SI2256108T1 - Substituirani triazinski kinazni inhibitorji - Google Patents

Substituirani triazinski kinazni inhibitorji

Info

Publication number
SI2256108T1
SI2256108T1 SI200332475A SI200332475A SI2256108T1 SI 2256108 T1 SI2256108 T1 SI 2256108T1 SI 200332475 A SI200332475 A SI 200332475A SI 200332475 A SI200332475 A SI 200332475A SI 2256108 T1 SI2256108 T1 SI 2256108T1
Authority
SI
Slovenia
Prior art keywords
kinase inhibitors
substituted triazine
triazine kinase
substituted
inhibitors
Prior art date
Application number
SI200332475A
Other languages
English (en)
Inventor
Gee-Hong Kuo
Alan Deangelis
Aihua Wang
Yan Zhang
Stuart L Emanuel
Steve A Middleton
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of SI2256108T1 publication Critical patent/SI2256108T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SI200332475A 2002-07-18 2003-07-18 Substituirani triazinski kinazni inhibitorji SI2256108T1 (sl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39694802P 2002-07-18 2002-07-18
EP10176670.7A EP2256108B1 (en) 2002-07-18 2003-07-18 Substituted triazine kinase inhibitors

Publications (1)

Publication Number Publication Date
SI2256108T1 true SI2256108T1 (sl) 2016-05-31

Family

ID=30770960

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200332475A SI2256108T1 (sl) 2002-07-18 2003-07-18 Substituirani triazinski kinazni inhibitorji

Country Status (9)

Country Link
US (1) US7205298B2 (sl)
EP (2) EP2256108B1 (sl)
AU (1) AU2003259153A1 (sl)
CY (1) CY1117951T1 (sl)
DK (1) DK2256108T3 (sl)
ES (2) ES2392426T3 (sl)
HU (1) HUE029020T2 (sl)
SI (1) SI2256108T1 (sl)
WO (1) WO2004009562A1 (sl)

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Also Published As

Publication number Publication date
ES2392426T3 (es) 2012-12-10
US7205298B2 (en) 2007-04-17
HUE029020T2 (en) 2017-02-28
ES2575522T3 (es) 2016-06-29
US20040082581A1 (en) 2004-04-29
EP1546121B1 (en) 2012-08-29
EP2256108A1 (en) 2010-12-01
CY1117951T1 (el) 2017-05-17
EP1546121A1 (en) 2005-06-29
AU2003259153A1 (en) 2004-02-09
DK2256108T3 (en) 2016-04-11
EP2256108B1 (en) 2016-03-23
EP1546121A4 (en) 2007-08-15
WO2004009562A1 (en) 2004-01-29

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