JP2006510609A5 - - Google Patents

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Publication number
JP2006510609A5
JP2006510609A5 JP2004546967A JP2004546967A JP2006510609A5 JP 2006510609 A5 JP2006510609 A5 JP 2006510609A5 JP 2004546967 A JP2004546967 A JP 2004546967A JP 2004546967 A JP2004546967 A JP 2004546967A JP 2006510609 A5 JP2006510609 A5 JP 2006510609A5
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JP
Japan
Prior art keywords
methanone
ylmethylphenyl
phenyl
isopropylpiperazin
dihydrochloride
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004546967A
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English (en)
Japanese (ja)
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JP2006510609A (ja
JP4596918B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2003/033343 external-priority patent/WO2004037801A1/en
Publication of JP2006510609A publication Critical patent/JP2006510609A/ja
Publication of JP2006510609A5 publication Critical patent/JP2006510609A5/ja
Application granted granted Critical
Publication of JP4596918B2 publication Critical patent/JP4596918B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2004546967A 2002-10-23 2003-10-21 ピペラジニルおよびジアザパニルベンズアミドおよびベンズチオアミド Expired - Fee Related JP4596918B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42049502P 2002-10-23 2002-10-23
PCT/US2003/033343 WO2004037801A1 (en) 2002-10-23 2003-10-21 Piperazinyl and diazapanyl benzamides and benzthioamides

Publications (3)

Publication Number Publication Date
JP2006510609A JP2006510609A (ja) 2006-03-30
JP2006510609A5 true JP2006510609A5 (https=) 2006-09-21
JP4596918B2 JP4596918B2 (ja) 2010-12-15

Family

ID=32176579

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004546967A Expired - Fee Related JP4596918B2 (ja) 2002-10-23 2003-10-21 ピペラジニルおよびジアザパニルベンズアミドおよびベンズチオアミド

Country Status (32)

Country Link
US (2) US7414047B2 (https=)
EP (1) EP1558595B1 (https=)
JP (1) JP4596918B2 (https=)
KR (1) KR101067732B1 (https=)
CN (1) CN100558718C (https=)
AR (1) AR041697A1 (https=)
AT (1) ATE449766T1 (https=)
AU (1) AU2003301552B2 (https=)
BR (1) BRPI0315644B8 (https=)
CA (1) CA2504269C (https=)
CR (1) CR7807A (https=)
CY (1) CY1109924T1 (https=)
DE (1) DE60330269D1 (https=)
DK (1) DK1558595T3 (https=)
EA (1) EA009860B1 (https=)
EG (1) EG25097A (https=)
ES (1) ES2335584T3 (https=)
HR (1) HRP20050352B1 (https=)
IL (1) IL168207A (https=)
ME (1) ME00334B (https=)
MX (2) MX339074B (https=)
MY (1) MY140886A (https=)
NO (1) NO330741B1 (https=)
NZ (2) NZ576432A (https=)
PL (1) PL215454B1 (https=)
PT (1) PT1558595E (https=)
RS (1) RS51681B (https=)
SI (1) SI1558595T1 (https=)
TW (1) TWI352594B (https=)
UA (1) UA80573C2 (https=)
WO (1) WO2004037801A1 (https=)
ZA (1) ZA200504067B (https=)

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EP1558595B1 (en) 2002-10-23 2009-11-25 Janssen Pharmaceutica N.V. Piperazinyl and diazapanyl benzamides and benzthioamides
GB0324159D0 (en) 2003-10-15 2003-11-19 Glaxo Group Ltd Novel compounds
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US7423147B2 (en) * 2004-03-31 2008-09-09 Janssen Pharmaceutical, N.V. Pyridine compounds as histamine H3 modulators
SI1948607T1 (sl) * 2005-09-16 2010-07-30 Janssen Pharmaceutica Nv Ciklopropil amini kot modulatorji histaminskega H3 receptorja
US7795426B2 (en) 2005-10-31 2010-09-14 Janssen Pharmaceutica Nv Processes for the preparation of cyclopropyl-amide derivatives
EP2404911A1 (en) 2005-10-31 2012-01-11 Janssen Pharmaceutica NV Novel processes for the preparation of piperazinyl and diazapanyl benzamide derivatives
EP1951699B1 (en) * 2005-10-31 2012-10-10 Janssen Pharmaceutica NV Processes for the preparation of cyclopropyl-amide derivatives
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WO2007143422A2 (en) * 2006-05-30 2007-12-13 Janssen Pharmaceutica N.V. Substituted pyridyl amide compounds as modulators of the histamine h3 receptor
BRPI0712823A2 (pt) 2006-06-23 2012-07-24 Abbott Lab derivados de ciclopropil amina como moduladores de receptor de histamina h3
US9108948B2 (en) 2006-06-23 2015-08-18 Abbvie Inc. Cyclopropyl amine derivatives
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SI2121636T1 (sl) 2006-12-14 2017-06-30 Janssen Pharmaceutica N.V. Postopek za pripravo derivatov piperazinila in diazepanil benzamida
US8288389B2 (en) 2007-09-06 2012-10-16 Glaxo Group Limited Piperazine derivative having affinity for the histamine H3 receptor
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US20100130477A1 (en) * 2008-11-25 2010-05-27 Astrazeneca Ab Spirocyclobutyl Piperidine Derivatives
DK2429996T3 (en) * 2009-03-18 2017-06-19 Janssen Pharmaceutica Nv Process for the preparation of histamine h3 receptor modulators
US9186353B2 (en) 2009-04-27 2015-11-17 Abbvie Inc. Treatment of osteoarthritis pain
WO2012037258A1 (en) 2010-09-16 2012-03-22 Abbott Laboratories Processes for preparing 1,2-substituted cyclopropyl derivatives
RU2700595C1 (ru) * 2019-07-30 2019-09-18 Общество с ограниченной ответственностью "Кью Эм Фарма" Производное 3,6,9-триазатрициклотетрадекана и его применение для лечения депрессии
WO2022113008A1 (en) 2020-11-27 2022-06-02 Richter Gedeon Nyrt. Histamine h3 receptor antagonists/inverse agonists for the treatment of autism spectrum disorder

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GB0324159D0 (en) 2003-10-15 2003-11-19 Glaxo Group Ltd Novel compounds

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