JP2006524636A5 - - Google Patents

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Publication number
JP2006524636A5
JP2006524636A5 JP2006500346A JP2006500346A JP2006524636A5 JP 2006524636 A5 JP2006524636 A5 JP 2006524636A5 JP 2006500346 A JP2006500346 A JP 2006500346A JP 2006500346 A JP2006500346 A JP 2006500346A JP 2006524636 A5 JP2006524636 A5 JP 2006524636A5
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JP
Japan
Prior art keywords
nme
nhme
nhco
halo
oxo
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JP2006500346A
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English (en)
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JP2006524636A (ja
JP4015176B2 (ja
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Priority claimed from GBGB0327748.0A external-priority patent/GB0327748D0/en
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Priority claimed from PCT/IB2004/001433 external-priority patent/WO2004096810A1/en
Publication of JP2006524636A publication Critical patent/JP2006524636A/ja
Publication of JP2006524636A5 publication Critical patent/JP2006524636A5/ja
Application granted granted Critical
Publication of JP4015176B2 publication Critical patent/JP4015176B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Description

より好ましくは、R10は、ハロ、メチル、エチル、イソプロピル、ヒドロキシ、メトキシ、NH、NHMe、NMe、NHCO Bu、COH、CO Bu、オキソ、ベンジル、−CHOH、−CHNH、CHNHMe、−CHNMeまたは−CHNMe Buである。
JP2006500346A 2003-04-29 2004-04-22 高血圧症の治療に有用な5,7−ジアミノピラゾロ4,3−ジピリミジン類 Expired - Fee Related JP4015176B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0309780 2003-04-29
GBGB0327748.0A GB0327748D0 (en) 2003-11-28 2003-11-28 Novel pharmaceuticals
PCT/IB2004/001433 WO2004096810A1 (en) 2003-04-29 2004-04-22 5,7-diaminopyrazolo`4,3-d!pyrimidines useful in the treatment of hypertension

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2007067736A Division JP2007217419A (ja) 2003-04-29 2007-03-16 高血圧症の治療に有用な5,7−ジアミノピラゾロ4,3−ジピリミジン類

Publications (3)

Publication Number Publication Date
JP2006524636A JP2006524636A (ja) 2006-11-02
JP2006524636A5 true JP2006524636A5 (ja) 2007-09-27
JP4015176B2 JP4015176B2 (ja) 2007-11-28

Family

ID=33420887

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2006500346A Expired - Fee Related JP4015176B2 (ja) 2003-04-29 2004-04-22 高血圧症の治療に有用な5,7−ジアミノピラゾロ4,3−ジピリミジン類
JP2007067736A Pending JP2007217419A (ja) 2003-04-29 2007-03-16 高血圧症の治療に有用な5,7−ジアミノピラゾロ4,3−ジピリミジン類

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2007067736A Pending JP2007217419A (ja) 2003-04-29 2007-03-16 高血圧症の治療に有用な5,7−ジアミノピラゾロ4,3−ジピリミジン類

Country Status (32)

Country Link
US (2) US7262192B2 (ja)
EP (1) EP1620437B1 (ja)
JP (2) JP4015176B2 (ja)
KR (1) KR100824193B1 (ja)
AR (1) AR044116A1 (ja)
AT (1) ATE433978T1 (ja)
AU (1) AU2004234158B2 (ja)
BR (1) BRPI0409903A (ja)
CA (1) CA2523831C (ja)
CL (1) CL2004000889A1 (ja)
CO (1) CO5640118A2 (ja)
CR (1) CR8051A (ja)
DE (1) DE602004021585D1 (ja)
DK (1) DK1620437T3 (ja)
EA (1) EA008596B1 (ja)
EC (1) ECSP056130A (ja)
ES (1) ES2326119T3 (ja)
GE (1) GEP20084329B (ja)
HK (1) HK1087108A1 (ja)
IS (1) IS8009A (ja)
MA (1) MA27771A1 (ja)
MX (1) MXPA05011643A (ja)
NL (1) NL1026074C2 (ja)
NO (1) NO333850B1 (ja)
NZ (1) NZ542097A (ja)
OA (1) OA13050A (ja)
PA (1) PA8601701A1 (ja)
PE (1) PE20050462A1 (ja)
RS (1) RS20050810A (ja)
TW (1) TWI273908B (ja)
UY (1) UY28290A1 (ja)
WO (1) WO2004096810A1 (ja)

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