JP2007514712A5 - - Google Patents

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Publication number
JP2007514712A5
JP2007514712A5 JP2006544440A JP2006544440A JP2007514712A5 JP 2007514712 A5 JP2007514712 A5 JP 2007514712A5 JP 2006544440 A JP2006544440 A JP 2006544440A JP 2006544440 A JP2006544440 A JP 2006544440A JP 2007514712 A5 JP2007514712 A5 JP 2007514712A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2006544440A
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English (en)
Japanese (ja)
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JP4936897B2 (ja
JP2007514712A (ja
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Priority claimed from PCT/EP2004/053501 external-priority patent/WO2005058913A1/en
Publication of JP2007514712A publication Critical patent/JP2007514712A/ja
Publication of JP2007514712A5 publication Critical patent/JP2007514712A5/ja
Application granted granted Critical
Publication of JP4936897B2 publication Critical patent/JP4936897B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2006544440A 2003-12-18 2004-12-15 抗増殖剤としてのピリド−およびピリミドピリミジン誘導体 Expired - Lifetime JP4936897B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EPPCT/EP03/51062 2003-12-18
EPPCT/EP03/51058 2003-12-18
EP0351062 2003-12-18
EP0351058 2003-12-18
PCT/EP2004/053501 WO2005058913A1 (en) 2003-12-18 2004-12-15 Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents

Publications (3)

Publication Number Publication Date
JP2007514712A JP2007514712A (ja) 2007-06-07
JP2007514712A5 true JP2007514712A5 (enExample) 2012-03-08
JP4936897B2 JP4936897B2 (ja) 2012-05-23

Family

ID=34702160

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006544440A Expired - Lifetime JP4936897B2 (ja) 2003-12-18 2004-12-15 抗増殖剤としてのピリド−およびピリミドピリミジン誘導体

Country Status (18)

Country Link
US (3) US7799772B2 (enExample)
EP (1) EP1697384B1 (enExample)
JP (1) JP4936897B2 (enExample)
KR (1) KR101174672B1 (enExample)
AR (1) AR046957A1 (enExample)
AU (1) AU2004298448B2 (enExample)
CA (1) CA2549869C (enExample)
DE (1) DE602004012891T2 (enExample)
EA (1) EA013904B1 (enExample)
ES (1) ES2305887T3 (enExample)
IL (1) IL176357A (enExample)
MX (1) MXPA06007017A (enExample)
MY (1) MY146415A (enExample)
NO (1) NO337701B1 (enExample)
NZ (1) NZ547794A (enExample)
TW (1) TWI347187B (enExample)
UA (1) UA83881C2 (enExample)
WO (1) WO2005058913A1 (enExample)

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JP6800158B2 (ja) 2015-02-20 2020-12-16 ライジェル ファーマシューティカルズ， インコーポレイテッド Ｇｄｆ−８阻害剤
MX2018004109A (es) 2015-10-05 2018-09-27 Univ Columbia Activadores de flujo autofágico y fosfolipasa d y depuración de acumulaciones de proteína que incluyen tau y tratamiento de proteinopatías.
US10724102B2 (en) 2015-10-26 2020-07-28 Loxo Oncology, Inc. Point mutations in TRK inhibitor-resistant cancer and methods relating to the same
SG11201808559PA (en) 2016-04-04 2018-10-30 Loxo Oncology Inc Liquid formulations of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide
US10045991B2 (en) 2016-04-04 2018-08-14 Loxo Oncology, Inc. Methods of treating pediatric cancers
FI3800189T3 (fi) 2016-05-18 2023-07-31 Loxo Oncology Inc (s)-n-(5-((r)-2-(2,5-difluorifenyyli)pyrrolidin-1-yyli)pyratsolo[1,5-a]pyrimidin-3-yyli)-3-hydroksipyrrolidiini-1-karboksamidin valmistaminen
JOP20190092A1 (ar) 2016-10-26 2019-04-25 Array Biopharma Inc عملية لتحضير مركبات بيرازولو[1، 5-a]بيريميدين وأملاح منها
JOP20190213A1 (ar) 2017-03-16 2019-09-16 Array Biopharma Inc مركبات حلقية ضخمة كمثبطات لكيناز ros1
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ES2435454T3 (es) 2007-06-21 2013-12-19 Janssen Pharmaceutica, N.V. Indolin-2-onas y aza-indolin-2-onas
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