JP2007508301A5 - - Google Patents

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Publication number
JP2007508301A5
JP2007508301A5 JP2006533949A JP2006533949A JP2007508301A5 JP 2007508301 A5 JP2007508301 A5 JP 2007508301A5 JP 2006533949 A JP2006533949 A JP 2006533949A JP 2006533949 A JP2006533949 A JP 2006533949A JP 2007508301 A5 JP2007508301 A5 JP 2007508301A5
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JP
Japan
Prior art keywords
alkyl
amino
tetrahydro
benzyl
carboxylic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2006533949A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007508301A (ja
JP4773969B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2004/030907 external-priority patent/WO2005037796A1/en
Publication of JP2007508301A publication Critical patent/JP2007508301A/ja
Publication of JP2007508301A5 publication Critical patent/JP2007508301A5/ja
Application granted granted Critical
Publication of JP4773969B2 publication Critical patent/JP4773969B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2006533949A 2003-10-08 2004-10-07 脂質代謝異常の治療ための化合物及び方法 Expired - Fee Related JP4773969B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US50973603P 2003-10-08 2003-10-08
US60/509,736 2003-10-08
PCT/US2004/030907 WO2005037796A1 (en) 2003-10-08 2004-10-07 Compounds and methods for treating dyslipidemia

Publications (3)

Publication Number Publication Date
JP2007508301A JP2007508301A (ja) 2007-04-05
JP2007508301A5 true JP2007508301A5 (https=) 2011-05-19
JP4773969B2 JP4773969B2 (ja) 2011-09-14

Family

ID=34465112

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006533949A Expired - Fee Related JP4773969B2 (ja) 2003-10-08 2004-10-07 脂質代謝異常の治療ための化合物及び方法

Country Status (25)

Country Link
US (1) US7749992B2 (https=)
EP (2) EP2098512A1 (https=)
JP (1) JP4773969B2 (https=)
KR (1) KR20060085675A (https=)
CN (1) CN1863778A (https=)
AT (1) ATE442358T1 (https=)
AU (1) AU2004282101A1 (https=)
BR (1) BRPI0414186A (https=)
CA (1) CA2537942A1 (https=)
CY (1) CY1110537T1 (https=)
DE (1) DE602004023100D1 (https=)
DK (1) DK1670768T3 (https=)
EA (1) EA200600737A1 (https=)
EC (1) ECSP066484A (https=)
ES (1) ES2332051T3 (https=)
HR (1) HRP20090581T1 (https=)
IL (1) IL173819A0 (https=)
MA (1) MA28268A1 (https=)
MX (1) MXPA06003927A (https=)
NO (1) NO20062074L (https=)
PL (1) PL1670768T3 (https=)
PT (1) PT1670768E (https=)
SI (1) SI1670768T1 (https=)
WO (1) WO2005037796A1 (https=)
ZA (1) ZA200602888B (https=)

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WO2005097805A1 (en) * 2004-03-26 2005-10-20 Eli Lilly And Company Compounds and methods for treating dyslipidemia
AU2005267436A1 (en) 2004-06-24 2006-02-02 Eli Lilly And Company Compounds and methods for treating dyslipidemia
US7790770B2 (en) 2005-11-23 2010-09-07 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
US7652023B2 (en) * 2005-11-23 2010-01-26 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
AR077208A1 (es) * 2009-06-30 2011-08-10 Lilly Co Eli Derivados del acido trans-4-[[(5s)-5-[[[3,5-bis(trifluorometil) fenil] metil] (2-metil-2h-tetrazol-5-il) amino) -2,3,4,5-tetrahidro-7,9-dimetil-1h-1-benzazepin-1-il) metil)-ciclohexancarboxilico y sus formas cristalinas, composiciones farmaceuticas que los comprenden, su uso para preparar un medicam
CN103833636B (zh) * 2014-03-31 2015-09-02 武汉武药制药有限公司 一种莫扎伐普坦中间体的合成方法
CA3002525A1 (en) * 2015-07-31 2017-02-09 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists and compositions and methods of use
CN110291383B (zh) * 2017-02-23 2021-12-28 株式会社Ihi Oh自由基检测探测器、oh自由基测定装置以及oh自由基测定方法
MX2021004593A (es) 2018-10-24 2021-06-15 Viiv Healthcare Uk No 5 Ltd Inhibidores de la replicacion del virus de la inmunodeficiencia humana.
CN115397424A (zh) 2020-04-15 2022-11-25 Viiv保健英国第五有限公司 人类免疫缺陷病毒复制的抑制剂
CN113636977B (zh) * 2021-09-01 2022-12-20 温州大学 2-芳基苯并氮杂卓及其衍生物的合成方法
CN117088814A (zh) * 2023-02-16 2023-11-21 烟台大学 一种三氟甲硫化氮杂-8/9元环化合物的制备方法

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WO2005097805A1 (en) * 2004-03-26 2005-10-20 Eli Lilly And Company Compounds and methods for treating dyslipidemia
AU2005267436A1 (en) * 2004-06-24 2006-02-02 Eli Lilly And Company Compounds and methods for treating dyslipidemia

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