Ag | Dosage regimen of an s1p receptor agonist |
| AU2015275246B2 (en) * | 2008-12-22 | 2018-02-01 | Novartis Ag | Dosage regimen for a S1P receptor agonist |
| US20110124605A1 (en) * | 2009-11-20 | 2011-05-26 | Shreeram Aradhye | Use of an S1P Receptor Agonist |
| US8791100B2 (en) | 2010-02-02 | 2014-07-29 | Novartis Ag | Aryl benzylamine compounds |
| AU2011249789B2 (en) * | 2010-05-06 | 2015-03-19 | Novartis Ag | Dosage regimen of diaryl sulfide derivatives |
| UA114283C2 (uk) | 2011-01-07 | 2017-05-25 | Новартіс Аг | Композиції імуносупресантів |
| SG10201602279PA (en) * | 2011-10-21 | 2016-04-28 | Novartis Ag | Dosage regimen for an s1p receptor modulator or agonist |
| HUE050733T2 (hu) | 2012-08-17 | 2021-01-28 | Actelion Pharmaceuticals Ltd | Eljárás (2Z,5Z)-5-(3-klór-4-((R)-2,3-dihidroxipropoxi)benzilidén)-2-(pro-pilimino)-3-(O-tolil)tiazolidin-4-on elõállítására és ezen eljárásban alkalmazott köztitermék |
| CN102887829B (zh) * | 2012-09-05 | 2014-07-02 | 中国科学院上海药物研究所 | 芬戈莫德粘酸盐及其晶体的制备方法和用途 |
| US10675254B2 (en) | 2013-10-11 | 2020-06-09 | Teikoku Seiyaku Co., Ltd. | Sphingosine-1-phosphate receptor agonist iontophoretic devices and methods of using the same |
| WO2015053878A1 (en) | 2013-10-11 | 2015-04-16 | Teikoku Pharma Usa, Inc. | Topical sphingosine-1-phosphate receptor agonist formulations and methods of using the same |
| MA41139A (fr) | 2014-12-11 | 2017-10-17 | Actelion Pharmaceuticals Ltd | Combinaison pharmaceutique comportant un agoniste sélectif du récepteur sip1 |
| HRP20220359T8 (hr) | 2014-12-11 | 2022-05-27 | Actelion Pharmaceuticals Ltd | Režim doziranja ponesimoda, selektivnog agonista receptora s1p1 |
| WO2016135644A1 (en) | 2015-02-26 | 2016-09-01 | Novartis Ag | Treatment of autoimmune disease in a patient receiving additionally a beta-blocker |
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| US11629124B2 (en) | 2017-03-09 | 2023-04-18 | Novartis Ag | Solid forms comprising an oxime ether compound, compositions and methods of use thereof |
| AU2020372647A1 (en) | 2019-10-31 | 2022-06-16 | Idorsia Pharmaceuticals Ltd | Combination of a CXCR7 antagonist with an S1P1 receptor modulator |
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| JPH1180026A (ja) * | 1997-09-02 | 1999-03-23 | Yoshitomi Pharmaceut Ind Ltd | 新規免疫抑制剤、その使用方法およびその同定方法 |
| BR0112484A (pt) | 2000-07-13 | 2003-09-23 | Sankyo Co | Composto ou um seu sal, éster ou outro derivado farmacologicamente aceitável, composição farmacêutica, uso de um composto ou de um seu sal, éster ou outro derivado farmacologicamente aceitável, e, processo para a preparação do mesmo |
| AU8533101A (en) | 2000-08-31 | 2002-03-13 | Merck & Co Inc | Phosphate derivatives as immunoregulatory agents |
| JP4012823B2 (ja) | 2001-03-26 | 2007-11-21 | ノバルティス アクチエンゲゼルシャフト | ２−アミノ−誘導体 |
| JP2002316985A (ja) | 2001-04-20 | 2002-10-31 | Sankyo Co Ltd | ベンゾチオフェン誘導体 |
| NZ529044A (en) * | 2001-06-08 | 2008-03-28 | Novartis Ag | Treatment or prophylaxis of insulin-producing cell graft rejection |
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| BRPI0212894B8 (pt) | 2001-09-27 | 2021-05-25 | Kyorin Seiyaku Kk | composto ou sal do mesmo farmaceuticamente aceitável e composição farmacêutica |
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- 2005-11-28 KR KR1020147018084A patent/KR20140095109A/ko not_active Withdrawn
- 2005-11-28 EP EP10179081A patent/EP2359821A1/en not_active Withdrawn
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| JP2012107059A (ja) * | 2004-11-29 | 2012-06-07 | Novartis Ag | Ｓ１ｐ受容体アゴニストの投与レジメン |
| JP2012500247A (ja) * | 2008-08-18 | 2012-01-05 | ノバルティス アーゲー | 末梢神経障害の治療のための化合物 |
| JP2012512881A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | １−［４−［１−（４−シクロヘキシル−３−トリフルオロメチル−ベンジルオキシイミノ）−エチル］−２−エチル−ベンジル］−アゼチジン−３−カルボン酸ヘミフマル酸塩 |
| JP2012512885A (ja) * | 2008-12-18 | 2012-06-07 | ノバルティス アーゲー | 新規な塩 |
| JP2012513401A (ja) * | 2008-12-22 | 2012-06-14 | ノバルティス アーゲー | Ｓ１ｐ受容体アゴニストの投与レジメン |
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| JP2019167360A (ja) * | 2008-12-22 | 2019-10-03 | ノバルティス アーゲー | Ｓ１ｐ受容体アゴニストの投与レジメン |
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