ATE354568T1 - Nicht-imidazol aryloxypiperidine als h3 rezeptor liganden - Google Patents
Nicht-imidazol aryloxypiperidine als h3 rezeptor ligandenInfo
- Publication number
- ATE354568T1 ATE354568T1 AT01959582T AT01959582T ATE354568T1 AT E354568 T1 ATE354568 T1 AT E354568T1 AT 01959582 T AT01959582 T AT 01959582T AT 01959582 T AT01959582 T AT 01959582T AT E354568 T1 ATE354568 T1 AT E354568T1
- Authority
- AT
- Austria
- Prior art keywords
- aryloxypiperidine
- imidazole
- receptor ligands
- treat
- compounds
- Prior art date
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4402—Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 2, e.g. pheniramine, bisacodyl
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4465—Non condensed piperidines, e.g. piperocaine only substituted in position 4
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AT01959582T ATE354568T1 (de) | 2000-08-08 | 2001-08-06 | Nicht-imidazol aryloxypiperidine als h3 rezeptor liganden |
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EP (1) | EP1311482B1 (de) |
JP (1) | JP2004511438A (de) |
KR (1) | KR100852362B1 (de) |
CN (1) | CN100396668C (de) |
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-
2001
- 2001-08-06 PT PT01959582T patent/PT1311482E/pt unknown
- 2001-08-06 US US09/922,619 patent/US7071191B2/en not_active Expired - Lifetime
- 2001-08-06 AU AU8112101A patent/AU8112101A/xx active Pending
- 2001-08-06 DE DE60126785T patent/DE60126785T2/de not_active Expired - Fee Related
- 2001-08-06 ES ES01959582T patent/ES2282279T3/es not_active Expired - Lifetime
- 2001-08-06 PL PL01360373A patent/PL360373A1/xx not_active IP Right Cessation
- 2001-08-06 CA CA002419036A patent/CA2419036A1/en not_active Abandoned
- 2001-08-06 DK DK01959582T patent/DK1311482T3/da active
- 2001-08-06 AU AU2001281121A patent/AU2001281121B2/en not_active Expired
- 2001-08-06 CN CNB018167020A patent/CN100396668C/zh not_active Expired - Fee Related
- 2001-08-06 AT AT01959582T patent/ATE354568T1/de not_active IP Right Cessation
- 2001-08-06 EP EP01959582A patent/EP1311482B1/de not_active Expired - Lifetime
- 2001-08-06 WO PCT/US2001/024660 patent/WO2002012190A2/en active IP Right Grant
- 2001-08-06 BR BR0113161-3A patent/BR0113161A/pt not_active IP Right Cessation
- 2001-08-06 MX MXPA03001268A patent/MXPA03001268A/es active IP Right Grant
- 2001-08-06 JP JP2002518168A patent/JP2004511438A/ja active Pending
- 2001-08-06 CZ CZ2003686A patent/CZ2003686A3/cs unknown
- 2001-08-06 KR KR1020037001879A patent/KR100852362B1/ko not_active IP Right Cessation
- 2001-08-06 HU HU0302893A patent/HUP0302893A3/hu unknown
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Also Published As
Publication number | Publication date |
---|---|
KR100852362B1 (ko) | 2008-08-14 |
EP1311482B1 (de) | 2007-02-21 |
ES2282279T3 (es) | 2007-10-16 |
MXPA03001268A (es) | 2004-09-06 |
JP2004511438A (ja) | 2004-04-15 |
BR0113161A (pt) | 2004-04-06 |
US7071191B2 (en) | 2006-07-04 |
AU2001281121B2 (en) | 2007-08-23 |
HUP0302893A3 (en) | 2006-04-28 |
WO2002012190A2 (en) | 2002-02-14 |
PT1311482E (pt) | 2007-04-30 |
CZ2003686A3 (cs) | 2003-08-13 |
US7241778B2 (en) | 2007-07-10 |
US20020040024A1 (en) | 2002-04-04 |
CN100396668C (zh) | 2008-06-25 |
WO2002012190A3 (en) | 2002-08-01 |
US20050227979A1 (en) | 2005-10-13 |
CA2419036A1 (en) | 2002-02-14 |
DE60126785D1 (de) | 2007-04-05 |
EP1311482A2 (de) | 2003-05-21 |
PL360373A1 (en) | 2004-09-06 |
HUP0302893A2 (hu) | 2003-12-29 |
DK1311482T3 (da) | 2007-05-07 |
DE60126785T2 (de) | 2007-10-25 |
CN1468221A (zh) | 2004-01-14 |
KR20030048007A (ko) | 2003-06-18 |
AU8112101A (en) | 2002-02-18 |
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