JP2006510609A5 - - Google Patents

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Publication number
JP2006510609A5
JP2006510609A5 JP2004546967A JP2004546967A JP2006510609A5 JP 2006510609 A5 JP2006510609 A5 JP 2006510609A5 JP 2004546967 A JP2004546967 A JP 2004546967A JP 2004546967 A JP2004546967 A JP 2004546967A JP 2006510609 A5 JP2006510609 A5 JP 2006510609A5
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JP
Japan
Prior art keywords
methanone
ylmethylphenyl
phenyl
isopropylpiperazin
dihydrochloride
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004546967A
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English (en)
Japanese (ja)
Other versions
JP4596918B2 (ja
JP2006510609A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2003/033343 external-priority patent/WO2004037801A1/en
Publication of JP2006510609A publication Critical patent/JP2006510609A/ja
Publication of JP2006510609A5 publication Critical patent/JP2006510609A5/ja
Application granted granted Critical
Publication of JP4596918B2 publication Critical patent/JP4596918B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2004546967A 2002-10-23 2003-10-21 ピペラジニルおよびジアザパニルベンズアミドおよびベンズチオアミド Expired - Fee Related JP4596918B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42049502P 2002-10-23 2002-10-23
PCT/US2003/033343 WO2004037801A1 (en) 2002-10-23 2003-10-21 Piperazinyl and diazapanyl benzamides and benzthioamides

Publications (3)

Publication Number Publication Date
JP2006510609A JP2006510609A (ja) 2006-03-30
JP2006510609A5 true JP2006510609A5 (https=) 2006-09-21
JP4596918B2 JP4596918B2 (ja) 2010-12-15

Family

ID=32176579

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004546967A Expired - Fee Related JP4596918B2 (ja) 2002-10-23 2003-10-21 ピペラジニルおよびジアザパニルベンズアミドおよびベンズチオアミド

Country Status (32)

Country Link
US (2) US7414047B2 (https=)
EP (1) EP1558595B1 (https=)
JP (1) JP4596918B2 (https=)
KR (1) KR101067732B1 (https=)
CN (1) CN100558718C (https=)
AR (1) AR041697A1 (https=)
AT (1) ATE449766T1 (https=)
AU (1) AU2003301552B2 (https=)
BR (1) BRPI0315644B8 (https=)
CA (1) CA2504269C (https=)
CR (1) CR7807A (https=)
CY (1) CY1109924T1 (https=)
DE (1) DE60330269D1 (https=)
DK (1) DK1558595T3 (https=)
EA (1) EA009860B1 (https=)
EG (1) EG25097A (https=)
ES (1) ES2335584T3 (https=)
HR (1) HRP20050352B1 (https=)
IL (1) IL168207A (https=)
ME (1) ME00334B (https=)
MX (2) MXPA05004384A (https=)
MY (1) MY140886A (https=)
NO (1) NO330741B1 (https=)
NZ (2) NZ539595A (https=)
PL (1) PL215454B1 (https=)
PT (1) PT1558595E (https=)
RS (1) RS51681B (https=)
SI (1) SI1558595T1 (https=)
TW (1) TWI352594B (https=)
UA (1) UA80573C2 (https=)
WO (1) WO2004037801A1 (https=)
ZA (1) ZA200504067B (https=)

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SI1558595T1 (sl) 2002-10-23 2010-03-31 Janssen Pharmaceutica Nv Piperazinilni in diazapanilni benzamidi in benztioamidi
GB0324159D0 (en) 2003-10-15 2003-11-19 Glaxo Group Ltd Novel compounds
AU2005230902A1 (en) * 2004-03-31 2005-10-20 Janssen Pharmaceutica, N.V. Non-imidazole heterocyclic compounds as histamine H3-receptor ligands
DE602005025222D1 (de) 2004-03-31 2011-01-20 Janssen Pharmaceutica Nv Heterocyclische nichtimidazolverbindungen als modulatoren des histamin-h3-rezeptors
KR101336106B1 (ko) * 2005-09-16 2013-12-05 얀센 파마슈티카 엔.브이. 히스타민 ｈ3 수용체의 조절제로서 사이클로프로필 아민
US7728129B2 (en) * 2005-10-31 2010-06-01 Janssen Pharmaceutica Nv Processes for the preparation of piperazinyl and diazapanyl benzamide derivatives
MX367916B (es) * 2005-10-31 2019-09-11 Janssen Pharmaceutica N V Star Procedimientos para la preparacion de derivados de ciclopropilamida.
US7795426B2 (en) * 2005-10-31 2010-09-14 Janssen Pharmaceutica Nv Processes for the preparation of cyclopropyl-amide derivatives
US8158791B2 (en) * 2005-11-10 2012-04-17 Msd K.K. Aza-substituted spiro derivatives
EA015555B1 (ru) * 2006-05-30 2011-08-30 Янссен Фармацевтика Н.В. Замещенные пиридиламидные соединения в качестве модуляторов гистаминового h-рецептора
CN103382174A (zh) 2006-06-23 2013-11-06 雅培制药有限公司 作为组胺h3受体调节物的环丙胺衍生物
US9108948B2 (en) 2006-06-23 2015-08-18 Abbvie Inc. Cyclopropyl amine derivatives
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HRP20170621T1 (hr) * 2006-12-14 2017-07-28 Janssen Pharmaceutica N.V. Postupak za pripremanje derivata piperazinil i diazepanil benzamida
TW200918527A (en) * 2007-09-06 2009-05-01 Glaxo Group Ltd Piperazine derivative having affinity for the histamine H3 receptor
AR068509A1 (es) * 2007-09-19 2009-11-18 Jerini Ag Antagosnistas del receptor de bradiquinina b1
EA018582B1 (ru) 2007-11-20 2013-09-30 Янссен Фармацевтика Н.В. Соединения циклоалкилокси- и гетероциклоалкилоксипиридина как модуляторы гистаминового рецептора н
US20100130477A1 (en) * 2008-11-25 2010-05-27 Astrazeneca Ab Spirocyclobutyl Piperidine Derivatives
PT3216784T (pt) * 2009-03-18 2019-04-01 Janssen Pharmaceutica Nv Processo para a preparação de moduladores do recetor h3 de histamina
US9186353B2 (en) 2009-04-27 2015-11-17 Abbvie Inc. Treatment of osteoarthritis pain
US8853390B2 (en) 2010-09-16 2014-10-07 Abbvie Inc. Processes for preparing 1,2-substituted cyclopropyl derivatives
RU2700595C1 (ru) * 2019-07-30 2019-09-18 Общество с ограниченной ответственностью "Кью Эм Фарма" Производное 3,6,9-триазатрициклотетрадекана и его применение для лечения депрессии
WO2022113008A1 (en) 2020-11-27 2022-06-02 Richter Gedeon Nyrt. Histamine h3 receptor antagonists/inverse agonists for the treatment of autism spectrum disorder

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